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SRPK
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN24738 | ZT-12-037-01 | 2328073-61-4 | ZT-12-037-01 is a potent and selective STK19 inhibitor with an IC50 value of 24.04nM |
| CSN19078 | WNK463 | 2012607-27-9 | WNK463 is a potant With-No-Lysine (WNK) kinase inhibitor with IC50s of 5/1/6/9 nM for WNK1/2/3/4. |
| CSN23723 | WNK-IN-11 | 2123489-30-3 | WNK-IN-11 is a potent, selective and orally active inhibitor of WNK1 kinase with IC50 of 6 nM. |
| CSN22078 | TMPA | 1258275-73-8 | TMPA is an antagonist of nuclear receptor Nur77 and LKB1 interaction. |
| CSN23884 | STK16-IN-1 | 1223001-53-3 | STK16-IN-1 is a serine/threonine protein kinase 16 (STK16) inhibitor with IC50 of 295 nM. |
| CSN13762 | SRPIN340 | 218156-96-8 | SRPIN340 is an inhibitor of serine/arginine-rich protein kinase SRPK1 with IC50 of 0.89 μM. |
| CSN23673 | SPHINX31 | 1818389-84-2 | SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kinase 1 (SRPK1), with an IC50 of 5.9 nM. SPHINX31 inhibits phosphorylation of serine/arginine-rich splicing factor 1 (SRSF1). SPHINX31 is a potential topical therapeutic for neovascular eye disease[1]. |
| CSN23063 | (Rac)-CCT 250863 | 1364269-06-6 | rac-CCT-250863 is a potent Nek2 inhibitor. exhibiting selectivity for Nek2 over PLK1, MPS1, Cdk2 and Aurora A. |
| CSN20434 | PROTAC TBK1 C3i | 2052306-13-3 | PROTAC TBK1 C3i is a potent hit (TBK1 DC50 = 12 nM, Dmax = 96%) with excellent selectivity against a related kinase IKKε, which was further used as a chemical tool to assess TBK1 as a target in mutant K-Ras cancer cells. |
| CSN17458 | Pim1/AKK1-IN-1 | 1093222-27-5 | Pim1 AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively and also inhibits MPSK1 and TNIK. |
| CSN23000 | Nek2-IN-5 | 1507367-00-1 | NCL 00017509 is a potent and reversible NIMA related kinase 2 (Nek2) inhibitor with IC50 of 56 nM. |
| CSN17802 | ML281 | 1404437-62-2 | ML281 is a potent and selective serine/threonine kinase (STK33) inhibitor with IC50 of 14 nM. STK33 downregulation is toxic to KRAS-dependent cancer cell lines. |
| CSN27205 | ILK-IN-3 | 6975-75-3 | ILK-IN-3 is an integrin linked kinase inhibitor. |
| CSN18951 | OSU-T315 | 2070015-22-2 | ILK-IN-2 is a ILK inhibitor. |
| CSN17699 | ILK-IN-2 | 1333146-24-9 | ILK-IN-1 is an ILK inhibitor with IC50 of 0.6 μM. |
| CSN24084 | GSK8612 | 2361659-62-1 | GSK8612 is a potent and highly selective Tank-binding Kinase-1 (TBK1) inhibitor with pIC50 of 6.8 for recombinant TBK1. |
| CSN25836 | CMPD101 | 865608-11-3 | CMPD101 is a selective GRK2/3 inhibitor with IC50 values of 32 and 54 nM for GRK3 and GRK2, respectively. |
| CSN20021 | Bryostatin 1 | 83314-01-6 | Bryostatin 1 is a Protein kinase C (PKC) activator that binds with high affinity (Ki = 1.35 nM). |
| CSN42722 | Belumosudil mesylate | 2109704-99-4 | Belumosudil is a small molecule and selective inhibitor of ROCK2 with IC50 of 105 nM, which is over 200 fold selecivity over ROCK1 (IC50 =24 μM). |
| CSN12528 | 4μ8C | 14003-96-4 | 4μ8C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM. |
| CSN106900 | N-((1-(2-(3-Methoxyphenyl)-5-methylpyridin-4-yl)-1H-indol-3-yl)methyl)-2-methylpropan-1-amine | 2125724-72-1 |
