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CAS No.: 905281-76-7
Synonyms: AR-00341677
GDC-0879 is a potent, and selective B-Raf inhibitor with IC50 of 0.13 nM with activity against c-Raf as well, displaying no inhibition known to other protein kinases.
生物活性
实验方案
技术信息
CAS号 | 905281-76-7 | 储存条件 |
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分子式 | C19H18N4O2 | 运输 | 蓝冰 | |
分子量 | 334.37 | 别名 | AR-00341677 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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human A375 cells | - | Proliferation assay | - | Antiproliferative activity against human A375 cells expressing B-Raf V600E mutant and wild type Ras, IC50=0.5 μM | 22808911 |
human A375 cells | - | Function assay | - | Inhibition of b-Raf in human A375 cells assessed phosphorylation of ERK, IC50=1 μM | 22808911 |
human MALME3M cells | - | Function assay | - | Inhibition of ERK1/2 phosphorylation in human MALME3M cells, IC50=0.063 μM | 11717001 |
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