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CAS No.: 1636180-98-7
Synonyms: TH-4000;PR-610;Hypoxin
Tarloxotinib bromide, also known TH-4000 or PR-610, is a prodrug designed to selectively release a covalent (irreversible) EGFR tyrosine kinase inhibitor under severe hypoxia, a feature of many solid tumors. Tarloxotinib has the potential to effectively shut down aberrant EGFR signaling in a tumor-selective manner, thus potentially avoiding or reducing the systemic side effects associated with currently available EGFR tyrosine kinase inhibitors.
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技术信息
CAS号 | 1636180-98-7 | 储存条件 |
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分子式 | C24H24Br2ClN9O3 | 运输 | 蓝冰 | |
分子量 | 681.77 | 别名 | TH-4000;PR-610;Hypoxin;Tarloxotinib |
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