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CAS No.: 1361951-15-6
Synonyms: TP-3654
TP-3654 is a selective Pim kinase inhibitor with Ki values of 5nM, 239nM and 42nM for Pim-1, Pim-2 and Pim-3, respectively, as well as with an average EC50 of 67nM for cellular PIM-1 inhibition in the PIM-1/BAD overexpression system and with moderate potency to FLT3.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03715504 | Advanced Solid Tumors | Phase 1 | Not yet recruiting | March 2021 | United States, Utah ... more >> Huntsman Cancer Institute Not yet recruiting Salt Lake City, Utah, United States, 84112 Contact: Ignacio Garrido-Laguna, MD, PhD 801-585-0303 Principal Investigator: Ignacio Garrido-Laguna, MD, PhD Collapse << |
实验方案
技术信息
CAS号 | 1361951-15-6 | 储存条件 |
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分子式 | C22H25F3N4O | 运输 | 蓝冰 | |||||
分子量 | 418.46 | 别名 | TP-3654 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03715504 | Advanced Solid Tumors | Phase 1 | Not yet recruiting | March 2021 | United States, Utah ... more >> Huntsman Cancer Institute Not yet recruiting Salt Lake City, Utah, United States, 84112 Contact: Ignacio Garrido-Laguna, MD, PhD 801-585-0303 Principal Investigator: Ignacio Garrido-Laguna, MD, PhD Collapse << |
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