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SSTR
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN20318 | SSTR5 Antagonist C3p | 1628744-37-5 | SSTR5 antagonist C3p is a SSTR5 antagonist with improved PK profile and hERG inhibition activity. It can successfully exhibited a persistent glucose-lowering effect in an OGTT at a dose of 3 mg/kg. |
| CSN18258 | Pasireotide L-aspartate salt | 396091-77-3 | Pasireotide L-aspartate is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/< 7.0/9.9 respectively). |
| CSN18989 | Pasireotide ditrifluoroacetate | 396091-75-1 | Pasireotide ditrifluoroacetate is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/< 7.0/9.9 respectively). |
| CSN20632 | Octreotide | 83150-76-9 | Octreotide is an analog of somatostatin that binds to the somatostatin receptor 2/3/5. It can increase Gi activity and reduce the production of intracellular cAMP. |
| CSN11597 | Octreotide acetate | 79517-01-4 | Octreotide acetate is a long-acting octapeptide with pharmacologic actions mimicking those of the natural hormone somatostatin. |
| CSN20262 | Lanreotide | 108736-35-2 | Lanreotide, a synthetic cyclic octapeptide, is the analogue of somatostatin that can inhibit somatostatin receptor 2 (SSTR-2). |
| CSN20261 | Lanreotide Acetate | 127984-74-1 | Lanreotide acetate is an a synthetic cyclic octapeptide analogue of somatostatin exhibiting a high binding affinity for somatostatin receptor 2 (SSTR-2) and a lesser binding affinity for SSTR-5. |
| CSN26773 | J-2156 TFA | 2387505-73-7 | J-2156 TFA is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. J-2156 TFA is used for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws in rats[1][2]. |
| CSN25291 | FK962 | 283167-06-6 | FK962 is an enhancer of somatostatin release, with anti-dementia properties. |
| CSN41896 | J-2156 | 848647-56-3 | |
| CSN41277 | Cyclosomatostatin | 84211-54-1 | |
| CSN34246 | BIM-23056 | 150155-61-6 | |
| CSN43461 | SSTR5 antagonist 1 | 1628741-91-2 | |
| CSN51562 | N-((2R)-1-(((3-(Aminomethyl)cyclohexyl)methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide | 208706-12-1 |
