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CAS No.: 121584-18-7
Synonyms: PSC 833;SDZ PSC 833;伐司扑达
Valspodar is a P-glycoprotein (P-gp) inhibitor widely used in preclinical and clinical studies for overcoming multidrug resistance (MDR).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00005823 | Leukemia Myel... more >>odysplastic Syndromes Myelodysplastic/Myeloproliferative Neoplasms Collapse << | Phase 3 | Completed | - | United Kingdom ... more >> Queen Elizabeth Hospital at University of Birmingham Birmingham, England, United Kingdom, B15 2RR University College Hospital London, England, United Kingdom, WC1E 6AU University Hospital of Wales Cardiff, Wales, United Kingdom, CF14 4XN Collapse << |
NCT00972205 | - | - | Completed | - | - |
NCT00972205 | Cervical Ovar... more >>ian Lung Breast Renal Collapse << | Not Applicable | Completed | - | United States, Maryland ... more >> National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 Collapse << |
实验方案
技术信息
CAS号 | 121584-18-7 | 储存条件 |
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分子式 | C63H111N11O12 | 运输 | 蓝冰 | |
分子量 | 1214.62 | 别名 | PSC 833;SDZ PSC 833;伐司扑达 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00005823 | Leukemia Myel... more >>odysplastic Syndromes Myelodysplastic/Myeloproliferative Neoplasms Collapse << | Phase 3 | Completed | - | United Kingdom ... more >> Queen Elizabeth Hospital at University of Birmingham Birmingham, England, United Kingdom, B15 2RR University College Hospital London, England, United Kingdom, WC1E 6AU University Hospital of Wales Cardiff, Wales, United Kingdom, CF14 4XN Collapse << |
NCT00972205 | - | - | Completed | - | - |
NCT00972205 | Cervical Ovar... more >>ian Lung Breast Renal Collapse << | Not Applicable | Completed | - | United States, Maryland ... more >> National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 Collapse << |
NCT00002826 | Breast Cancer | Phase 2 | Completed | - | United States, California ... more >> Veterans Affairs Medical Center - Palo Alto Palo Alto, California, United States, 94304 Stanford University Medical Center Stanford, California, United States, 94305-5408 United States, New Jersey Hunterdon Regional Cancer Program Flemington, New Jersey, United States, 08822 Kimball Medical Center Lakewood, New Jersey, United States, 08701 Fox Chase Cancer Center at Virtua-Memorial Hospital Burlington County Mount Holly, New Jersey, United States, 08060 Cancer Institute of New Jersey New Brunswick, New Jersey, United States, 08901 St. Francis Medical Center Trenton, New Jersey, United States, 08629 United States, New York Albert Einstein Comprehensive Cancer Center Bronx, New York, United States, 10461 United States, Pennsylvania Fox Chase Cancer Center Philadelphia, Pennsylvania, United States, 19111 Collapse << |
NCT00002925 | Leukemia | Phase 1 Phase 2 | Completed | - | - |
NCT00002878 | Multiple Myeloma and Plasma Ce... more >>ll Neoplasm Collapse << | Phase 3 | Completed | - | - |
NCT00006363 | Adult Acute Basophilic Leukemi... more >>a Adult Acute Eosinophilic Leukemia Adult Acute Erythroid Leukemia (M6) Adult Acute Megakaryoblastic Leukemia (M7) Adult Acute Minimally Differentiated Myeloid Leukemia (M0) Adult Acute Monoblastic Leukemia (M5a) Adult Acute Monoblastic Leukemia and Acute Monocytic Leukemia (M5) Adult Acute Monocytic Leukemia (M5b) Adult Acute Myeloblastic Leukemia With Maturation (M2) Adult Acute Myeloblastic Leukemia Without Maturation (M1) Adult Acute Myeloid Leukemia With 11q23 (MLL) Abnormalities Adult Acute Myeloid Leukemia With Del(5q) Adult Acute Myeloid Leukemia With Inv(16)(p13;q22) Adult Acute Myeloid Leukemia With t(16;16)(p13;q22) Adult Acute Myeloid Leukemia With t(8;21)(q22;q22) Adult Acute Myelomonocytic Leukemia (M4) Adult Erythroleukemia (M6a) Adult Pure Erythroid Leukemia (M6b) Childhood Acute Basophilic Leukemia Childhood Acute Eosinophilic Leukemia Childhood Acute Erythroleukemia (M6) Childhood Acute Megakaryocytic Leukemia (M7) Childhood Acute Minimally Differentiated Myeloid Leukemia (M0) Childhood Acute Monoblastic Leukemia (M5a) Childhood Acute Monoblastic Leukemia and Acute Monocytic Leukemia (M5) Childhood Acute Monocytic Leukemia (M5b) Childhood Acute Myeloblastic Leukemia With Maturation (M2) Childhood Acute Myeloblastic Leukemia Without Maturation (M1) Childhood Acute Myelomonocytic Leukemia (M4) Childhood Myelodysplastic Syndromes de Novo Myelodysplastic Syndromes Untreated Adult Acute Myeloid Leukemia Untreated Childhood Acute Myeloid Leukemia and Other Myeloid Malignancies Collapse << | Phase 3 | Completed | - | United States, Illinois ... more >> Cancer and Leukemia Group B Chicago, Illinois, United States, 60606 Collapse << |
NCT00004217 | Leukemia | Phase 2 | Completed | - | - |
NCT00001383 | Breast Cancer ... more >> Cancer Carcinoma, Renal Cell Lymphoma Ovarian Cancer Collapse << | Phase 1 | Completed | - | United States, Maryland ... more >> National Cancer Institute (NCI) Bethesda, Maryland, United States, 20892 Collapse << |
NCT00001570 | Kidney Neoplasms ... more >> Neoplasm Metastasis Collapse << | Phase 1 | Completed | - | United States, Maryland ... more >> National Cancer Institute (NCI) Bethesda, Maryland, United States, 20892 Collapse << |
NCT00003190 | Adult Acute Megakaryoblastic L... more >>eukemia (M7) Adult Acute Minimally Differentiated Myeloid Leukemia (M0) Adult Acute Monoblastic Leukemia (M5a) Adult Acute Monocytic Leukemia (M5b) Adult Acute Myeloblastic Leukemia With Maturation (M2) Adult Acute Myeloblastic Leukemia Without Maturation (M1) Adult Acute Myeloid Leukemia With 11q23 (MLL) Abnormalities Adult Acute Myeloid Leukemia With Del(5q) Adult Acute Myeloid Leukemia With Inv(16)(p13;q22) Adult Acute Myeloid Leukemia With t(16;16)(p13;q22) Adult Acute Myeloid Leukemia With t(8;21)(q22;q22) Adult Acute Myelomonocytic Leukemia (M4) Adult Erythroleukemia (M6a) Adult Pure Erythroid Leukemia (M6b) Untreated Adult Acute Myeloid Leukemia Collapse << | Phase 3 | Completed | - | United States, Illinois ... more >> Cancer and Leukemia Group B Chicago, Illinois, United States, 60606 Collapse << |
NCT00001302 | Breast Cancer ... more >> Kidney Neoplasm Lymphoma Neoplasm Metastasis Ovarian Cancer Collapse << | Phase 1 | Completed | - | United States, Maryland ... more >> National Cancer Institute (NCI) Bethesda, Maryland, United States, 20892 Collapse << |
NCT00002937 | Breast Cancer | Phase 2 | Completed | - | United States, California ... more >> Beckman Research Institute, City of Hope Duarte, California, United States, 91010 USC/Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033-0800 University of California Davis Cancer Center Sacramento, California, United States, 95817 Canada, Ontario Toronto Sunnybrook Regional Cancer Centre Toronto, Ontario, Canada, M4N 3M5 Collapse << |
NCT00003207 | Sarcoma Unspe... more >>cified Adult Solid Tumor, Protocol Specific Collapse << | Phase 1 | Completed | - | United States, Missouri ... more >> Washington University School of Medicine Saint Louis, Missouri, United States, 63110 Collapse << |
NCT00002912 | Leukemia | Phase 1 | Completed | - | - |
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