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CAS No.: 198474-05-4
Synonyms: EOS200271;PF-0684003
PF-06840003 is a highly selective orally bioavailable IDO-1 inhibitor with IC50 of 0.41 μM.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02764151 | Oligodendroglioma ... more >> Astrocytoma Malignant Glioma Collapse << | Phase 1 | Active, not recruiting | December 26, 2018 | United States, California ... more >> Ronald Reagan UCLA Medical Center, Drug Information Center Los Angeles, California, United States, 90095-6894 Ronald Reagan UCLA Medical Center Los Angeles, California, United States, 90095-6894 UCLA Clinical & Translational Research Center Los Angeles, California, United States, 90095 UCLA Oncology Center Los Angeles, California, United States, 90095 UCLA School of Medicine Los Angeles, California, United States, 90095 United States, Massachusetts Massachusetts General Hospital Boston, Massachusetts, United States, 02114 Dana-Farber Cancer Institute Boston, Massachusetts, United States, 02215 United States, New Mexico University of New Mexico Comprehensive Cancer Center Albuquerque, New Mexico, United States, 87102 United States, New York Columbia University Medical Center New York, New York, United States, 10019 Columbia University Medical Center New York, New York, United States, 10032 CUMC Research Pharmacy New York, New York, United States, 10032 Columbia Doctors Tarrytown Tarrytown, New York, United States, 10591 United States, North Carolina Duke Cancer Center Durham, North Carolina, United States, 27710 Duke University Medical Center, Duke Cancer Center Durham, North Carolina, United States, 27710 Collapse << |
实验方案
技术信息
CAS号 | 198474-05-4 | 储存条件 |
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分子式 | C12H9FN2O2 | 运输 | 蓝冰 | |||||||
分子量 | 232.21 | 别名 | EOS200271;PF-0684003 | |||||||
溶解度 |
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动物实验配方 |