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CAS No.: 136790-76-6
Synonyms: RU-0211;SPI-0211;鲁比前列酮
Lubiprostone is an ClC-2 chloride channel activator used in the treatment of idiopathic chronic constipation.
生物活性
动物研究 | ||||||||||||||||||||||||||||||||||
剂量 | Mice: 500 μg/kg/day[3] (p.o.) | |||||||||||||||||||||||||||||||||
给药途径 | p.o. | |||||||||||||||||||||||||||||||||
动物药代数据 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00953017 | - | - | Completed | - | - |
NCT03720613 | - | - | Not yet recruiting | November 1, 2025 | - |
NCT00577499 | - | - | Terminated(Recruitment was sub... more >>optimal) Collapse << | - | - |
实验方案
技术信息
CAS号 | 136790-76-6 | 储存条件 |
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分子式 | C20H32F2O5 | 运输 | 蓝冰 | |||||||
分子量 | 390.46 | 别名 | RU-0211;SPI-0211;鲁比前列酮 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00953017 | - | - | Completed | - | - |
NCT03720613 | - | - | Not yet recruiting | November 1, 2025 | - |
NCT00577499 | - | - | Terminated(Recruitment was sub... more >>optimal) Collapse << | - | - |
NCT02481947 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Completed | - | - |
NCT00399542 | Irritable Bowel Syndrome ... more >> Constipation Collapse << | Phase 3 | Completed | - | - |
NCT01298219 | Opioid-induced Bowel Dysfuncti... more >>on Collapse << | Phase 3 | Completed | - | - |
NCT00399542 | - | - | Completed | - | - |
NCT00380250 | Irritable Bowel Syndrome With ... more >>Constipation Collapse << | Phase 3 | Completed | - | - |
NCT00611442 | Bowel Preparation for Colonosc... more >>opy Collapse << | Not Applicable | Completed | - | United States, Texas ... more >> Brooke Army Medical Center Fort Sam Houston, Texas, United States, 78234 Collapse << |
NCT00611442 | - | - | Completed | - | - |
NCT01372423 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Completed | - | - |
NCT01162863 | Irritable Bowel Syndrome ... more >> Constipation Collapse << | Not Applicable | Completed | - | United States, Michigan ... more >> University of Michigan Health System Ann Arbor, Michigan, United States, 48103 Collapse << |
NCT00985569 | - | - | Withdrawn(Enrollment was never... more >> begun.) Collapse << | November 2010 | United States, Florida ... more >> Geriatric Medical Associates Brooksville, Florida, United States Cassellberry Family Practice Casselberry, Florida, United States Osler Geriatrics Melbourne, Florida, United States Collapse << |
NCT00953017 | Colonoscopy | Phase 4 | Completed | - | United States, Texas ... more >> Brooke Army Medical Center San Antonio, Texas, United States, 78248 Collapse << |
NCT01993875 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Completed | - | United States, Alabama ... more >> Anniston, Alabama, United States, 36207 United States, California Anaheim, California, United States, 92801 United States, Florida Deland, Florida, United States, 32720 Hollywood, Florida, United States, 33024 Orlando, Florida, United States, 32809 South Miami, Florida, United States, 33143 United States, Kansas Overland Park, Kansas, United States, 66212 United States, New Jersey Marlton, New Jersey, United States, 08053 United States, North Carolina Raleigh, North Carolina, United States, 27612 United States, Utah Salt Lake City, Utah, United States, 84106 United States, Wisconsin West Bend, Wisconsin, United States, 53095 Collapse << |
NCT01674530 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Completed | - | - |
NCT00934479 | Other Constipation ... more >> Irritable Bowel Syndrome Collapse << | Phase 1 | Completed | - | United States, Arizona ... more >> Mayo Clinic Arizona Scottsdale, Arizona, United States, 85259 Collapse << |
NCT00452335 | Constipation | Phase 4 | Completed | - | United States, Arizona ... more >> Phoenix Children's Hospital Pheonix, Arizona, United States, 85016 United States, Arkansas Arkansas Pediatric Clinic Little Rock, Arkansas, United States, 72005 United States, California Children's Hospital and Research Center Oakland Oakland, California, United States, 94609 United States, Florida Nemours Children's Clinic - Jacksonville Jacksonville, Florida, United States, 32207 Nemours Children's Clinic - Pensacola Pensacola, Florida, United States, 32504 United States, Illinois Center for Children's Digestive Health Park Ridge, Illinois, United States, 60068 University of Illinois at Peoria Peoria, Illinois, United States, 61613 University of Illinois at Chicago Springfield, Illinois, United States, 62708-0787 United States, Indiana Indiana University Indianapolis, Indiana, United States, 46202 United States, Kansas University of Kansas Medical Center Kansas City, Kansas, United States, 66160 United States, Massachusetts Children's Hospital Boston Boston, Massachusetts, United States, 02115 United States, Nebraska The Center for Human Nutrition, Inc. Omaha, Nebraska, United States, 68105 United States, New Jersey AHS Hospital Corporation Morristown, New Jersey, United States, 07962 United States, Ohio Children's Research Institute Columbus, Ohio, United States, 43205 Pediatric Associates of Fairfield, Inc. Fairfield, Ohio, United States, 45014 United States, Pennsylvania Regional Gastroenterology Associates of Lancaster, Ltd. Lancaster, Pennsylvania, United States, 17604 United States, Tennessee Southeastern Clinical Research Chattanooga, Tennessee, United States, 37403 Jackson Clinic Jackson, Tennessee, United States, 38305 United States, Wisconsin Medical College of Wisconsin Milwaukee, Wisconsin, United States, 53226 Collapse << |
NCT00452335 | - | - | Completed | - | - |
NCT00595946 | Opioid-Induced Bowel Dysfuncti... more >>on Collapse << | Phase 3 | Completed | - | - |
NCT00595946 | - | - | Completed | - | - |
NCT00597428 | Opioid-Induced Bowel Dysfuncti... more >>on Collapse << | Phase 3 | Completed | - | - |
NCT01460225 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 4 | Completed | - | United States, New Hampshire ... more >> Dartmouth-Hitchcock Medical Center Lebanon, New Hampshire, United States, 03756 Collapse << |
NCT00380250 | - | - | Completed | - | - |
NCT01162863 | - | - | Completed | - | - |
NCT01460225 | - | - | Completed | - | - |
NCT00620061 | Opioid-Induced Bowel Dysfuncti... more >>on Collapse << | Phase 3 | Completed | - | - |
NCT00689026 | Diabetes Mellitus, Type 1 ... more >> Diabetes Mellitus, Type 2 Collapse << | Not Applicable | Terminated | - | United States, Georgia ... more >> Medical College of Georgia Augusta, Georgia, United States, 30912 Collapse << |
NCT00662363 | Constipation | Not Applicable | Completed | - | United States, Illinois ... more >> Rehabilitation Institute of Chicago Chicago, Illinois, United States, 60302 Collapse << |
NCT00597428 | - | - | Completed | - | - |
NCT00662363 | - | - | Completed | - | - |
NCT00746395 | - | - | Completed | - | - |
NCT00746395 | Inflammatory Bowel Disease | Phase 4 | Completed | - | United States, Alabama ... more >> USA Pavilion at Infirmary West Mobile, Alabama, United States, 36693 Collapse << |
NCT00844831 | Constipation | Phase 4 | Completed | - | United States, Kentucky ... more >> University of Louisville Louisville, Kentucky, United States, 40202 Collapse << |
NCT00689026 | - | - | Terminated | - | - |
NCT02042183 | Constipation - Functional | Phase 3 | Completed | - | - |
NCT01096290 | Constipation | Phase 4 | Completed | - | United States, Alabama ... more >> USA Pavilion at Infirmary West Mobile, Alabama, United States, 36693 Collapse << |
NCT00669461 | - | - | Terminated(Lack of recruitment... more >>) Collapse << | - | - |
NCT00706004 | Constipation ... more >>Cystic Fibrosis Collapse << | Not Applicable | Completed | - | United States, Arkansas ... more >> University of Arkansas for Medical Sciences Little Rock, Arkansas, United States, 72205 Collapse << |
NCT00706004 | - | - | Completed | - | - |
NCT02544152 | Irritable Bowel Syndrome | Phase 2 | Terminated | - | United States, Alabama ... more >> E Squared Research, Inc. Huntsville, Alabama, United States, 35801 United States, Arkansas Arkansas Gastroenterology North Little Rock, Arkansas, United States, 72117 United States, California GW Research Inc. Chula Vista, California, United States, 91910 Inland Empire Liver Foundation Rialto, California, United States, 92377 United States, Florida Prestige Clinical Research Center Miami, Florida, United States, 33133 Advanced Gastroenterology Associates, LLC Palm Harbor, Florida, United States, 34684 United States, Maryland Meritus Center for Clinical Research Hagerstown, Maryland, United States, 21742 United States, Minnesota Mayo Clinic Rochester, Minnesota, United States, 55905 United States, North Carolina PMG Research of Charlotte Charlotte, North Carolina, United States, 28210 PMG Research of Charlotte Concord, North Carolina, United States, 28025 Cumberland Research Associates, LLC Fayetteville, North Carolina, United States, 28304 Wake Research Associates, LLC Raleigh, North Carolina, United States, 27612 United States, Tennessee Clinical Research Solutions Jackson, Tennessee, United States, 38305 United States, Texas Houston Endoscopy Research Center Houston, Texas, United States, 77079 Wellness Clinical Research Associates McKinney, Texas, United States, 75071 Advanced Clinical Research Associates Plano, Texas, United States, 75093 Collapse << |
NCT00844831 | - | - | Completed | - | - |
NCT01166789 | Irritable Bowel Syndrome | Phase 1 | Completed | - | United States, North Carolina ... more >> UNC Clinical and Translational Research Center Chapel Hill, North Carolina, United States, 27599 Collapse << |
NCT00953043 | - | - | Completed | - | - |
NCT00908076 | Parkinson's Disease | Phase 4 | Completed | - | United States, Florida ... more >> University of South Florida Tampa, Florida, United States, 33606 United States, Texas Baylor College of Medicine PDCMDC Houston, Texas, United States, 77030 Collapse << |
NCT00908076 | - | - | Completed | - | - |
NCT00645801 | Colonoscopy | Phase 4 | Completed | - | United States, Michigan ... more >> Henry Ford Hospital Detroit, Michigan, United States, 48202 Henry Ford Health System Novi, Michigan, United States, 48377 Collapse << |
NCT00953043 | Healthy | Phase 4 | Completed | - | United States, Minnesota ... more >> Mayo Clinic Rochester, Minnesota, United States, 55905 Collapse << |
NCT01170039 | Constipation ... more >>Diabetes Collapse << | Phase 4 | Completed | - | United States, Georgia ... more >> Atlanta Veterans Administration Hospital Atlanta, Georgia, United States, 30033 The Emory Clinic Atlanta, Georgia, United States, 30322 Collapse << |
NCT00669461 | Constipation ... more >>Parkinson's Disease Collapse << | Not Applicable | Terminated(Lack of recruitment... more >>) Collapse << | - | United States, Arkansas ... more >> University of Arkansas for Medical Sciences Little Rock, Arkansas, United States, 72205 Collapse << |
NCT01236534 | - | - | Completed | - | - |
NCT01839734 | HIV | Phase 2 | Unknown | June 2015 | United States, Illinois ... more >> Ruth M. Rothstein CORE Center Chicago, Illinois, United States, 60612 Collapse << |
NCT01190020 | Chronic Constipation, Methanog... more >>enesis Collapse << | Phase 1 | Unknown | - | United States, Iowa ... more >> University of Iowa Hospitals and Clinics Recruiting Iowa City, Iowa, United States, 52242 Collapse << |
NCT01170039 | - | - | Completed | - | - |
NCT03010631 | Healthy Volunteers | Phase 3 | Completed | - | United States, Texas ... more >> ICON San Antonio, Texas, United States, 78209 Collapse << |
NCT01447849 | Constipation | Phase 2 Phase 3 | Completed | - | United States, Texas ... more >> Texas Tech University Health Sciences Center El Paso, Texas, United States, 79905 Collapse << |
NCT01085643 | Constipation-predominant Irrit... more >>able Bowel Syndrome Collapse << | Not Applicable | Completed | - | United States, California ... more >> Cedars-Sinai Medical Center Los Angeles, California, United States, 90048 Collapse << |
NCT01085643 | - | - | Completed | - | - |
NCT02138136 | Constipation - Functional | Phase 3 | Completed | - | - |
NCT01447849 | - | - | Completed | - | - |
NCT02651155 | - | - | Completed | - | - |
NCT01469819 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 2 Phase 3 | Completed | - | United States, Texas ... more >> Texas Tech University Health Sciences Center El Paso, Texas, United States, 79905 Collapse << |
NCT01236534 | Multiple Sclerosis ... more >> Constipation Collapse << | Phase 4 | Completed | - | United States, New York ... more >> University of Rochester Rochester, New York, United States, 14642 Collapse << |
NCT01469819 | - | - | Completed | - | - |
NCT01324284 | Colorectal Carcinoma | Phase 3 | Completed | - | - |
NCT03097861 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Completed | - | - |
NCT02695719 | Constipation | Phase 3 | Completed | - | Korea, Republic of ... more >> Cheonan-si, Chungcheongnam-do, Korea, Republic of Seongnam-si, Gyeonggi-do, Korea, Republic of Iksan-si, Jeollabuk-do, Korea, Republic of Daejeon, Korea, Republic of Seoul, Korea, Republic of Collapse << |
NCT02651155 | Constipation | Phase 3 | Completed | - | Russian Federation ... more >> Saint-Petersburg, Pushkin, Russian Federation Barnaul, Russian Federation Kazan, Russian Federation Kemerovo, Russian Federation Krasnodar, Russian Federation Moscow, Russian Federation Novosibirsk, Russian Federation Omsk, Russian Federation Saint Petersburg, Russian Federation Saint-Petersburg, Russian Federation Samara, Russian Federation Ulyanovsk, Russian Federation Yaroslavl, Russian Federation Collapse << |
NCT02729909 | Constipation | Phase 3 | Completed | - | Mexico ... more >> Mexicali, Baja California Norte, Mexico Mexico, Distrito Federal, Mexico Cuautitlan Izcalli, Estado de Mexico, Mexico Tlalnepantla, Estado de Mexico, Mexico Leon, Guanajuato, Mexico Morelia, Michoacan, Mexico Monterrey, Nuevo Le0n, Mexico Culiacan, Sinaloa, Mexico Chihuahua, Mexico Durango, Mexico Collapse << |
NCT02766777 | Constipation - Functional | Phase 3 | Completed | - | United States, Arkansas ... more >> Northwest Arkansas Pediatric Clinic Fayetteville, Arkansas, United States, 72703 United States, Illinois Methodist Medical Center Peoria, Illinois, United States, 61602 United States, Louisiana Willis-Knighton Physician Network Shreveport, Louisiana, United States, 71101 United States, Nebraska Pioneer Clinical Research Bellevue, Nebraska, United States, 68005 United States, Ohio PriMed Clinical Research Beavercreek, Ohio, United States, 45431 United States, Oregon Cyn3rgy Research Gresham, Oregon, United States, 97030 United States, South Carolina Coastal Clinical Research Charleston, South Carolina, United States, 29414 Coastal Pediatrics Associates - Mount Pleasant Mount Pleasant, South Carolina, United States, 29464 Spartanburg Medical Research Spartanburg, South Carolina, United States, 29303 United States, Texas 3rd Coast Research Associates Corpus Christi, Texas, United States, 78413 United States, Utah Bridgerland Clinical Research Logan, Utah, United States, 84341 Wee Care Pediatrics Syracuse, Utah, United States, 84075 United States, Virginia Pediatric Research of Charlottesville, LLC Charlottesville, Virginia, United States, 22902 Collapse << |
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