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CAS No.: 2220184-50-7

CDK12-IN-3 Catalog No. CSN22379

Synonyms: AZ-1992;Compound 7;Cmpd 7

CMPD 7 is a potent and selective CDK12 inhibitor with an IC50 of 491 nM in enzymatic assay.

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  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
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    NCT00101296Acute Myeloid Leukemia With Mu... more >>ltilineage Dysplasia Following Myelodysplastic Syndrome Adult Acute Erythroid Leukemia (M6) Adult Acute Megakaryoblastic Leukemia (M7) Adult Acute Minimally Differentiated Myeloid Leukemia (M0) Adult Acute Monoblastic Leukemia (M5a) Adult Acute Monoblastic Leukemia and Acute Monocytic Leukemia (M5) Adult Acute Monocytic Leukemia (M5b) Adult Acute Myeloblastic Leukemia With Maturation (M2) Adult Acute Myeloblastic Leukemia Without Maturation (M1) Adult Acute Myeloid Leukemia With 11q23 (MLL) Abnormalities Adult Acute Myeloid Leukemia With Del(5q) Adult Acute Myeloid Leukemia With Inv(16)(p13;q22) Adult Acute Myeloid Leukemia With t(16;16)(p13;q22) Adult Acute Myeloid Leukemia With t(8;21)(q22;q22) Adult Acute Myelomonocytic Leukemia (M4) Adult Erythroleukemia (M6a) Adult Pure Erythroid Leukemia (M6b) Recurrent Adult Acute Myeloid Leukemia Untreated Adult Acute Myeloid Leukemia Collapse <<Phase 1Completed-United States, California ... more >> City of Hope Duarte, California, United States, 91010 Collapse <<
    NCT00710892Acute Lymphoblastic Leukemia ... more >> Non-Hodgkin's Lymphoma Myelodysplastic Syndrome Chronic Myeloid Leukemia Collapse <<Phase 1Active, not recruitingJuly 2026United States, Texas ... more >> Texas Children's Hospital Houston, Texas, United States, 77030 The Methodist Hospital Houston, Texas, United States, 77030 Collapse <<
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技术信息

CAS号 2220184-50-7 储存条件
分子式 C23H28F2N8O 运输 蓝冰
分子量 470.52 别名 AZ-1992;Compound 7;Cmpd 7

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