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CAS No.: 503468-95-9
Synonyms: NU7441;Ku-57788
NU7441 is a potent and selective DNA-PK inhibitor with IC50 of 14 nM and also inhibits PI3K with IC50 of 5 μM in cell-free assays.
生物活性
靶点 | DNA-PK IC50:14nM | PI3K IC50:5μM |
实验方案
技术信息
CAS号 | 503468-95-9 | 储存条件 |
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分子式 | C25H19NO3S | 运输 | 蓝冰 | |||||||||||||
分子量 | 413.49 | 别名 | NU7441;Ku-57788 | |||||||||||||
溶解度 |
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动物实验配方 |
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Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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23132-87 | - | Growth Inhibition Assay | - | IC50=5.32024 μM | SANGER |
639-V | - | Growth Inhibition Assay | - | IC50=1.44128 μM | SANGER |
647-V | - | Growth Inhibition Assay | - | IC50=15.2705 μM | SANGER |
697 | - | Growth Inhibition Assay | - | IC50=3.44993 μM | SANGER |
786-0 | - | Growth Inhibition Assay | - | IC50=7.09786 μM | SANGER |
8305C | - | Growth Inhibition Assay | - | IC50=3.61736 μM | SANGER |
8505C | - | Growth Inhibition Assay | - | IC50=25.1845 μM | SANGER |
8-MG-BA | - | Growth Inhibition Assay | - | IC50=13.7513 μM | SANGER |
A101D | - | Growth Inhibition Assay | - | IC50=2.61338 μM | SANGER |
A172 | - | Growth Inhibition Assay | - | IC50=0.15316 μM | SANGER |
A204 | - | Growth Inhibition Assay | - | IC50=18.5452 μM | SANGER |
A2058 | - | Growth Inhibition Assay | - | IC50=10.6404 μM | SANGER |
A253 | - | Growth Inhibition Assay | - | IC50=21.4481 μM | SANGER |
A427 | - | Growth Inhibition Assay | - | IC50=5.53661 μM | SANGER |
A431 | - | Growth Inhibition Assay | - | IC50=39.1894 μM | SANGER |
A549 | - | Growth Inhibition Assay | - | IC50=9.09612 μM | SANGER |
A704 | - | Growth Inhibition Assay | - | IC50=4.40888 μM | SANGER |
ACN | - | Growth Inhibition Assay | - | IC50=7.7433 μM | SANGER |
AGS | - | Growth Inhibition Assay | - | IC50=14.1319 μM | SANGER |
ALL-PO | - | Growth Inhibition Assay | - | IC50=49.9268 μM | SANGER |
AM-38 | - | Growth Inhibition Assay | - | IC50=30.0606 μM | SANGER |
AN3-CA | - | Growth Inhibition Assay | - | IC50=4.25813 μM | SANGER |
AsPC-1 | - | Growth Inhibition Assay | - | IC50=30.8053 μM | SANGER |
AU565 | - | Growth Inhibition Assay | - | IC50=7.59833 μM | SANGER |
BALL-1 | - | Growth Inhibition Assay | - | IC50=12.2662 μM | SANGER |
BB30-HNC | - | Growth Inhibition Assay | - | IC50=25.2483 μM | SANGER |
BB49-HNC | - | Growth Inhibition Assay | - | IC50=10.8586 μM | SANGER |
BB65-RCC | - | Growth Inhibition Assay | - | IC50=23.7863 μM | SANGER |
BCPAP | - | Growth Inhibition Assay | - | IC50=22.611 μM | SANGER |
BE-13 | - | Growth Inhibition Assay | - | IC50=21.6113 μM | SANGER |
Becker | - | Growth Inhibition Assay | - | IC50=13.058 μM | SANGER |
BFTC-905 | - | Growth Inhibition Assay | - | IC50=2.16687 μM | SANGER |
BFTC-909 | - | Growth Inhibition Assay | - | IC50=14.5055 μM | SANGER |
BHT-101 | - | Growth Inhibition Assay | - | IC50=3.59985 μM | SANGER |
BHY | - | Growth Inhibition Assay | - | IC50=32.9495 μM | SANGER |
BPH-1 | - | Growth Inhibition Assay | - | IC50=10.7145 μM | SANGER |
BT-549 | - | Growth Inhibition Assay | - | IC50=48.3729 μM | SANGER |
C32 | - | Growth Inhibition Assay | - | IC50=10.8347 μM | SANGER |
C-33-A | - | Growth Inhibition Assay | - | IC50=32.7728 μM | SANGER |
Ca9-22 | - | Growth Inhibition Assay | - | IC50=29.4299 μM | SANGER |
CAKI-1 | - | Growth Inhibition Assay | - | IC50=9.1661 μM | SANGER |
CAL-12T | - | Growth Inhibition Assay | - | IC50=7.94352 μM | SANGER |
CAL-27 | - | Growth Inhibition Assay | - | IC50=14.0727 μM | SANGER |
CAL-51 | - | Growth Inhibition Assay | - | IC50=4.24854 μM | SANGER |
CAL-54 | - | Growth Inhibition Assay | - | IC50=11.4811 μM | SANGER |
CAL-62 | - | Growth Inhibition Assay | - | IC50=47.4068 μM | SANGER |
CAL-72 | - | Growth Inhibition Assay | - | IC50=10.8094 μM | SANGER |
CAPAN-1 | - | Growth Inhibition Assay | - | IC50=7.24359 μM | SANGER |
CaR-1 | - | Growth Inhibition Assay | - | IC50=28.5582 μM | SANGER |
CAS-1 | - | Growth Inhibition Assay | - | IC50=44.0991 μM | SANGER |
CGTH-W-1 | - | Growth Inhibition Assay | - | IC50=23.0641 μM | SANGER |
ChaGo-K-1 | - | Growth Inhibition Assay | - | IC50=5.56599 μM | SANGER |
CHL-1 | - | Growth Inhibition Assay | - | IC50=1.21368 μM | SANGER |
CHP-134 | - | Growth Inhibition Assay | - | IC50=8.24185 μM | SANGER |
CHP-212 | - | Growth Inhibition Assay | - | IC50=28.7401 μM | SANGER |
COLO-320-HSR | - | Growth Inhibition Assay | - | IC50=25.2208 μM | SANGER |
COLO-679 | - | Growth Inhibition Assay | - | IC50=11.946 μM | SANGER |
COLO-684 | - | Growth Inhibition Assay | - | IC50=11.7267 μM | SANGER |
CP50-MEL-B | - | Growth Inhibition Assay | - | IC50=13.6232 μM | SANGER |
CP66-MEL | - | Growth Inhibition Assay | - | IC50=48.0704 μM | SANGER |
CTB-1 | - | Growth Inhibition Assay | - | IC50=1.11546 μM | SANGER |
CW-2 | - | Growth Inhibition Assay | - | IC50=21.2705 μM | SANGER |
D-263MG | - | Growth Inhibition Assay | - | IC50=6.91068 μM | SANGER |
D-283MED | - | Growth Inhibition Assay | - | IC50=12.0569 μM | SANGER |
D-336MG | - | Growth Inhibition Assay | - | IC50=19.9322 μM | SANGER |
D-392MG | - | Growth Inhibition Assay | - | IC50=37.3344 μM | SANGER |
D-423MG | - | Growth Inhibition Assay | - | IC50=1.69361 μM | SANGER |
D-542MG | - | Growth Inhibition Assay | - | IC50=21.9069 μM | SANGER |
D-566MG | - | Growth Inhibition Assay | - | IC50=14.7706 μM | SANGER |
Daoy | - | Growth Inhibition Assay | - | IC50=32.0838 μM | SANGER |
DB | - | Growth Inhibition Assay | - | IC50=24.1028 μM | SANGER |
DBTRG-05MG | - | Growth Inhibition Assay | - | IC50=3.28085 μM | SANGER |
DEL | - | Growth Inhibition Assay | - | IC50=2.35564 μM | SANGER |
Detroit562 | - | Growth Inhibition Assay | - | IC50=33.6657 μM | SANGER |
DK-MG | - | Growth Inhibition Assay | - | IC50=27.1817 μM | SANGER |
DMS-114 | - | Growth Inhibition Assay | - | IC50=15.3291 μM | SANGER |
DU-4475 | - | Growth Inhibition Assay | - | IC50=9.96939 μM | SANGER |
EFO-27 | - | Growth Inhibition Assay | - | IC50=4.66525 μM | SANGER |
EGI-1 | - | Growth Inhibition Assay | - | IC50=16.5365 μM | SANGER |
EKVX | - | Growth Inhibition Assay | - | IC50=4.22524 μM | SANGER |
EM-2 | - | Growth Inhibition Assay | - | IC50=10.2426 μM | SANGER |
EPLC-272H | - | Growth Inhibition Assay | - | IC50=7.16246 μM | SANGER |
ES1 | - | Growth Inhibition Assay | - | IC50=29.8544 μM | SANGER |
ES4 | - | Growth Inhibition Assay | - | IC50=32.3922 μM | SANGER |
ES5 | - | Growth Inhibition Assay | - | IC50=13.1356 μM | SANGER |
ES7 | - | Growth Inhibition Assay | - | IC50=3.46729 μM | SANGER |
ES8 | - | Growth Inhibition Assay | - | IC50=6.97588 μM | SANGER |
ETK-1 | - | Growth Inhibition Assay | - | IC50=21.8152 μM | SANGER |
EW-1 | - | Growth Inhibition Assay | - | IC50=33.9322 μM | SANGER |
EW-13 | - | Growth Inhibition Assay | - | IC50=20.5443 μM | SANGER |
EW-22 | - | Growth Inhibition Assay | - | IC50=21.376 μM | SANGER |
FADU | - | Growth Inhibition Assay | - | IC50=8.03654 μM | SANGER |
FTC-133 | - | Growth Inhibition Assay | - | IC50=12.0076 μM | SANGER |
G-361 | - | Growth Inhibition Assay | - | IC50=2.2168 μM | SANGER |
G-401 | - | Growth Inhibition Assay | - | IC50=10.7626 μM | SANGER |
G-402 | - | Growth Inhibition Assay | - | IC50=7.30051 μM | SANGER |
GAMG | - | Growth Inhibition Assay | - | IC50=7.64131 μM | SANGER |
GB-1 | - | Growth Inhibition Assay | - | IC50=15.6437 μM | SANGER |
GCIY | - | Growth Inhibition Assay | - | IC50=5.51378 μM | SANGER |
GCT | - | Growth Inhibition Assay | - | IC50=39.1852 μM | SANGER |
GI-ME-N | - | Growth Inhibition Assay | - | IC50=9.70137 μM | SANGER |
GMS-10 | - | Growth Inhibition Assay | - | IC50=10.8971 μM | SANGER |
GOTO | - | Growth Inhibition Assay | - | IC50=3.9149 μM | SANGER |
GT3TKB | - | Growth Inhibition Assay | - | IC50=12.3074 μM | SANGER |
H4 | - | Growth Inhibition Assay | - | IC50=47.6621 μM | SANGER |
HAL-01 | - | Growth Inhibition Assay | - | IC50=45.1379 μM | SANGER |
HCC1806 | - | Growth Inhibition Assay | - | IC50=19.1591 μM | SANGER |
HCC1937 | - | Growth Inhibition Assay | - | IC50=9.69865 μM | SANGER |
HCC2157 | - | Growth Inhibition Assay | - | IC50=21.36 μM | SANGER |
HCC2998 | - | Growth Inhibition Assay | - | IC50=26.0283 μM | SANGER |
HCC70 | - | Growth Inhibition Assay | - | IC50=5.03939 μM | SANGER |
HCE-4 | - | Growth Inhibition Assay | - | IC50=29.8786 μM | SANGER |
HDLM-2 | - | Growth Inhibition Assay | - | IC50=0.32345 μM | SANGER |
HEC-1 | - | Growth Inhibition Assay | - | IC50=20.4978 μM | SANGER |
HH | - | Growth Inhibition Assay | - | IC50=1.18093 μM | SANGER |
HL-60 | - | Growth Inhibition Assay | - | IC50=1.3819 μM | SANGER |
HLE | - | Growth Inhibition Assay | - | IC50=22.697 μM | SANGER |
HMV-II | - | Growth Inhibition Assay | - | IC50=39.5047 μM | SANGER |
HO-1-N-1 | - | Growth Inhibition Assay | - | IC50=24.3093 μM | SANGER |
HOP-62 | - | Growth Inhibition Assay | - | IC50=11.7508 μM | SANGER |
HOP-92 | - | Growth Inhibition Assay | - | IC50=12.5233 μM | SANGER |
HOS | - | Growth Inhibition Assay | - | IC50=8.37589 μM | SANGER |
HPAF-II | - | Growth Inhibition Assay | - | IC50=21.8923 μM | SANGER |
Hs-578-T | - | Growth Inhibition Assay | - | IC50=20.5583 μM | SANGER |
HSC-2 | - | Growth Inhibition Assay | - | IC50=5.41773 μM | SANGER |
HSC-3 | - | Growth Inhibition Assay | - | IC50=23.8527 μM | SANGER |
HT | - | Growth Inhibition Assay | - | IC50=8.3649 μM | SANGER |
HT-1080 | - | Growth Inhibition Assay | - | IC50=8.25093 μM | SANGER |
HT-1376 | - | Growth Inhibition Assay | - | IC50=16.8446 μM | SANGER |
HT-144 | - | Growth Inhibition Assay | - | IC50=18.7427 μM | SANGER |
HT-3 | - | Growth Inhibition Assay | - | IC50=38.4436 μM | SANGER |
HTC-C3 | - | Growth Inhibition Assay | - | IC50=11.0714 μM | SANGER |
HuCCT1 | - | Growth Inhibition Assay | - | IC50=42.5289 μM | SANGER |
HuH-7 | - | Growth Inhibition Assay | - | IC50=2.56702 μM | SANGER |
HuO-3N1 | - | Growth Inhibition Assay | - | IC50=0.46636 μM | SANGER |
HuO9 | - | Growth Inhibition Assay | - | IC50=7.71743 μM | SANGER |
HuP-T4 | - | Growth Inhibition Assay | - | IC50=30.9638 μM | SANGER |
IA-LM | - | Growth Inhibition Assay | - | IC50=4.27935 μM | SANGER |
IGR-1 | - | Growth Inhibition Assay | - | IC50=48.6645 μM | SANGER |
IGROV-1 | - | Growth Inhibition Assay | - | IC50=5.25292 μM | SANGER |
IST-MEL1 | - | Growth Inhibition Assay | - | IC50=4.58263 μM | SANGER |
IST-MES1 | - | Growth Inhibition Assay | - | IC50=40.1502 μM | SANGER |
IST-SL1 | - | Growth Inhibition Assay | - | IC50=6.69369 μM | SANGER |
J-RT3-T3-5 | - | Growth Inhibition Assay | - | IC50=6.63291 μM | SANGER |
JVM-3 | - | Growth Inhibition Assay | - | IC50=3.48077 μM | SANGER |
K5 | - | Growth Inhibition Assay | - | IC50=10.9071 μM | SANGER |
K-562 | - | Growth Inhibition Assay | - | IC50=19.8926 μM | SANGER |
KALS-1 | - | Growth Inhibition Assay | - | IC50=2.69633 μM | SANGER |
KARPAS-299 | - | Growth Inhibition Assay | - | IC50=7.32622 μM | SANGER |
KG-1 | - | Growth Inhibition Assay | - | IC50=2.67924 μM | SANGER |
KGN | - | Growth Inhibition Assay | - | IC50=16.5586 μM | SANGER |
KINGS-1 | - | Growth Inhibition Assay | - | IC50=21.6316 μM | SANGER |
KM12 | - | Growth Inhibition Assay | - | IC50=25.5807 μM | SANGER |
KM-H2 | - | Growth Inhibition Assay | - | IC50=36.4743 μM | SANGER |
KNS-62 | - | Growth Inhibition Assay | - | IC50=8.37762 μM | SANGER |
KNS-81-FD | - | Growth Inhibition Assay | - | IC50=32.0128 μM | SANGER |
KP-N-YN | - | Growth Inhibition Assay | - | IC50=27.8043 μM | SANGER |
KP-N-YS | - | Growth Inhibition Assay | - | IC50=1.14231 μM | SANGER |
KU-19-19 | - | Growth Inhibition Assay | - | IC50=4.32921 μM | SANGER |
KURAMOCHI | - | Growth Inhibition Assay | - | IC50=15.971 μM | SANGER |
KYSE-150 | - | Growth Inhibition Assay | - | IC50=47.1052 μM | SANGER |
KYSE-410 | - | Growth Inhibition Assay | - | IC50=5.47636 μM | SANGER |
KYSE-450 | - | Growth Inhibition Assay | - | IC50=28.8091 μM | SANGER |
KYSE-510 | - | Growth Inhibition Assay | - | IC50=43.1754 μM | SANGER |
L-363 | - | Growth Inhibition Assay | - | IC50=4.77116 μM | SANGER |
LAMA-84 | - | Growth Inhibition Assay | - | IC50=0.98833 μM | SANGER |
LAN-6 | - | Growth Inhibition Assay | - | IC50=21.0396 μM | SANGER |
LB1047-RCC | - | Growth Inhibition Assay | - | IC50=6.17522 μM | SANGER |
LB2241-RCC | - | Growth Inhibition Assay | - | IC50=2.14146 μM | SANGER |
LB2518-MEL | - | Growth Inhibition Assay | - | IC50=31.0744 μM | SANGER |
LB373-MEL-D | - | Growth Inhibition Assay | - | IC50=27.1294 μM | SANGER |
LB996-RCC | - | Growth Inhibition Assay | - | IC50=11.0723 μM | SANGER |
LCLC-103H | - | Growth Inhibition Assay | - | IC50=44.8703 μM | SANGER |
LCLC-97TM1 | - | Growth Inhibition Assay | - | IC50=8.21122 μM | SANGER |
LNCaP-Clone-FGC | - | Growth Inhibition Assay | - | IC50=17.5201 μM | SANGER |
LoVo | - | Growth Inhibition Assay | - | IC50=0.86749 μM | SANGER |
LOXIMVI | - | Growth Inhibition Assay | - | IC50=15.8919 μM | SANGER |
LU-134-A | - | Growth Inhibition Assay | - | IC50=4.59685 μM | SANGER |
LXF-289 | - | Growth Inhibition Assay | - | IC50=3.91041 μM | SANGER |
M14 | - | Growth Inhibition Assay | - | IC50=13.0335 μM | SANGER |
MDA-MB-157 | - | Growth Inhibition Assay | - | IC50=40.9462 μM | SANGER |
MDA-MB-361 | - | Growth Inhibition Assay | - | IC50=19.0714 μM | SANGER |
MDA-MB-415 | - | Growth Inhibition Assay | - | IC50=5.00314 μM | SANGER |
ME-180 | - | Growth Inhibition Assay | - | IC50=15.4783 μM | SANGER |
MEL-HO | - | Growth Inhibition Assay | - | IC50=4.77989 μM | SANGER |
MG-63 | - | Growth Inhibition Assay | - | IC50=3.62676 μM | SANGER |
MHH-ES-1 | - | Growth Inhibition Assay | - | IC50=32.4872 μM | SANGER |
MHH-NB-11 | - | Growth Inhibition Assay | - | IC50=6.32721 μM | SANGER |
MHH-PREB-1 | - | Growth Inhibition Assay | - | IC50=2.16609 μM | SANGER |
MIA-PaCa-2 | - | Growth Inhibition Assay | - | IC50=7.36823 μM | SANGER |
MKN1 | - | Growth Inhibition Assay | - | IC50=24.68 μM | SANGER |
MKN7 | - | Growth Inhibition Assay | - | IC50=28.5964 μM | SANGER |
MLMA | - | Growth Inhibition Assay | - | IC50=5.83606 μM | SANGER |
MN-60 | - | Growth Inhibition Assay | - | IC50=24.8519 μM | SANGER |
MOLT-4 | - | Growth Inhibition Assay | - | IC50=2.21888 μM | SANGER |
Mo-T | - | Growth Inhibition Assay | - | IC50=48.279 μM | SANGER |
MS-1 | - | Growth Inhibition Assay | - | IC50=15.5623 μM | SANGER |
MV-4-11 | - | Growth Inhibition Assay | - | IC50=2.3739 μM | SANGER |
MZ2-MEL | - | Growth Inhibition Assay | - | IC50=14.1488 μM | SANGER |
MZ7-mel | - | Growth Inhibition Assay | - | IC50=15.1067 μM | SANGER |
NB10 | - | Growth Inhibition Assay | - | IC50=26.234 μM | SANGER |
NB13 | - | Growth Inhibition Assay | - | IC50=25.5898 μM | SANGER |
NB14 | - | Growth Inhibition Assay | - | IC50=6.79761 μM | SANGER |
NB5 | - | Growth Inhibition Assay | - | IC50=10.7559 μM | SANGER |
NB69 | - | Growth Inhibition Assay | - | IC50=5.3242 μM | SANGER |
NB7 | - | Growth Inhibition Assay | - | IC50=1.24745 μM | SANGER |
NBsusSR | - | Growth Inhibition Assay | - | IC50=6.82502 μM | SANGER |
NCI-H1048 | - | Growth Inhibition Assay | - | IC50=21.2258 μM | SANGER |
NCI-H1092 | - | Growth Inhibition Assay | - | IC50=13.7475 μM | SANGER |
NCI-H1155 | - | Growth Inhibition Assay | - | IC50=10.8376 μM | SANGER |
NCI-H1299 | - | Growth Inhibition Assay | - | IC50=48.7248 μM | SANGER |
NCI-H1304 | - | Growth Inhibition Assay | - | IC50=15.8928 μM | SANGER |
NCI-H1355 | - | Growth Inhibition Assay | - | IC50=5.296 μM | SANGER |
NCI-H1395 | - | Growth Inhibition Assay | - | IC50=34.0799 μM | SANGER |
NCI-H1437 | - | Growth Inhibition Assay | - | IC50=10.5725 μM | SANGER |
NCI-H1563 | - | Growth Inhibition Assay | - | IC50=11.1011 μM | SANGER |
NCI-H1703 | - | Growth Inhibition Assay | - | IC50=31.0905 μM | SANGER |
NCI-H1755 | - | Growth Inhibition Assay | - | IC50=10.2428 μM | SANGER |
NCI-H1770 | - | Growth Inhibition Assay | - | IC50=0.02143 μM | SANGER |
NCI-H1793 | - | Growth Inhibition Assay | - | IC50=1.4584 μM | SANGER |
NCI-H2030 | - | Growth Inhibition Assay | - | IC50=13.2062 μM | SANGER |
NCI-H2228 | - | Growth Inhibition Assay | - | IC50=31.4651 μM | SANGER |
NCI-H2291 | - | Growth Inhibition Assay | - | IC50=18.4345 μM | SANGER |
NCI-H2347 | - | Growth Inhibition Assay | - | IC50=6.93213 μM | SANGER |
NCI-H2452 | - | Growth Inhibition Assay | - | IC50=21.8647 μM | SANGER |
NCI-H28 | - | Growth Inhibition Assay | - | IC50=8.16962 μM | SANGER |
NCI-H292 | - | Growth Inhibition Assay | - | IC50=1.74013 μM | SANGER |
NCI-H358 | - | Growth Inhibition Assay | - | IC50=44.0304 μM | SANGER |
NCI-H520 | - | Growth Inhibition Assay | - | IC50=36.7541 μM | SANGER |
NCI-H522 | - | Growth Inhibition Assay | - | IC50=22.8431 μM | SANGER |
NCI-H526 | - | Growth Inhibition Assay | - | IC50=0.28407 μM | SANGER |
NCI-H596 | - | Growth Inhibition Assay | - | IC50=19.6391 μM | SANGER |
NCI-H630 | - | Growth Inhibition Assay | - | IC50=22.0296 μM | SANGER |
NCI-H650 | - | Growth Inhibition Assay | - | IC50=11.8961 μM | SANGER |
NCI-H727 | - | Growth Inhibition Assay | - | IC50=22.735 μM | SANGER |
NCI-H82 | - | Growth Inhibition Assay | - | IC50=7.26659 μM | SANGER |
NCI-SNU-1 | - | Growth Inhibition Assay | - | IC50=0.60994 μM | SANGER |
NEC8 | - | Growth Inhibition Assay | - | IC50=1.5535 μM | SANGER |
NKM-1 | - | Growth Inhibition Assay | - | IC50=7.74955 μM | SANGER |
NOMO-1 | - | Growth Inhibition Assay | - | IC50=37.8089 μM | SANGER |
NOS-1 | - | Growth Inhibition Assay | - | IC50=3.65312 μM | SANGER |
NTERA-S-cl-D1 | - | Growth Inhibition Assay | - | IC50=32.0739 μM | SANGER |
NUGC-3 | - | Growth Inhibition Assay | - | IC50=15.6245 μM | SANGER |
NY | - | Growth Inhibition Assay | - | IC50=3.45022 μM | SANGER |
OAW-42 | - | Growth Inhibition Assay | - | IC50=8.95964 μM | SANGER |
OE33 | - | Growth Inhibition Assay | - | IC50=47.1429 μM | SANGER |
OS-RC-2 | - | Growth Inhibition Assay | - | IC50=11.0559 μM | SANGER |
OVCAR-4 | - | Growth Inhibition Assay | - | IC50=7.31328 μM | SANGER |
OVCAR-8 | - | Growth Inhibition Assay | - | IC50=45.3564 μM | SANGER |
P12-ICHIKAWA | - | Growth Inhibition Assay | - | IC50=44.6112 μM | SANGER |
P30-OHK | - | Growth Inhibition Assay | - | IC50=29.3048 μM | SANGER |
PA-1 | - | Growth Inhibition Assay | - | IC50=1.58294 μM | SANGER |
PANC-03-27 | - | Growth Inhibition Assay | - | IC50=16.7662 μM | SANGER |
PANC-08-13 | - | Growth Inhibition Assay | - | IC50=3.41278 μM | SANGER |
PC-3 | - | Growth Inhibition Assay | - | IC50=8.27392 μM | SANGER |
PFSK-1 | - | Growth Inhibition Assay | - | IC50=5.62194 μM | SANGER |
QIMR-WIL | - | Growth Inhibition Assay | - | IC50=3.41341 μM | SANGER |
Ramos-2G6-4C10 | - | Growth Inhibition Assay | - | IC50=2.19909 μM | SANGER |
RCC10RGB | - | Growth Inhibition Assay | - | IC50=20.6719 μM | SANGER |
RD | - | Growth Inhibition Assay | - | IC50=22.7518 μM | SANGER |
RH-1 | - | Growth Inhibition Assay | - | IC50=16.825 μM | SANGER |
RH-18 | - | Growth Inhibition Assay | - | IC50=4.44953 μM | SANGER |
RMG-I | - | Growth Inhibition Assay | - | IC50=27.2029 μM | SANGER |
RO82-W-1 | - | Growth Inhibition Assay | - | IC50=7.74533 μM | SANGER |
RPMI-7951 | - | Growth Inhibition Assay | - | IC50=28.2456 μM | SANGER |
RPMI-8226 | - | Growth Inhibition Assay | - | IC50=38.9519 μM | SANGER |
RPMI-8866 | - | Growth Inhibition Assay | - | IC50=17.0699 μM | SANGER |
RS4-11 | - | Growth Inhibition Assay | - | IC50=2.56023 μM | SANGER |
RT-112 | - | Growth Inhibition Assay | - | IC50=29.4611 μM | SANGER |
RVH-421 | - | Growth Inhibition Assay | - | IC50=6.07338 μM | SANGER |
RXF393 | - | Growth Inhibition Assay | - | IC50=29.2906 μM | SANGER |
SCC-4 | - | Growth Inhibition Assay | - | IC50=31.9181 μM | SANGER |
SF126 | - | Growth Inhibition Assay | - | IC50=4.60715 μM | SANGER |
SF295 | - | Growth Inhibition Assay | - | IC50=40.8066 μM | SANGER |
SJSA-1 | - | Growth Inhibition Assay | - | IC50=20.5688 μM | SANGER |
SKG-IIIa | - | Growth Inhibition Assay | - | IC50=13.0554 μM | SANGER |
SK-LMS-1 | - | Growth Inhibition Assay | - | IC50=27.0704 μM | SANGER |
SK-LU-1 | - | Growth Inhibition Assay | - | IC50=23.4683 μM | SANGER |
SK-MEL-1 | - | Growth Inhibition Assay | - | IC50=1.79479 μM | SANGER |
SK-MEL-2 | - | Growth Inhibition Assay | - | IC50=20.1559 μM | SANGER |
SK-MEL-28 | - | Growth Inhibition Assay | - | IC50=10.8202 μM | SANGER |
SK-MEL-3 | - | Growth Inhibition Assay | - | IC50=2.1649 μM | SANGER |
SK-MEL-30 | - | Growth Inhibition Assay | - | IC50=3.42598 μM | SANGER |
SK-MES-1 | - | Growth Inhibition Assay | - | IC50=24.0161 μM | SANGER |
SK-N-AS | - | Growth Inhibition Assay | - | IC50=0.62216 μM | SANGER |
SK-NEP-1 | - | Growth Inhibition Assay | - | IC50=2.38783 μM | SANGER |
SK-OV-3 | - | Growth Inhibition Assay | - | IC50=27.7593 μM | SANGER |
SK-PN-DW | - | Growth Inhibition Assay | - | IC50=12.1902 μM | SANGER |
SK-UT-1 | - | Growth Inhibition Assay | - | IC50=3.1531 μM | SANGER |
SN12C | - | Growth Inhibition Assay | - | IC50=4.71898 μM | SANGER |
SNB75 | - | Growth Inhibition Assay | - | IC50=48.1874 μM | SANGER |
SNU-423 | - | Growth Inhibition Assay | - | IC50=13.381 μM | SANGER |
SNU-449 | - | Growth Inhibition Assay | - | IC50=8.2793 μM | SANGER |
SNU-C2B | - | Growth Inhibition Assay | - | IC50=44.7903 μM | SANGER |
SW1088 | - | Growth Inhibition Assay | - | IC50=27.5042 μM | SANGER |
SW13 | - | Growth Inhibition Assay | - | IC50=40.519 μM | SANGER |
SW1573 | - | Growth Inhibition Assay | - | IC50=27.11 μM | SANGER |
SW1783 | - | Growth Inhibition Assay | - | IC50=16.0993 μM | SANGER |
SW684 | - | Growth Inhibition Assay | - | IC50=17.0154 μM | SANGER |
SW900 | - | Growth Inhibition Assay | - | IC50=44.0758 μM | SANGER |
SW962 | - | Growth Inhibition Assay | - | IC50=3.20352 μM | SANGER |
SW982 | - | Growth Inhibition Assay | - | IC50=7.30203 μM | SANGER |
T47D | - | Growth Inhibition Assay | - | IC50=18.488 μM | SANGER |
TCCSUP | - | Growth Inhibition Assay | - | IC50=47.6264 μM | SANGER |
TE-1 | - | Growth Inhibition Assay | - | IC50=41.8714 μM | SANGER |
TE-11 | - | Growth Inhibition Assay | - | IC50=11.9315 μM | SANGER |
TE-12 | - | Growth Inhibition Assay | - | IC50=39.2448 μM | SANGER |
TE-5 | - | Growth Inhibition Assay | - | IC50=15.2333 μM | SANGER |
TE-6 | - | Growth Inhibition Assay | - | IC50=38.124 μM | SANGER |
TE-8 | - | Growth Inhibition Assay | - | IC50=44.5658 μM | SANGER |
TE-9 | - | Growth Inhibition Assay | - | IC50=30.8737 μM | SANGER |
TGBC11TKB | - | Growth Inhibition Assay | - | IC50=22.049 μM | SANGER |
TI-73 | - | Growth Inhibition Assay | - | IC50=16.9408 μM | SANGER |
TK10 | - | Growth Inhibition Assay | - | IC50=17.0079 μM | SANGER |
TYK-nu | - | Growth Inhibition Assay | - | IC50=4.80128 μM | SANGER |
U031 | - | Growth Inhibition Assay | - | IC50=3.59368 μM | SANGER |
U-118-MG | - | Growth Inhibition Assay | - | IC50=26.0808 μM | SANGER |
U251 | - | Growth Inhibition Assay | - | IC50=39.0124 μM | SANGER |
U-87-MG | - | Growth Inhibition Assay | - | IC50=45.1022 μM | SANGER |
UM-UC-3 | - | Growth Inhibition Assay | - | IC50=6.64334 μM | SANGER |
VA-ES-BJ | - | Growth Inhibition Assay | - | IC50=8.34686 μM | SANGER |
VM-CUB-1 | - | Growth Inhibition Assay | - | IC50=10.6164 μM | SANGER |
VMRC-RCZ | - | Growth Inhibition Assay | - | IC50=2.77328 μM | SANGER |
WM-115 | - | Growth Inhibition Assay | - | IC50=11.6824 μM | SANGER |
YH-13 | - | Growth Inhibition Assay | - | IC50=3.87189 μM | SANGER |
YKG-1 | - | Growth Inhibition Assay | - | IC50=44.781 μM | SANGER |
ZR-75-30 | - | Growth Inhibition Assay | - | IC50=16.9361 μM | SANGER |
靶点 | Description | IC50 |
---|---|---|
DNA-PK | IC50:14nM | |
PI3K | IC50:5μM |
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