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CAS No.: 1456632-41-9
Synonyms: SH5-07
SH5-07 is an inhibitor of STAT3 with IC50 of 3.9±0.6 μM with antitumor effects and it can suppresse human glioma and breast cancer.
生物活性
实验方案
技术信息
CAS号 | 1456632-41-9 | 储存条件 |
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分子式 | C29H28F5N3O5S | 运输 | 蓝冰 | |||||
分子量 | 625.61 | 别名 | SH5-07 | |||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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127EF cells | - | Cytotoxicity assay | - | Cytotoxicity against human 127EF cells assessed as cell viability after 3 days by Alamar Blue assay, IC50=0.1955 μM | 24900612 |
147EF cells | - | Function assay | 2 to 72 hrs | Inhibition of STAT3 in human 147EF cells assessed as reduction of phosphorylated Bcl-xL level after 2 to 72 hrs by Western blotting analysis | 24900612 |
25EF cells | - | Cytotoxicity assay | - | Cytotoxicity against human 25EF cells assessed as cell viability after 3 days by Alamar Blue assay, IC50=1.1205 μM | 24900612 |
30M cells | - | Cytotoxicity assay | - | Cytotoxicity against human 30M cells assessed as cell viability after 3 days by Alamar Blue assay, IC50=0.1 μM | 24900612 |
67EF cells | - | Cytotoxicity assay | - | Cytotoxicity against human 67EF cells assessed as cell viability after 3 days by Alamar Blue assay, IC50=0.2145 μM | 24900612 |
73EF cells | - | Cytotoxicity assay | - | Cytotoxicity against human 73EF cells assessed as cell viability after 3 days by Alamar Blue assay, IC50=0.8635 μM | 24900612 |
84EF cells | - | Cytotoxicity assay | - | Cytotoxicity against human 84EF cells assessed as cell viability after 3 days by Alamar Blue assay, IC50=0.295 μM | 24900612 |
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