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SRPK

SRPK

货号 产品名 CAS号 信息
CSN24738 ZT-12-037-01 2328073-61-4 ZT-12-037-01 is a potent and selective STK19 inhibitor with an IC50 value of 24.04nM
CSN19078 WNK463 2012607-27-9 WNK463 is a potant With-No-Lysine (WNK) kinase inhibitor with IC50s of 5/1/6/9 nM for WNK1/2/3/4.
CSN23723 WNK-IN-11 2123489-30-3 WNK-IN-11 is a potent, selective and orally active inhibitor of WNK1 kinase with IC50 of 6 nM.
CSN22078 TMPA 1258275-73-8 TMPA is an antagonist of nuclear receptor Nur77 and LKB1 interaction.
CSN23884 STK16-IN-1 1223001-53-3 STK16-IN-1 is a serine/threonine protein kinase 16 (STK16) inhibitor with IC50 of 295 nM.
CSN13762 SRPIN340 218156-96-8 SRPIN340 is an inhibitor of serine/arginine-rich protein kinase SRPK1 with IC50 of 0.89 μM.
CSN23673 SPHINX31 1818389-84-2 SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kinase 1 (SRPK1), with an IC50 of 5.9 nM. SPHINX31 inhibits phosphorylation of serine/arginine-rich splicing factor 1 (SRSF1). SPHINX31 is a potential topical therapeutic for neovascular eye disease[1].
CSN23063 (Rac)-CCT 250863 1364269-06-6 rac-CCT-250863 is a potent Nek2 inhibitor. exhibiting selectivity for Nek2 over PLK1, MPS1, Cdk2 and Aurora A.
CSN20434 PROTAC TBK1 degrader-2 2052306-13-3 PROTAC TBK1 C3i is a potent hit (TBK1 DC50 = 12 nM, Dmax = 96%) with excellent selectivity against a related kinase IKKε, which was further used as a chemical tool to assess TBK1 as a target in mutant K-Ras cancer cells.
CSN17458 Pim1/AKK1-IN-1 1093222-27-5 Pim1 AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively and also inhibits MPSK1 and TNIK.
CSN23000 Nek2-IN-5 1507367-00-1 NCL 00017509 is a potent and reversible NIMA related kinase 2 (Nek2) inhibitor with IC50 of 56 nM.
CSN17802 ML281 1404437-62-2 ML281 is a potent and selective serine/threonine kinase (STK33) inhibitor with IC50 of 14 nM. STK33 downregulation is toxic to KRAS-dependent cancer cell lines.
CSN27205 ILK-IN-3   6975-75-3 ILK-IN-3 is an integrin linked kinase inhibitor.
CSN18951 OSU-T315 2070015-22-2 ILK-IN-2 is a ILK inhibitor.
CSN17699 ILK-IN-2 1333146-24-9 ILK-IN-1 is an ILK inhibitor with IC50 of 0.6 μM.
CSN24084 4-(((5-Bromo-2-((3-methyl-1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)amino)methyl)benzenesulfonamide 2361659-62-1 GSK8612 is a potent and highly selective Tank-binding Kinase-1 (TBK1) inhibitor with pIC50 of 6.8 for recombinant TBK1.
CSN25836 CMPD101 865608-11-3 CMPD101 is a selective GRK2/3 inhibitor with IC50 values of 32 and 54 nM for GRK3 and GRK2, respectively.
CSN20021 Bryostatin 1 83314-01-6 Bryostatin 1 is a Protein kinase C (PKC) activator that binds with high affinity (Ki = 1.35 nM).
CSN42722 Belumosudil mesylate 2109704-99-4 Belumosudil is a small molecule and selective inhibitor of ROCK2 with IC50 of 105 nM, which is over 200 fold selecivity over ROCK1 (IC50 =24 μM).
CSN12528 4μ8C 14003-96-4 4μ8C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM.
CSN106900 WNK-IN-1 2125724-72-1
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