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CAS No.: 874101-00-5
Synonyms: CH4987655
RO4987655 is an orally active small molecule, targeting mitogen-activated protein kinase kinase 1 (MAP2K1/MEK1 IC50=5.2 nM), with potential antineoplastic activity.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00817518 | Neoplasms | Phase 1 | Completed | - | France ... more >> Marseille, France, 13385 Paris, France, 75231 Paris, France, 75651 Villejuif, France, 94805 Germany Essen, Germany, 45122 Netherlands Amsterdam, Netherlands, 1066 CX Spain Barcelona, Spain, 08003 Madrid, Spain, 28050 Sevilla, Spain, 41013 United Kingdom Cambridge, United Kingdom, CB2 2QQ London, United Kingdom, SW3 6JJ Oxford, United Kingdom, OX3 7LJ Collapse << |
实验方案
技术信息
CAS号 | 874101-00-5 | 储存条件 |
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分子式 | C20H19F3IN3O5 | 运输 | 蓝冰 | |||
分子量 | 565.28 | 别名 | CH4987655 | |||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00817518 | Neoplasms | Phase 1 | Completed | - | France ... more >> Marseille, France, 13385 Paris, France, 75231 Paris, France, 75651 Villejuif, France, 94805 Germany Essen, Germany, 45122 Netherlands Amsterdam, Netherlands, 1066 CX Spain Barcelona, Spain, 08003 Madrid, Spain, 28050 Sevilla, Spain, 41013 United Kingdom Cambridge, United Kingdom, CB2 2QQ London, United Kingdom, SW3 6JJ Oxford, United Kingdom, OX3 7LJ Collapse << |
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