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CAS No.: 1034688-30-6

GSK2018682 Catalog No. CSN21216

Synonyms: 2018682

GSK-2018682 is a sphingosine 1 phosphate receptor (S1PR)-1 agonist potentially for the treatment of multiple sclerosis. GSK-2018682 induced acute, transient and non-symptomatic decreases in heart rate and blood pressure.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT01431937Multiple Sclerosis, Relapsing-... more >>Remitting Collapse <<Phase 1Completed-Australia, New South Wales ... more >> GSK Investigational Site Randwick, New South Wales, Australia, 2031 Australia, South Australia GSK Investigational Site Adelaide, South Australia, Australia, 5000 Australia, Western Australia GSK Investigational Site Nedlands, Western Australia, Australia, 6009 Collapse <<
    NCT01387217Multiple SclerosisPhase 1Completed-Australia, New South Wales ... more >> GSK Investigational Site Randwick, New South Wales, Australia, 2031 Australia, South Australia GSK Investigational Site Adelaide, South Australia, Australia, 5000 Collapse <<
    NCT01466322Multiple Sclerosis, Relapsing-... more >>Remitting Collapse <<Phase 1Completed-Australia, Queensland ... more >> GSK Investigational Site Herston, Queensland, Australia, 4006 Collapse <<

实验方案

技术信息

CAS号 1034688-30-6 储存条件
分子式 C22H21ClN4O4 运输 蓝冰
分子量 440.88 别名 2018682
溶解度
DMSO125.0 mg/mL (283.5 mM)
WaterInsoluble
动物实验配方

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