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CAS No.: 1636180-98-7

Tarloxotinib bromide Catalog No. CSN26545

Synonyms: TH-4000;PR-610;Hypoxin

Tarloxotinib bromide, also known TH-4000 or PR-610, is a prodrug designed to selectively release a covalent (irreversible) EGFR tyrosine kinase inhibitor under severe hypoxia, a feature of many solid tumors. Tarloxotinib has the potential to effectively shut down aberrant EGFR signaling in a tumor-selective manner, thus potentially avoiding or reducing the systemic side effects associated with currently available EGFR tyrosine kinase inhibitors.

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CAS号 1636180-98-7 储存条件
分子式 C24H24Br2ClN9O3 运输 蓝冰
分子量 681.77 别名 TH-4000;PR-610;Hypoxin;Tarloxotinib

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