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CAS No.: 923359-38-0

SAR407899 Catalog No. CSN18583

Synonyms: SAR407899

SAR407899 is a potent, ATP-competitive ROCK inhibitor woth Ki value of 36 nM/41 nM for human ROCK/Rat ROCK respectively.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 靶点ROCK

    Ki:36nM
    ROCK (rat)

    Ki:41nM
  • 描述
  • 动物研究
    剂量

    Rat: 3 mg/kg[2] (i.v.); 1 mg/kg - 30 mg/kg[2] (p.o.)

    给药途径

    i.v., p.o.

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT01485900Chronic Kidney DiseasePhase 1Completed-Moldova, Republic of ... more >> Investigational Site Number 498002 Chisinau, Moldova, Republic of, 2025 Romania Investigational Site Number 642001 Bucuresti, Romania Collapse <<
    NCT00914277Erectile DysfunctionPhase 2Completed-France ... more >> Sanofi-Aventis Administrative Office Paris, France Collapse <<
    NCT03236311Microvascular Coronary Artery ... more >>Disease Collapse <<Phase 2Terminated((Recruitment was ea... more >>rly terminated due to slow recruitment. Not linked to any safety concern.)) Collapse <<-United States, California ... more >> Investigational Site Number 8400003 Los Angeles, California, United States, 90048 United States, Florida Investigational Site Number 8400001 Jacksonville, Florida, United States, 32209 Investigational Site Number 8400013 Wellington, Florida, United States, 33449 United States, Maryland Investigational Site Number 8400008 Baltimore, Maryland, United States, 21287 United States, Massachusetts Investigational Site Number 8400006 Boston, Massachusetts, United States, 02115 United States, Pennsylvania Investigational Site Number 8400010 Philadelphia, Pennsylvania, United States, 19104 Denmark Investigational Site Number 2080001 København Nv, Denmark, 2400 Korea, Republic of Investigational Site Number 4100002 Seoul, Korea, Republic of, 03722 Investigational Site Number 4100003 Seoul, Korea, Republic of, 06351 Netherlands Investigational Site Number 5280001 Nijmegen, Netherlands, 6525 GA Sweden Investigational Site Number 7520001 Lund, Sweden, 221 85 Collapse <<
  • 参考文献

实验方案

技术信息

CAS号 923359-38-0 储存条件
分子式 C14H16N2O2 运输 蓝冰
分子量 244.29 别名 SAR407899
溶解度
DMSO6.0 mg/mL (24.6 mM)
动物实验配方

大规格询价

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