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CAS No.: 1439934-41-4
CTX-0294885 is a bisanilino pyrimidine and exhibits inhibitory activity against a broad range of kinases in vitro, further developed into a Sepharose-supported kinase capture reagent. CTX-0294885 is a broad spectrum kinase inhibitor that inhibited FAK, FLT3, JAK2, JAK3, Src, Aurora kinase A, and VEGF receptor 3 (IC50s = 4, 1, 3, 28, 2, 18, and 3 nM, respectively) in an initial screen.
生物活性
实验方案
技术信息
CAS号 | 1439934-41-4 | 储存条件 |
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分子式 | C22H24ClN7O | 运输 | 蓝冰 | |||
分子量 | 437.93 | 别名 | ||||
溶解度 |
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动物实验配方 |
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