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CAS No.: 415903-37-6
Synonyms: CJ-023423;RQ-00000007;AAT-007
Grapiprant is a selective EP4 receptor antagonist whose physiological ligand is prostaglandin E2 (PGE2).
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03658772 | Microsatellite Stable Colorect... more >>al Cancer Collapse << | Phase 1 | Recruiting | August 2020 | United States, Arizona ... more >> Mayo Clinic Cancer Center - Scottsdale Not yet recruiting Phoenix, Arizona, United States, 85054 Contact: Mayo Clinical Trials Office 855-776-0015 United States, Colorado University of Colorado Denver-Anschutz Medical Campus Not yet recruiting Aurora, Colorado, United States, 80045 Contact: Elizabeth Freas elizabeth.freas@ucdenver.edu United States, Tennessee Sarah Cannon Research Institute, LLC (SCRI) Recruiting Nashville, Tennessee, United States, 37203 Contact: Lisa Morris Lisa.MorrisLaperriere@SarahCannon.com United States, Texas New Experimental Therapeutics of San Antonio-NEXT Oncology Recruiting San Antonio, Texas, United States, 78240 Contact: Sarah Gomez sgomez@nextsat.com Collapse << |
NCT03696212 | Non-small Cell Lung Cancer Ade... more >>nocarcinoma Collapse << | Phase 1 Phase 2 | Not yet recruiting | September 2020 | United States, California ... more >> Stanford University Medical Center Not yet recruiting Stanford, California, United States, 94305 Contact: Melanie San Pedro 650-724-1388 msanpedro@stanford.edu United States, Michigan Barbara Ann Karmanos Cancer Institute Not yet recruiting Detroit, Michigan, United States, 48201 Contact: Amanda Newman 313-576-8411 newmana@karmanos.org United States, Pennsylvania University of Pennsylvania Abramson Cancer Center Not yet recruiting Philadelphia, Pennsylvania, United States, 19104 Contact: Melissa Volpe 215-220-9703 Melisssa.volpe@uphs.upenn.edu Fox Chase Cancer Center Not yet recruiting Philadelphia, Pennsylvania, United States, 19111 United States, Virginia Virginia Cancer Specialists Not yet recruiting Fairfax, Virginia, United States, 22031 Collapse << |
实验方案
技术信息
CAS号 | 415903-37-6 | 储存条件 |
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分子式 | C26H29N5O3S | 运输 | 蓝冰 | |||
分子量 | 491.61 | 别名 | CJ-023423;RQ-00000007;AAT-007;CAS#415903-37-6 | |||
溶解度 |
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动物实验配方 |