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CAS No.: 1088965-37-0
Synonyms: GSK923295A
GSK923295 is a specific allosteric CENP-E inhibito with Ki value of 3.2 nM.
生物活性
靶点 | CENPE Ki:3.2nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00504790 | Cancer | Phase 1 | Completed | - | United States, California ... more >> GSK Investigational Site Duarte, California, United States, 91010 United States, Michigan GSK Investigational Site Detroit, Michigan, United States, 48201 United States, Wisconsin GSK Investigational Site Madison, Wisconsin, United States, 53792-5666 Collapse << |
实验方案
技术信息
CAS号 | 1088965-37-0 | 储存条件 |
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分子式 | C32H38ClN5O4 | 运输 | 蓝冰 | |||||||
分子量 | 592.13 | 别名 | GSK923295A | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00504790 | Cancer | Phase 1 | Completed | - | United States, California ... more >> GSK Investigational Site Duarte, California, United States, 91010 United States, Michigan GSK Investigational Site Detroit, Michigan, United States, 48201 United States, Wisconsin GSK Investigational Site Madison, Wisconsin, United States, 53792-5666 Collapse << |
靶点 | Description | IC50 |
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CENPE | Ki:3.2nM |
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