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CAS No.: 182431-12-5
Synonyms: AEGR-733;BMS-201038;AEGR 773
Lomitapide is an inhibitor of microsomal triglyceride-transfer protein (MTP) wtih in vitro IC50 of 8 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00474240 | Hypercholesterolemia | Phase 2 | Completed | - | United States, Alabama ... more >> Medical Affiliated Research Center Huntsville, Alabama, United States, 35801 United States, Florida Jacksonville Center for Clinical research Jacksonville, Florida, United States, 32205 Jacksonville Center For Clinical Research Jacksonville, Florida, United States, 32216 Renstar Medical Research Ocala, Florida, United States, 34471 United States, Georgia North Georgia Clinical Research Woodstock, Georgia, United States, 30189 United States, Illinois Radiant Research Chicago, Illinois, United States, 60610 United States, Indiana Medsphere Medical Research Center Evansville, Indiana, United States, 47714 Midwest Institute for Clinical Research Indianapolis, Indiana, United States, 46260 United States, Maine Maine Research Associates Auburn, Maine, United States, 04210 United States, Maryland Health Trends Research Baltimore, Maryland, United States, 21209 United States, North Carolina Piedmont Medical Research Associates Winston-Salem, North Carolina, United States, 27103 United States, Ohio Sterling Research Group Cincinnati, Ohio, United States, 45246 United States, South Carolina Coastal Carolina Research Center Goose Creek, South Carolina, United States, 29445 United States, Texas Dallas Diabetes and Endocrine Center Dallas, Texas, United States, 75230 Diabetes and Glandular Disease Research Dallas, Texas, United States, 78229 United States, Virginia Hampton Roads Center for Clinical Research Norfolk, Virginia, United States, 23502 National Clinical Research Richmond, Virginia, United States, 23294 Collapse << |
NCT00474240 | - | - | Completed | - | - |
NCT00559962 | - | - | Completed | - | - |
实验方案
技术信息
CAS号 | 182431-12-5 | 储存条件 |
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分子式 | C39H37F6N3O2 | 运输 | 蓝冰 | |
分子量 | 693.72 | 别名 | AEGR-733;BMS-201038;AEGR 773;Lojuxta;洛美他派 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00474240 | Hypercholesterolemia | Phase 2 | Completed | - | United States, Alabama ... more >> Medical Affiliated Research Center Huntsville, Alabama, United States, 35801 United States, Florida Jacksonville Center for Clinical research Jacksonville, Florida, United States, 32205 Jacksonville Center For Clinical Research Jacksonville, Florida, United States, 32216 Renstar Medical Research Ocala, Florida, United States, 34471 United States, Georgia North Georgia Clinical Research Woodstock, Georgia, United States, 30189 United States, Illinois Radiant Research Chicago, Illinois, United States, 60610 United States, Indiana Medsphere Medical Research Center Evansville, Indiana, United States, 47714 Midwest Institute for Clinical Research Indianapolis, Indiana, United States, 46260 United States, Maine Maine Research Associates Auburn, Maine, United States, 04210 United States, Maryland Health Trends Research Baltimore, Maryland, United States, 21209 United States, North Carolina Piedmont Medical Research Associates Winston-Salem, North Carolina, United States, 27103 United States, Ohio Sterling Research Group Cincinnati, Ohio, United States, 45246 United States, South Carolina Coastal Carolina Research Center Goose Creek, South Carolina, United States, 29445 United States, Texas Dallas Diabetes and Endocrine Center Dallas, Texas, United States, 75230 Diabetes and Glandular Disease Research Dallas, Texas, United States, 78229 United States, Virginia Hampton Roads Center for Clinical Research Norfolk, Virginia, United States, 23502 National Clinical Research Richmond, Virginia, United States, 23294 Collapse << |
NCT00474240 | - | - | Completed | - | - |
NCT00559962 | - | - | Completed | - | - |
NCT00359281 | Healthy | Phase 2 | Completed | - | United States, Pennsylvania ... more >> University of Pennsylvania Philadelphia, Pennsylvania, United States, 19104 Collapse << |
NCT00559962 | Hyperlipidemia | Phase 2 | Completed | - | United States, California ... more >> Scripps Clinic San Diego, California, United States, 92128 Radiant Research Santa Rosa, California, United States, 95405 United States, District of Columbia MedStar Research Institute Washington, District of Columbia, United States, 20003 United States, Illinois Radiant Research Chicago, Illinois, United States, 60610 United States, Iowa University of Iowa Iowa City, Iowa, United States, 52242 United States, Kentucky LMARC Louisville, Kentucky, United States, 40213 United States, Maine Maine Research Associates Auburn, Maine, United States, 04210 United States, Maryland Health Trends Research Baltimore, Maryland, United States, 21209 Johns Hopkins Baltimore, Maryland, United States, 21287 United States, Missouri Washington Univ. School of Medicine Saint Louis, Missouri, United States, 63110 United States, Ohio Sterling Research Group Cincinnati, Ohio, United States, 45219 United States, Pennsylvania University of Pennsylvania Philadelphia, Pennsylvania, United States, 19104 United States, Texas Baylor College of Medicine Houston, Texas, United States, 77030 Clinical Trial Network Houston, Texas, United States, 77074 dgd Research San Antonio, Texas, United States, 78229 Collapse << |
NCT00405067 | Hypercholesterolemia | Phase 2 | Completed | - | United States, New Jersey ... more >> Pharmanet, Inc Princeton, New Jersey, United States, 08540-6242 Collapse << |
NCT00405067 | - | - | Completed | - | - |
NCT00690443 | - | - | Completed | - | - |
NCT00690443 | Hypercholesterolemia | Phase 2 | Completed | - | United States, Florida ... more >> Linda Murray, DO - Radiant Research Pinellas Park, Florida, United States, 33781 United States, Minnesota Sheila Rodstein, MD Edina, Minnesota, United States, 55435 United States, Ohio Dennis McCluskey, MD - Radiant Research Mogadore, Ohio, United States, 44260 United States, Texas Michele Reynolds, MD Dallas, Texas, United States, 75231 William Jennings, MD - Radiant Research San Antonio, Texas, United States, 78229 Collapse << |
NCT00730236 | Homozygous Familial Hyperchole... more >>sterolemia Collapse << | Phase 3 | Completed | - | United States, California ... more >> Cedars-Sinai Medical Center Los Angeles, California, United States, 90048 United States, Pennsylvania University of Pennsylvania Philadelphia, Pennsylvania, United States, 19104 Canada, Ontario Robarts Research Institute London, Ontario, Canada, N6A 5K8 Canada, Quebec Lipid Clinic and University of Montreal Community Genomic Medicine Center Chicoutimi, Quebec, Canada, G7H 5H6 Italy Dipartimento di Medicina Clinica e Della Patalogie Emergenti Palermo, Sicily, Italy Medicina Interna Universitaria Ferrara, Italy Centro Universitario Dislipidemie Milano, Italy Dipartimento di Clinica e Terapia Medica Roma, Italy South Africa Cardiology Research Bloemfontein, South Africa, 9300 University of Capetown Cape town, South Africa, 7925 Collapse << |
NCT00730236 | - | - | Completed | - | - |
NCT01760187 | Healthy Volunteer | Phase 1 | Completed | - | United Kingdom ... more >> Richmond Pharmacology Ltd Croydon, Surrey, United Kingdom, CR7 7YE Collapse << |
NCT01556906 | Homozygous Familial Hyperchole... more >>sterolemia Collapse << | Phase 2 | Completed | - | United States, Pennsylvania ... more >> University of Pennsylvania Philadelphia, Pennsylvania, United States, 19104 Collapse << |
NCT01556906 | - | - | Completed | - | - |
NCT01915771 | Intra-subject Variability of P... more >>harmacokinetics Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Richmond Pharmacology Croydon, Surrey, United Kingdom, CR7 7YE Collapse << |
NCT02399839 | - | - | Enrolling by invitation | March 2028 | - |
NCT00359281 | - | - | Completed | - | - |
NCT02080468 | Healthy | Phase 1 | Completed | - | United States, Texas ... more >> Covance Clinical Research Unit, Inc Dallas, Texas, United States, 75247 Collapse << |
NCT00943306 | Familial Hypercholesterolemia | Phase 3 | Completed | - | United States, California ... more >> Cedars-Sinai Medical Center Los Angeles, California, United States, 90048 United States, Pennsylvania University of Pennsylvania Philadelphia, Pennsylvania, United States, 19104 Canada, Ontario Robarts Research Institute London, Ontario, Canada, N6A 5K8 Canada, Quebec Lipid Clinic and University of Montreal Community Genomic Medicine Center Chicoutimi, Quebec, Canada, G7H 5H6 Italy Medicina Interna Universitaria Ferrara, Sicily, Italy Dipartimento di Medicina Clinica e Delle Patologie Emergenti Palermo, Sicily, Italy Centro Universitario Dislipidemie Milano, Italy DAI Ematologia, Oncologia, Anatomia Patologica e Medicina Roma, Italy South Africa Cardiology Research Bloemfontein, South Africa, 9300 University of Capetown Cape town, South Africa, 7925 Collapse << |
NCT00943306 | - | - | Completed | - | - |
NCT02135705 | - | - | Enrolling by invitation | September 2028 | United States, Michigan ... more >> Complete Family Care Sterling Heights, Michigan, United States, 48314 Collapse << |
NCT02765841 | Homozygous Familial Hyperchole... more >>sterolemia Collapse << | Phase 3 | Withdrawn | December 2019 | - |
NCT02044419 | Healthy | Phase 1 | Completed | - | United Kingdom ... more >> Richmond Pharmacology Ltd Croydon, Surrey, United Kingdom, CR7 7YE Collapse << |
NCT02044419 | - | - | Completed | - | - |
NCT02399852 | - | - | Withdrawn | December 2021 | - |
NCT01760187 | - | - | Completed | - | - |
NCT02080455 | Effect of Atorvastatin on the ... more >>Pharmacokinetics of Lomitapide Collapse << | Phase 1 | Completed | - | United States, Texas ... more >> Covance Clinical Research Unit, Inc Dallas, Texas, United States, 75247 Collapse << |
NCT02173158 | - | - | Completed | - | - |
NCT02173158 | Familial Hypercholesterolemia ... more >>- Homozygous Collapse << | Phase 3 | Completed | - | Japan ... more >> Kurume-shi, Fukuoka, Japan, 830-8522 Kanazawa, Ishikawa, Japan, 920-8641 Osakashi, Osaka, Japan, 530-00001 Suita-shi, Osaka, Japan, 565-8565 Tokorozawa, Saitama, Japan, 359-1142 Bunkyo-ku, Tokyo, Japan, 113-8519 Collapse << |
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