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CAS No.: 2079896-25-4
GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4±0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00175565 | Chronic Obstructive Pulmonary ... more >>Disease Emphysema Chronic Bronchitis Collapse << | Phase 4 | Completed | - | Canada, Alberta ... more >> University of Alberta Edmonton, Alberta, Canada, T6G 2R7 Canada, British Columbia University of British Columbia Vancouver, British Columbia, Canada, V6Z 1Y7 Collapse << |
实验方案
技术信息
CAS号 | 2079896-25-4 | 储存条件 |
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分子式 | C17H21BrN4O | 运输 | 蓝冰 | |
分子量 | 377.28 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00175565 | Chronic Obstructive Pulmonary ... more >>Disease Emphysema Chronic Bronchitis Collapse << | Phase 4 | Completed | - | Canada, Alberta ... more >> University of Alberta Edmonton, Alberta, Canada, T6G 2R7 Canada, British Columbia University of British Columbia Vancouver, British Columbia, Canada, V6Z 1Y7 Collapse << |
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