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CAS No.: 1443763-60-7
Synonyms: BAY 1161909;Mps1-IN-5
BAY 1161909 inhibits Mps1 kinase activity with IC50 of < 1 nM when assay with 10 μM ATP, with IC50 of < 1.9 nM when assay with 2 mM ATP.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02138812 | Medical Oncology | Phase 1 | Terminated(As another Mps1 inh... more >>ibitor was being developed in parallel, the strategic decision was to move forward with the development of the follow up compound only.) Collapse << | - | United States, California ... more >> Santa Monica, California, United States, 90403 United States, Connecticut New Haven, Connecticut, United States, 06510 United States, Massachusetts Boston, Massachusetts, United States, 02215 United States, Michigan Detroit, Michigan, United States, 48201 United States, Tennessee Nashville, Tennessee, United States, 37203 United States, Texas San Antonio, Texas, United States, 78229 Collapse << |
实验方案
技术信息
CAS号 | 1443763-60-7 | 储存条件 |
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分子式 | C29H26FN5O4S | 运输 | 蓝冰 | |||||||
分子量 | 559.61 | 别名 | BAY 1161909;Mps1-IN-5 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02138812 | Medical Oncology | Phase 1 | Terminated(As another Mps1 inh... more >>ibitor was being developed in parallel, the strategic decision was to move forward with the development of the follow up compound only.) Collapse << | - | United States, California ... more >> Santa Monica, California, United States, 90403 United States, Connecticut New Haven, Connecticut, United States, 06510 United States, Massachusetts Boston, Massachusetts, United States, 02215 United States, Michigan Detroit, Michigan, United States, 48201 United States, Tennessee Nashville, Tennessee, United States, 37203 United States, Texas San Antonio, Texas, United States, 78229 Collapse << |
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