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CAS No.: 159351-69-6

Everolimus/依维莫司 Catalog No. CSN16716

Synonyms: RAD001;SDZ-RAD;RAD 001.SDZ-RAD

Everolimus is a mTOR inhibitor of FKBP12 with IC50 of 1.6-2.4 nM.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 靶点FKBP12

    IC50:1.6-2.4nM
  • 描述
  • 细胞研究
  • Cell Data
  • 更多
  • 动物研究
    剂量

    Nude Mice: 0.05 mg/kg - 15 mg/kg[2] (p.o.)

    给药途径

    p.o.

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02812940Graft-versus-Host DiseasePhase 2RecruitingJune 2019Germany ... more >> University of Cologne Recruiting Cologne, Germany, 50924 Contact: Christoph Scheid, MD PhD    49221478 ext 6296    c.scheid@uni-koeln.de    Sub-Investigator: Udo Holtick, MD Collapse <<
    NCT02008019ChondrosarcomaPhase 2Suspended(The study was suspen... more >>ded since july 27th 2016 because of unavailability of Everolimus) Collapse <<August 2019France ... more >> Institut Bergonié Bordeaux, Gironde, France, 33076 Institut Claudius Regaud Toulouse, Haute Garonne, France, 31052 Centre Hospitalier Universitaire de Limoges, Hôpital Dupuytren Limoges, Haute Vienne, France, 87042 Institut Régional du Cancer de Montpellier Montpellier, Hérault, France, 34298 Centre Hospitalier Régional Universitaire de Tours, Hôpital Trousseau Tours, Indre et Loire, France, 37044 Centre Hospitalier Universitaire de Nantes, Hôtel Dieu Nantes, Loire Atlantique, France, 44093 Institut de Cancérologie de l'Ouest - René Gauducheau Saint-Herblain, Loire Atlantique, France, 44805 Institut de Cancérologie de Lorraine Vandoeuvre-les-Nancy, Meurthe et Moselle, France, 54511 Centre Oscar Lambret Lille, Nord, France, 59000 CHRU de Lille - Hôpital Roger Salengro Lille, Nord, France, 59037 Centre Léon Bérard Lyon, Rhône, France, 69373 Institut Gustave Roussy Villejuif, Val de Marne, France, 94805 Collapse <<
    NCT02025712Hormone Receptor Positive Mali... more >>gnant Neoplasm of Breast Collapse <<Phase 2Unknown-China ... more >> Unimed Medical Institute Not yet recruiting Hong Kong, China Contact: Louis Chow    (852)28610286       Principal Investigator: Louis Chow Collapse <<
  • 更多
  • 参考文献

实验方案

技术信息

CAS号 159351-69-6 储存条件
分子式 C53H83NO14 运输 蓝冰
分子量 958.22 别名 RAD001;SDZ-RAD;RAD 001.SDZ-RAD;Brand name Afinitor;Zortress;Certican;Xience V;依维莫司
溶解度
DMSO360.0 mg/mL (375.7 mM) warming
Waterinsoluble
动物实验配方
IP2% DMSO+2% Tween80+40% PEG300+water3.6 mg/mLclear
PO0.5% CMC-Na32 mg/mLsuspension

大规格询价

号为必填项

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