400-920-2911 sales@csnpharm.cn
CAS No.: 106566-58-9
Synonyms: AS101;IVX-Q-101;PRX-0001
AS101 is a potent Caspase-1 inhibitor which can inhibit IL-10 synthesis and potentiates IL-1α, IL-2 and TNF-α release through Caspase, performing as an immunomodulator.
生物活性
动物研究 | |
剂量 | Mice: 0.5 mg/kg, 1 mg/kg (i.p.) Rat: 0.25 mg/kg - 1 mg/kg[2] (i.p.) |
给药途径 | i.p. |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03666481 | Morbid Obesity ... more >> Bariatric Surgery Candidate Collapse << | Not Applicable | Completed | - | Spain ... more >> Sport Research Center. Miguel Hernández University of Elche. Elche, Alicante, Spain, 03202 Collapse << |
NCT01056159 | Asthma | Phase 1 | Completed | - | United States, California ... more >> Teva Clinical Study Site Los Angeles, California, United States, 90025 Teva Clinical Study Site Los Angeles, California, United States, 90048 United States, Colorado Teva Clinical Study Site Denver, Colorado, United States, 80230 Teva Clinical Study Site Lakewood, Colorado, United States, 80401 United States, Illinois Teva Clinical Study Site Normal, Illinois, United States, 61761 United States, Massachusetts Teva Clinical Study Site North Dartmouth, Massachusetts, United States, 02747 United States, Minnesota Teva Clinical Study Site Minneapolis, Minnesota, United States, 55402 United States, Nebraska Teva Clinical Study Site Bellevue, Nebraska, United States, 68123 United States, Oregon Teva Clinical Study Site Lake Oswego, Oregon, United States, 97035 Collapse << |
NCT02030457 | Pharmacokinetics | Phase 1 | Completed | - | United States, Texas ... more >> Teva Investigational Site San Antonio, Texas, United States Collapse << |
实验方案
技术信息
CAS号 | 106566-58-9 | 储存条件 |
|
|||||
分子式 | C2H8Cl3NO2Te | 运输 | 蓝冰 | |||||
分子量 | 312.05 | 别名 | AS101;IVX-Q-101;PRX-0001;PRX-0002;PRX-001;WAX-120337 | |||||
溶解度 |
|
动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03666481 | Morbid Obesity ... more >> Bariatric Surgery Candidate Collapse << | Not Applicable | Completed | - | Spain ... more >> Sport Research Center. Miguel Hernández University of Elche. Elche, Alicante, Spain, 03202 Collapse << |
NCT01056159 | Asthma | Phase 1 | Completed | - | United States, California ... more >> Teva Clinical Study Site Los Angeles, California, United States, 90025 Teva Clinical Study Site Los Angeles, California, United States, 90048 United States, Colorado Teva Clinical Study Site Denver, Colorado, United States, 80230 Teva Clinical Study Site Lakewood, Colorado, United States, 80401 United States, Illinois Teva Clinical Study Site Normal, Illinois, United States, 61761 United States, Massachusetts Teva Clinical Study Site North Dartmouth, Massachusetts, United States, 02747 United States, Minnesota Teva Clinical Study Site Minneapolis, Minnesota, United States, 55402 United States, Nebraska Teva Clinical Study Site Bellevue, Nebraska, United States, 68123 United States, Oregon Teva Clinical Study Site Lake Oswego, Oregon, United States, 97035 Collapse << |
NCT02030457 | Pharmacokinetics | Phase 1 | Completed | - | United States, Texas ... more >> Teva Investigational Site San Antonio, Texas, United States Collapse << |
NCT03626012 | Amyotrophic Lateral Sclerosis | Phase 1 | Recruiting | July 11, 2022 | United States, California ... more >> Research Site Active, not recruiting La Jolla, California, United States, 92037 United States, Maryland Research Site Active, not recruiting Baltimore, Maryland, United States, 21287 United States, Massachusetts Research Site Active, not recruiting Boston, Massachusetts, United States, 02114 Research Site Recruiting Cambridge, Massachusetts, United States, 02142 United States, Tennessee Research Site Active, not recruiting Knoxville, Tennessee, United States, 37920 Collapse << |
NCT00002013 | HIV Infections | Not Applicable | Completed | - | United States, California ... more >> Los Angeles County - USC Med Ctr Los Angeles, California, United States, 900331084 Collapse << |
NCT02623699 | Amyotrophic Lateral Sclerosis | Phase 1 | Active, not recruiting | March 19, 2019 | United States, Arizona ... more >> Barrow Neurological Institute Phoenix, Arizona, United States, 85013 United States, California University of California San Diego Medical Center La Jolla, California, United States, 92093-0949 California Pacific Medical Center San Francisco, California, United States, 94115 United States, Florida Compass Research, LLC Orlando, Florida, United States, 32806 United States, Georgia The Emory Clinic Atlanta, Georgia, United States, 30322 United States, Maryland Johns Hopkins Hospital Baltimore, Maryland, United States, 21287 United States, Massachusetts Massachusetts General Hospital, MA Boston, Massachusetts, United States, 02114 United States, Missouri Washington University School of Medicine Saint Louis, Missouri, United States, 63110 United States, Tennessee Volunteer Research Group, LLC Knoxville, Tennessee, United States, 37920 Belgium UZ Leuven Leuven, Belgium, 3000 Canada, Ontario Sunnybrook Health Sciences Centre Toronto, Ontario, Canada, M4N 3M5 Canada, Quebec Montreal Neurological Institute Clinical Research Unit Montreal, Quebec, Canada, H3A 2B4 France Groupe Hospitalier Pitie-Salpetriere Paris, France, 75651 Germany Universitaetsklinikum Ulm Ulm, Baden Wuerttemberg, Germany, 89081 Italy Università degli Studi di Torino Torino, Italy, 10126 Sweden Norrlands universitetssjukhus Umea, Sweden, 90185 United Kingdom Sheffield Institute for Translational Neuroscience Sheffield, South Yorkshire, United Kingdom, S10 2HQ Collapse << |
NCT00002033 | HIV Infections | Not Applicable | Completed | - | Brazil ... more >> Escola Paulista De-Medicina Sao Paulo, Brazil Faculdade De-Ciencias Medica Da Sao Paulo, Brazil Hosp De-Servidor Publico Estadual Sao Paulo, Brazil Instituto Do Cancer Arnaldo Vieiro Sao Paulo, Brazil Collapse << |
NCT00418249 | Alopecia | Phase 2 | Unknown | - | Israel ... more >> Not yet recruiting Tel Aviv, Israel Contact: Danny Ben Amitai 972-3-9253770 Collapse << |
NCT00001006 | HIV Infections | Phase 1 | Completed | - | United States, New York ... more >> Mount Sinai Med Ctr New York, New York, United States, 10029 Collapse << |
NCT00002266 | HIV Infections | Not Applicable | Completed | - | United States, Arizona ... more >> Univ of Arizona / Health Science Ctr Tucson, Arizona, United States, 85724 Collapse << |
NCT00788424 | Mild to Moderate Psoriasis | Phase 2 | Withdrawn(Sponsor's considerat... more >>ions) Collapse << | - | Israel ... more >> Hadassah Medical Organization Jerusalem, Israel Collapse << |
NCT00926354 | Chemotherapy Induced Thrombocy... more >>topenia Collapse << | Phase 2 | Terminated(Sponsor's considera... more >>tions) Collapse << | - | Israel ... more >> Meir Medical Center Kfar Saba, Israel Collapse << |
NCT01010373 | Acute Myeloid Leukemia ... more >> Myelodysplastic Syndrome Collapse << | Phase 2 | Suspended(The sponsor is curre... more >>ntly focusing on different indications) Collapse << | January 2016 | Israel ... more >> Sheba Medical Center Tel Hashomer, Israel Collapse << |
NCT01555112 | Wart; External Genital Organs ... more >> Condyloma Acuminata Collapse << | Phase 1 Phase 2 | Completed | - | Israel ... more >> Gynecology department, Haemek MC Afula, Israel Collapse << |
NCT03216538 | Neovascular Age-related Macula... more >>r Degeneration Collapse << | Phase 1 Phase 2 | Recruiting | March 2019 | Israel ... more >> Meir MC Recruiting Kfar Saba, Israel Contact: Joseph Ferencz, MD 054-6312518 j@ferencz.info Collapse << |
NCT01943630 | External Genital Warts | Phase 2 | Unknown | May 2017 | Israel ... more >> Ha'Emek Medical Center, Department of Gynecology and obstetrics Recruiting Afula, Israel, 1834111 Contact: Shabtai Romano, MD +972-4-6494331 shabtai_r@clalit.org.il Contact papillomatrial@gmail.com Principal Investigator: Shabtai Romano, MD Sub-Investigator: Moshe Bustan, MD Kaplan Medical Center, Department of Gynecology Recruiting Rehovot, Israel, 76100 Contact: Alon Ben-Arie, MD 972-8-9441325 Alon_B@clalit.org.il Contact Papillomatrial@gmail.com Principal Investigator: Alon Ben-Arie, MD Sub-Investigator: Dora Milman, MD Ziv Medical Center, Department of Gynecology and obstetrics Recruiting Safed, Israel, 13100 Contact: Inbar Ben-Shachar, MD 972-4-6828959 Inbar.b@ziv.health.gov.il Contact Papillomatrial@gmail.com Principal Investigator: Inbar Ben-Shachar, MD Sub-Investigator: David Peleg, MD Tel-Aviv Sourasky Medical Center, Department of Gynecology Recruiting Tel-Aviv, Israel, 64239 Contact: Dan Grisaru, MD PhD +972-3-6925604 dangr@tlvmc.gov.il Contact Papillomatrial@gmail.com Principal Investigator: Dan Grisaru, MD PhD Prof Sub-Investigator: Jacob Niv, MD Sub-Investigator: Yifat Oxhorn, MD Collapse << |
NCT00927212 | Atopic Dermatitis | Phase 2 | Terminated(The trial started a... more >>nd halted due sponsor's considerations.) Collapse << | - | Israel ... more >> Dermatology department, Sheba Medical Center Ramat-Gan, Israel Collapse << |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网