400-920-2911
上海市杨浦区翔殷路128号1号楼101
RSK
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN20281 | SL0101 | 77307-50-7 | SL0101 is a selective inhibitor of ribosomal S6 kinase (RSK) (IC50 = 89 nM for RSK2) which does not inhibit upstream kinases such as MEK, Raf and PKC. SL0101 Inhibits the growth of MCF-7 human breast cancer cells with no effect on the normal breast cell line. |
| CSN15894 | PF-4708671 | 1255517-76-0 | PF-4708671 is an inhibitor of S6K1 (p70 ribosomal S6 kinase 1) with Ki and IC50 of 20 nM and 160 nM, respectively. |
| CSN17965 | LJI308 | 1627709-94-7 | LJI308 is a potent pan-RSK inhibitor, with IC50 of 6 nM, 4 nM, and 13 nM for RSK1, RSK2, and RSK3, respectively. |
| CSN17966 | LJH685 | 1627710-50-2 | LJH685 is a potent pan-RSK inhibitor with IC50 of 6 nM, 5 nM and 4 nM for RSK1, RSK2, and RSK3, respectively. |
| CSN12314 | BI-D1870 | 501437-28-1 | BI-D1870 is an inhibitor of S6 ribosome which can inhibit RSK1, RSK2, RSK3, RSK4 with IC50 of 31 nM, 24 nM, 18 nM and 15 nM, respectively. |