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CAS No.: 761439-42-3
Synonyms: TAE 684
NVP-TAE684 is a potent and selective ALK inhibitor with IC50 of 3 nM in a cell-free assay, 100-fold more sensitive for ALK than InsR.
生物活性
靶点 | ALK IC50:3nM |
实验方案
技术信息
CAS号 | 761439-42-3 | 储存条件 |
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分子式 | C30H40ClN7O3S | 运输 | 蓝冰 | |||||
分子量 | 614.20 | 别名 | TAE 684 | |||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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697 | - | Growth Inhibition Assay | - | IC50=0.43215 μM | SANGER |
8-MG-BA | - | Growth Inhibition Assay | - | IC50=2.65414 μM | SANGER |
A101D | - | Growth Inhibition Assay | - | IC50=1.57113 μM | SANGER |
A388 | - | Growth Inhibition Assay | - | IC50=2.9617 μM | SANGER |
A4-Fuk | - | Growth Inhibition Assay | - | IC50=0.05565 μM | SANGER |
A704 | - | Growth Inhibition Assay | - | IC50=1.32689 μM | SANGER |
ACN | - | Growth Inhibition Assay | - | IC50=9.19157 μM | SANGER |
ALL-PO | - | Growth Inhibition Assay | - | IC50=0.24524 μM | SANGER |
ARH-77 | - | Growth Inhibition Assay | - | IC50=4.11067 μM | SANGER |
ATN-1 | - | Growth Inhibition Assay | - | IC50=0.33303 μM | SANGER |
BB30-HNC | - | Growth Inhibition Assay | - | IC50=1.13112 μM | SANGER |
BB65-RCC | - | Growth Inhibition Assay | - | IC50=2.37493 μM | SANGER |
BC-3 | - | Growth Inhibition Assay | - | IC50=4.13068 μM | SANGER |
Becker | - | Growth Inhibition Assay | - | IC50=4.47336 μM | SANGER |
BL-41 | - | Growth Inhibition Assay | - | IC50=1.76272 μM | SANGER |
BL-70 | - | Growth Inhibition Assay | - | IC50=0.99535 μM | SANGER |
BOKU | - | Growth Inhibition Assay | - | IC50=2.72764 μM | SANGER |
BV-173 | - | Growth Inhibition Assay | - | IC50=3.64088 μM | SANGER |
C2BBe1 | - | Growth Inhibition Assay | - | IC50=1.29117 μM | SANGER |
CAS-1 | - | Growth Inhibition Assay | - | IC50=1.98299 μM | SANGER |
CESS | - | Growth Inhibition Assay | - | IC50=5.58034 μM | SANGER |
CHP-126 | - | Growth Inhibition Assay | - | IC50=0.85957 μM | SANGER |
CMK | - | Growth Inhibition Assay | - | IC50=0.2553 μM | SANGER |
COLO-320-HSR | - | Growth Inhibition Assay | - | IC50=0.19776 μM | SANGER |
COLO-800 | - | Growth Inhibition Assay | - | IC50=0.76695 μM | SANGER |
COLO-824 | - | Growth Inhibition Assay | - | IC50=10.8669 μM | SANGER |
CPC-N | - | Growth Inhibition Assay | - | IC50=1.85096 μM | SANGER |
CTB-1 | - | Growth Inhibition Assay | - | IC50=4.97721 μM | SANGER |
CTV-1 | - | Growth Inhibition Assay | - | IC50=0.55624 μM | SANGER |
D-263MG | - | Growth Inhibition Assay | - | IC50=8.55396 μM | SANGER |
D-283MED | - | Growth Inhibition Assay | - | IC50=1.22379 μM | SANGER |
D-336MG | - | Growth Inhibition Assay | - | IC50=0.66169 μM | SANGER |
Daudi | - | Growth Inhibition Assay | - | IC50=1.78967 μM | SANGER |
DEL | - | Growth Inhibition Assay | - | IC50=0.000927 μM | SANGER |
DMS-114 | - | Growth Inhibition Assay | - | IC50=2.61524 μM | SANGER |
DMS-153 | - | Growth Inhibition Assay | - | IC50=4.66475 μM | SANGER |
DOHH-2 | - | Growth Inhibition Assay | - | IC50=0.31204 μM | SANGER |
DSH1 | - | Growth Inhibition Assay | - | IC50=10.3972 μM | SANGER |
DU-4475 | - | Growth Inhibition Assay | - | IC50=1.45853 μM | SANGER |
EB-3 | - | Growth Inhibition Assay | - | IC50=5.17504 μM | SANGER |
ECC4 | - | Growth Inhibition Assay | - | IC50=3.7756 μM | SANGER |
EKVX | - | Growth Inhibition Assay | - | IC50=8.47066 μM | SANGER |
EM-2 | - | Growth Inhibition Assay | - | IC50=1.851 μM | SANGER |
ES1 | - | Growth Inhibition Assay | - | IC50=2.81804 μM | SANGER |
ES4 | - | Growth Inhibition Assay | - | IC50=0.49109 μM | SANGER |
ES6 | - | Growth Inhibition Assay | - | IC50=0.77559 μM | SANGER |
ES8 | - | Growth Inhibition Assay | - | IC50=0.74975 μM | SANGER |
ETK-1 | - | Growth Inhibition Assay | - | IC50=1.34489 μM | SANGER |
EVSA-T | - | Growth Inhibition Assay | - | IC50=10.3192 μM | SANGER |
EW-1 | - | Growth Inhibition Assay | - | IC50=0.10256 μM | SANGER |
EW-11 | - | Growth Inhibition Assay | - | IC50=9.65396 μM | SANGER |
EW-16 | - | Growth Inhibition Assay | - | IC50=0.10568 μM | SANGER |
EW-24 | - | Growth Inhibition Assay | - | IC50=3.66434 μM | SANGER |
EW-3 | - | Growth Inhibition Assay | - | IC50=4.76248 μM | SANGER |
GB-1 | - | Growth Inhibition Assay | - | IC50=0.38867 μM | SANGER |
GCIY | - | Growth Inhibition Assay | - | IC50=0.95526 μM | SANGER |
GDM-1 | - | Growth Inhibition Assay | - | IC50=0.47116 μM | SANGER |
GI-1 | - | Growth Inhibition Assay | - | IC50=1.09798 μM | SANGER |
GI-ME-N | - | Growth Inhibition Assay | - | IC50=1.25208 μM | SANGER |
GR-ST | - | Growth Inhibition Assay | - | IC50=1.38757 μM | SANGER |
GT3TKB | - | Growth Inhibition Assay | - | IC50=2.39972 μM | SANGER |
HAL-01 | - | Growth Inhibition Assay | - | IC50=1.15283 μM | SANGER |
HC-1 | - | Growth Inhibition Assay | - | IC50=3.62028 μM | SANGER |
HCC1187 | - | Growth Inhibition Assay | - | IC50=1.86241 μM | SANGER |
HCC2157 | - | Growth Inhibition Assay | - | IC50=1.46659 μM | SANGER |
HCE-4 | - | Growth Inhibition Assay | - | IC50=1.6085 μM | SANGER |
HCE-T | - | Growth Inhibition Assay | - | IC50=1.08819 μM | SANGER |
HD-MY-Z | - | Growth Inhibition Assay | - | IC50=3.13203 μM | SANGER |
HEL | - | Growth Inhibition Assay | - | IC50=1.14895 μM | SANGER |
HL-60 | - | Growth Inhibition Assay | - | IC50=0.48142 μM | SANGER |
HOP-62 | - | Growth Inhibition Assay | - | IC50=0.65033 μM | SANGER |
HT-144 | - | Growth Inhibition Assay | - | IC50=1.6319 μM | SANGER |
HUTU-80 | - | Growth Inhibition Assay | - | IC50=0.47375 μM | SANGER |
IST-MES1 | - | Growth Inhibition Assay | - | IC50=0.98824 μM | SANGER |
IST-SL1 | - | Growth Inhibition Assay | - | IC50=8.89892 μM | SANGER |
IST-SL2 | - | Growth Inhibition Assay | - | IC50=2.12445 μM | SANGER |
K052 | - | Growth Inhibition Assay | - | IC50=10.9322 μM | SANGER |
K5 | - | Growth Inhibition Assay | - | IC50=1.06274 μM | SANGER |
KALS-1 | - | Growth Inhibition Assay | - | IC50=1.3408 μM | SANGER |
KARPAS-299 | - | Growth Inhibition Assay | - | IC50=0.02384 μM | SANGER |
KARPAS-422 | - | Growth Inhibition Assay | - | IC50=1.10022 μM | SANGER |
KARPAS-45 | - | Growth Inhibition Assay | - | IC50=0.84263 μM | SANGER |
KASUMI-1 | - | Growth Inhibition Assay | - | IC50=9.7877 μM | SANGER |
KE-37 | - | Growth Inhibition Assay | - | IC50=4.86196 μM | SANGER |
KG-1 | - | Growth Inhibition Assay | - | IC50=0.39561 μM | SANGER |
KGN | - | Growth Inhibition Assay | - | IC50=0.66168 μM | SANGER |
KINGS-1 | - | Growth Inhibition Assay | - | IC50=10.2347 μM | SANGER |
KM12 | - | Growth Inhibition Assay | - | IC50=3.33544 μM | SANGER |
KM-H2 | - | Growth Inhibition Assay | - | IC50=5.05323 μM | SANGER |
KMOE-2 | - | Growth Inhibition Assay | - | IC50=5.58659 μM | SANGER |
KP-N-RT-BM-1 | - | Growth Inhibition Assay | - | IC50=0.33123 μM | SANGER |
KS-1 | - | Growth Inhibition Assay | - | IC50=0.19343 μM | SANGER |
KU812 | - | Growth Inhibition Assay | - | IC50=6.42791 μM | SANGER |
KURAMOCHI | - | Growth Inhibition Assay | - | IC50=1.69573 μM | SANGER |
L-363 | - | Growth Inhibition Assay | - | IC50=0.82375 μM | SANGER |
L-540 | - | Growth Inhibition Assay | - | IC50=0.36988 μM | SANGER |
LAMA-84 | - | Growth Inhibition Assay | - | IC50=2.79912 μM | SANGER |
LAN-6 | - | Growth Inhibition Assay | - | IC50=0.17443 μM | SANGER |
LB1047-RCC | - | Growth Inhibition Assay | - | IC50=0.54549 μM | SANGER |
LB2241-RCC | - | Growth Inhibition Assay | - | IC50=0.9884 μM | SANGER |
LB647-SCLC | - | Growth Inhibition Assay | - | IC50=1.34986 μM | SANGER |
LB771-HNC | - | Growth Inhibition Assay | - | IC50=0.89757 μM | SANGER |
LB831-BLC | - | Growth Inhibition Assay | - | IC50=0.55023 μM | SANGER |
LB996-RCC | - | Growth Inhibition Assay | - | IC50=0.69389 μM | SANGER |
LC-2-ad | - | Growth Inhibition Assay | - | IC50=0.19692 μM | SANGER |
LOXIMVI | - | Growth Inhibition Assay | - | IC50=2.06786 μM | SANGER |
LP-1 | - | Growth Inhibition Assay | - | IC50=1.87143 μM | SANGER |
LS-1034 | - | Growth Inhibition Assay | - | IC50=0.6358 μM | SANGER |
LS-123 | - | Growth Inhibition Assay | - | IC50=1.51594 μM | SANGER |
LS-411N | - | Growth Inhibition Assay | - | IC50=0.67462 μM | SANGER |
LS-513 | - | Growth Inhibition Assay | - | IC50=2.22269 μM | SANGER |
LU-134-A | - | Growth Inhibition Assay | - | IC50=0.83912 μM | SANGER |
LU-65 | - | Growth Inhibition Assay | - | IC50=3.6871 μM | SANGER |
LXF-289 | - | Growth Inhibition Assay | - | IC50=1.03076 μM | SANGER |
MC116 | - | Growth Inhibition Assay | - | IC50=4.94126 μM | SANGER |
MDA-MB-134-VI | - | Growth Inhibition Assay | - | IC50=4.30601 μM | SANGER |
MEG-01 | - | Growth Inhibition Assay | - | IC50=4.27419 μM | SANGER |
MFH-ino | - | Growth Inhibition Assay | - | IC50=0.32523 μM | SANGER |
MHH-CALL-2 | - | Growth Inhibition Assay | - | IC50=0.02952 μM | SANGER |
MHH-PREB-1 | - | Growth Inhibition Assay | - | IC50=9.21219 μM | SANGER |
ML-2 | - | Growth Inhibition Assay | - | IC50=0.49031 μM | SANGER |
MMAC-SF | - | Growth Inhibition Assay | - | IC50=7.06492 μM | SANGER |
MN-60 | - | Growth Inhibition Assay | - | IC50=7.69215 μM | SANGER |
MOLT-16 | - | Growth Inhibition Assay | - | IC50=0.87589 μM | SANGER |
MOLT-4 | - | Growth Inhibition Assay | - | IC50=5.1183 μM | SANGER |
MONO-MAC-6 | - | Growth Inhibition Assay | - | IC50=0.33291 μM | SANGER |
MPP-89 | - | Growth Inhibition Assay | - | IC50=0.57884 μM | SANGER |
MRK-nu-1 | - | Growth Inhibition Assay | - | IC50=5.43633 μM | SANGER |
MSTO-211H | - | Growth Inhibition Assay | - | IC50=2.20041 μM | SANGER |
MV-4-11 | - | Growth Inhibition Assay | - | IC50=0.39446 μM | SANGER |
MZ1-PC | - | Growth Inhibition Assay | - | IC50=0.17835 μM | SANGER |
NALM-6 | - | Growth Inhibition Assay | - | IC50=0.90739 μM | SANGER |
NB1 | - | Growth Inhibition Assay | - | IC50=0.00162 μM | SANGER |
NB10 | - | Growth Inhibition Assay | - | IC50=1.57392 μM | SANGER |
NB13 | - | Growth Inhibition Assay | - | IC50=1.37293 μM | SANGER |
NB14 | - | Growth Inhibition Assay | - | IC50=0.43826 μM | SANGER |
NB17 | - | Growth Inhibition Assay | - | IC50=1.00639 μM | SANGER |
NB5 | - | Growth Inhibition Assay | - | IC50=1.58476 μM | SANGER |
NB6 | - | Growth Inhibition Assay | - | IC50=7.54899 μM | SANGER |
NB69 | - | Growth Inhibition Assay | - | IC50=0.31787 μM | SANGER |
NB7 | - | Growth Inhibition Assay | - | IC50=2.00555 μM | SANGER |
NCCIT | - | Growth Inhibition Assay | - | IC50=3.08862 μM | SANGER |
NCI-H1092 | - | Growth Inhibition Assay | - | IC50=8.01734 μM | SANGER |
NCI-H1304 | - | Growth Inhibition Assay | - | IC50=1.13338 μM | SANGER |
NCI-H1355 | - | Growth Inhibition Assay | - | IC50=0.55184 μM | SANGER |
NCI-H1395 | - | Growth Inhibition Assay | - | IC50=2.82012 μM | SANGER |
NCI-H1417 | - | Growth Inhibition Assay | - | IC50=4.28443 μM | SANGER |
NCI-H1522 | - | Growth Inhibition Assay | - | IC50=5.26322 μM | SANGER |
NCI-H1581 | - | Growth Inhibition Assay | - | IC50=2.11559 μM | SANGER |
NCI-H1648 | - | Growth Inhibition Assay | - | IC50=0.27855 μM | SANGER |
NCI-H187 | - | Growth Inhibition Assay | - | IC50=1.70036 μM | SANGER |
NCI-H1882 | - | Growth Inhibition Assay | - | IC50=1.2389 μM | SANGER |
NCI-H209 | - | Growth Inhibition Assay | - | IC50=8.64006 μM | SANGER |
NCI-H2126 | - | Growth Inhibition Assay | - | IC50=2.43674 μM | SANGER |
NCI-H2141 | - | Growth Inhibition Assay | - | IC50=5.14268 μM | SANGER |
NCI-H23 | - | Growth Inhibition Assay | - | IC50=4.87227 μM | SANGER |
NCI-H322M | - | Growth Inhibition Assay | - | IC50=7.33335 μM | SANGER |
NCI-H510A | - | Growth Inhibition Assay | - | IC50=3.18943 μM | SANGER |
NCI-H524 | - | Growth Inhibition Assay | - | IC50=1.64307 μM | SANGER |
NCI-H526 | - | Growth Inhibition Assay | - | IC50=2.19141 μM | SANGER |
NCI-H69 | - | Growth Inhibition Assay | - | IC50=1.55811 μM | SANGER |
NCI-H716 | - | Growth Inhibition Assay | - | IC50=1.07259 μM | SANGER |
NCI-H720 | - | Growth Inhibition Assay | - | IC50=1.36378 μM | SANGER |
NCI-H747 | - | Growth Inhibition Assay | - | IC50=0.4989 μM | SANGER |
NCI-N87 | - | Growth Inhibition Assay | - | IC50=3.2002 μM | SANGER |
NCI-SNU-1 | - | Growth Inhibition Assay | - | IC50=2.33256 μM | SANGER |
NCI-SNU-16 | - | Growth Inhibition Assay | - | IC50=0.72664 μM | SANGER |
NEC8 | - | Growth Inhibition Assay | - | IC50=0.41292 μM | SANGER |
NH-12 | - | Growth Inhibition Assay | - | IC50=4.96439 μM | SANGER |
NKM-1 | - | Growth Inhibition Assay | - | IC50=1.6866 μM | SANGER |
NMC-G1 | - | Growth Inhibition Assay | - | IC50=0.83233 μM | SANGER |
no-11 | - | Growth Inhibition Assay | - | IC50=5.47087 μM | SANGER |
NOMO-1 | - | Growth Inhibition Assay | - | IC50=2.17683 μM | SANGER |
NOS-1 | - | Growth Inhibition Assay | - | IC50=0.10294 μM | SANGER |
NTERA-S-cl-D1 | - | Growth Inhibition Assay | - | IC50=0.33396 μM | SANGER |
OCI-AML2 | - | Growth Inhibition Assay | - | IC50=0.48328 μM | SANGER |
OCUB-M | - | Growth Inhibition Assay | - | IC50=1.36143 μM | SANGER |
ONS-76 | - | Growth Inhibition Assay | - | IC50=2.63641 μM | SANGER |
OPM-2 | - | Growth Inhibition Assay | - | IC50=0.22669 μM | SANGER |
OS-RC-2 | - | Growth Inhibition Assay | - | IC50=2.42341 μM | SANGER |
OVCAR-4 | - | Growth Inhibition Assay | - | IC50=0.40569 μM | SANGER |
PF-382 | - | Growth Inhibition Assay | - | IC50=1.5696 μM | SANGER |
PSN1 | - | Growth Inhibition Assay | - | IC50=0.19631 μM | SANGER |
QIMR-WIL | - | Growth Inhibition Assay | - | IC50=3.32849 μM | SANGER |
RCC10RGB | - | Growth Inhibition Assay | - | IC50=7.22977 μM | SANGER |
REH | - | Growth Inhibition Assay | - | IC50=6.25618 μM | SANGER |
RKO | - | Growth Inhibition Assay | - | IC50=1.49922 μM | SANGER |
RL95-2 | - | Growth Inhibition Assay | - | IC50=0.50112 μM | SANGER |
RPMI-8226 | - | Growth Inhibition Assay | - | IC50=0.63526 μM | SANGER |
RXF393 | - | Growth Inhibition Assay | - | IC50=0.55794 μM | SANGER |
SCC-3 | - | Growth Inhibition Assay | - | IC50=0.0000603 μM | SANGER |
SCLC-21H | - | Growth Inhibition Assay | - | IC50=3.26859 μM | SANGER |
SF126 | - | Growth Inhibition Assay | - | IC50=1.11568 μM | SANGER |
SF268 | - | Growth Inhibition Assay | - | IC50=0.84042 μM | SANGER |
SF539 | - | Growth Inhibition Assay | - | IC50=0.000564 μM | SANGER |
SH-4 | - | Growth Inhibition Assay | - | IC50=3.28797 μM | SANGER |
SIG-M5 | - | Growth Inhibition Assay | - | IC50=0.29159 μM | SANGER |
SJSA-1 | - | Growth Inhibition Assay | - | IC50=0.63725 μM | SANGER |
SK-LMS-1 | - | Growth Inhibition Assay | - | IC50=1.15974 μM | SANGER |
SK-MEL-2 | - | Growth Inhibition Assay | - | IC50=10.9939 μM | SANGER |
SK-MM-2 | - | Growth Inhibition Assay | - | IC50=0.41609 μM | SANGER |
SK-N-DZ | - | Growth Inhibition Assay | - | IC50=1.78309 μM | SANGER |
SK-NEP-1 | - | Growth Inhibition Assay | - | IC50=0.23524 μM | SANGER |
SK-N-FI | - | Growth Inhibition Assay | - | IC50=6.60674 μM | SANGER |
SK-PN-DW | - | Growth Inhibition Assay | - | IC50=1.26348 μM | SANGER |
SK-UT-1 | - | Growth Inhibition Assay | - | IC50=2.47467 μM | SANGER |
SNB75 | - | Growth Inhibition Assay | - | IC50=4.2619 μM | SANGER |
SNU-C2B | - | Growth Inhibition Assay | - | IC50=2.03351 μM | SANGER |
SR | - | Growth Inhibition Assay | - | IC50=0.00277 μM | SANGER |
ST486 | - | Growth Inhibition Assay | - | IC50=3.53883 μM | SANGER |
SU-DHL-1 | - | Growth Inhibition Assay | - | IC50=0.04865 μM | SANGER |
SW872 | - | Growth Inhibition Assay | - | IC50=0.56724 μM | SANGER |
SW954 | - | Growth Inhibition Assay | - | IC50=1.19567 μM | SANGER |
SW962 | - | Growth Inhibition Assay | - | IC50=1.5613 μM | SANGER |
SW982 | - | Growth Inhibition Assay | - | IC50=0.16478 μM | SANGER |
TE-1 | - | Growth Inhibition Assay | - | IC50=0.69074 μM | SANGER |
TE-10 | - | Growth Inhibition Assay | - | IC50=0.71496 μM | SANGER |
TE-11 | - | Growth Inhibition Assay | - | IC50=0.16096 μM | SANGER |
TE-12 | - | Growth Inhibition Assay | - | IC50=0.53349 μM | SANGER |
TE-15 | - | Growth Inhibition Assay | - | IC50=0.51124 μM | SANGER |
TE-6 | - | Growth Inhibition Assay | - | IC50=2.1905 μM | SANGER |
TE-8 | - | Growth Inhibition Assay | - | IC50=0.4288 μM | SANGER |
TE-9 | - | Growth Inhibition Assay | - | IC50=1.11328 μM | SANGER |
TGBC1TKB | - | Growth Inhibition Assay | - | IC50=4.68515 μM | SANGER |
TGBC24TKB | - | Growth Inhibition Assay | - | IC50=0.30218 μM | SANGER |
TGW | - | Growth Inhibition Assay | - | IC50=0.85863 μM | SANGER |
TK10 | - | Growth Inhibition Assay | - | IC50=1.05063 μM | SANGER |
U-266 | - | Growth Inhibition Assay | - | IC50=1.73842 μM | SANGER |
VA-ES-BJ | - | Growth Inhibition Assay | - | IC50=2.01513 μM | SANGER |
靶点 | Description | IC50 |
---|---|---|
ALK | IC50:3nM |
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