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Transferase

Transferase

货号 产品名 CAS号 信息
CSN18065 Tipifarnib S-Enantiomer 192185-71-0 Tipifarnib S-enantiomer is the enantiomer of tipifarnib, a potent and specific farnesyltransferase inhibitor with an IC50 of 0.6 nM.
CSN12963 Tipifarnib 192185-72-1 Tipifarnib is an inhibitor of farnesyltransferase with IC50 of 0.6 nM.
CSN16117 Salirasib 162520-00-5 Salirasib is an inhibitor of prenylated protein methyltransferase (PPMTase) with Ki of 2.6 μM and can inhibit the methylation of Ras.
CSN22500 RP-64477 135239-65-5 RP-64477 is a potent inhibitor of the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT).
CSN20228 PF-9366 72882-78-1 PF-9366 is an allosteric inhibitor of Mat2A that binds an allosteric site on Mat2A that overlaps with the binding site for the Mat2A regulator, Mat2B, targeting S-adenosylmethionine biosynthesis, with IC50 of 420 nM and Kd of 170 nM, respectively.
CSN10813 Perillyl Alcohol 536-59-4 Perillyl Alcohol is a naturally occurring monocyclic terpene which can inhibit farnesyl transferase and geranylgeranyl transferase.
CSN20781 O6-Benzylguanine 19916-73-5 O6-Benzylguanine is an inactivator of O6-alkylguanine DNA alkyltransferase (AGT) and can prevent the repair of DNA damage induced by chemotherapeutics. It induces apoptosis and cell death. 
CSN25442 Tris DBA 51364-51-3 N-myristoyltransferase-1 (NMT-1) inhibitor that prevents activation of MAPK, PI 3-K and STAT3 signaling pathways. Exhibits antiproliferative activity against melanoma cells in vitro and in vivo. Also used as a cyclization catalyst.
CSN24695 Myriocin 35891-70-4 Myriocin is a potent SPT (serine palmitoyltransferase) inhibitor.
CSN11326 Lonafarnib 193275-84-2 Lonafarnib is a FPTase inhibitor. It can inhibit H-ras (IC50 = 1.9 nM), K-ras-4B (IC50 = 5.2 nM) and N-ras (IC50 = 2.8 nM).
CSN27242 Lifibrate 22204-91-7 Lifibrate is an inhibitor of cholinephosphotransferase (CPT), phosphatidyl-N-methylethanolamine N-methyltransferase (PME-NMT), and phosphatidyl-N,N-dimethylethanolamine N-methyltransferase (PDE-NMT).
CSN24041 L-Glutamic acid γ-(p-nitroanilide) 7300-59-6 L-Glutamic acid γ-(p-nitroanilide) is a substrate for γ-glutamyl transpeptidase.
CSN23739 L-Glutamic acid γ-(p-nitroanilide) HCl 67953-08-6 L-Glutamic acid γ-(p-nitroanilide) HCl is a substrate for GGT (gamma-glutamyltransferase), which is a transferase that catalyzes the transfer of gamma-glutamyl functional groups from molecules such as glutathione to an acceptor.
CSN12834 L-778123 HCl 253863-00-2 L-778123 HCl is an inhibitor of FPTase and GGPTase-I with IC50 of 2 nM and 98 nM in enzyme inhibition determination.
CSN27575 Isoastilbin   54081-48-0 Isoastilbin is a dihydroflavonol glycoside compound in Rhizoma Smilacis glabrae and Astragalus membranaceus. Isoastilbin inhibits glucosyltransferase (GTase) with an IC50 value of 54.3 μg/mL, and also inhibits tyrosinase activity. Isoastilbin shows neuroprotective, antioxidation, antimicrobial and anti-apoptotic properties and has the potential for Alzheimer’s disease research.
CSN25448 LY 78335 HCl 39959-66-5 High affinity inhibitor of phenylethanolamine-N-methyltransferase (PNMT) (Ki = 0.09 μM in vitro). Suppresses the release of growth hormone in an in vivo rat model.
CSN27598 GOT1 inhibitor 2c   732973-87-4 GOT1 inhibitor 2c is a GOT1 inhibitor with IC50 value of 8.2μM.
CSN19197 GGTI298 Trifluoroacetate 1217457-86-7 GGTI298 trifluoroacetate is geranylgeranyltransferase I inhibitor. It shows supression of the G1 phase of the cell cycle and induction of apoptosis.
CSN23732 GGTI-2418 501010-06-6 GGTI-2418 is a highly potent, competitive, and selective geranylgeranyltransferase I (GGTase I) inhibitor. GGTI-2418 inhibits GGTase I and FTase activities with IC50s of 9.5 nM and 53 μM, respectively. GGTI-2418 also increases p27(Kip1) and induces significant regression of breast tumors[1].
CSN11092 Geraniol 106-24-1 Geraniol is an inhibitor of glutathion S transferase with anticarcinogenic property.
CSN27300 GDP-Mannose disodium salt 148296-46-2 GDP-α-D-mannose disodium is the donor substrate for mannosyltransferases and the precursor of GDP-β-L-fucose. GDP-α-D-mannose disodium gives a competitive inhibition with respect to GTP (Ki 14.7 μM) and an uncompetitive inhibition with respect to mannose-1-P (Ki 115 μM) .
CSN20234 FTI-277 Trifluoroacetate 1217447-06-7 FTI-277 trifluoroacetate is an inhibitor of farnesyl transferase (FTase) and a highly potent Ras CAAX peptidomimetic which antagonizes both H- and K-Ras oncogenic signaling.
CSN18001 FTI-277 170006-73-2 FTI-277 is an inhibitor of farnesyl transferase (FTase) and a highly potent Ras CAAX peptidomimetic which antagonizes both H- and K-Ras oncogenic signaling.
CSN18044 FTI-277 HCl 180977-34-8 FTI-277 HCl is an inhibitor of farnesyl transferase (FTase) and a highly potent Ras CAAX peptidomimetic which antagonizes both H- and K-Ras oncogenic signaling.
CSN22128 FTI 276 170006-72-1 FTI-276 is a protein farnesyl transferase (PFT) inhibitor with IC50s of 0.9 and 0.5 nM for Plasmodium falciparum and human.
CSN25323 FTI-2148 251577-09-0 FTI-2148 is a RAS C-terminal mimetic dual farnesyl transferase (FT-1) and geranylgeranyl transferase-1 (GGT-1) inhibitor with IC50s of 1.4 nM and 1.7 μM for FT-1 and GGT-1, respectively.
CSN22389 E-5324 141799-76-0 E-5324 is potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT) with IC50s of 44 to 190 nM.
CSN21070 CP-609754 1190094-64-4 CP-609754, also known as CP-609,754, LNK 754 and OSI 754, is a selective inhibitor of arnesyltransferase with potential anticancer activity.
CSN24943 Benzoyleneurea 86-96-4 Benzoyleneurea scaffold is used in the synthesis of novel protein geranylgeranyltransferase-I inhibitors.
CSN24135 ATR-101 133825-80-6 ATR-101 is a selective inhibitor of acyl coenzyme A:cholesterol acyltransferase (ACAT1), it is in clinical development for the treatment of adrenocortical carcinoma (ACC).
CSN20465 ATR-101 HCl 133825-81-7 ATR-101 HCl is a selective inhibitor of acyl coenzyme A:cholesterol acyltransferase (ACAT1), it is in clinical development for the treatment of adrenocortical carcinoma (ACC).
CSN23571 Aminooxyacetic acid hemihydrochloride 2921-14-4 Aminooxyacetic acid hemihydrochloride is an inhibitor of malate-aspartate shuttle (MAS) and also exhibits suppression of GABA-T.
CSN10276 Amentoflavone 1617-53-4 Amentoflavone is an inhibitor of human UDP-glucuronosyltransferases with anti-inflammatory, antioxidative, and neuroprotective effects and it can be isolated from the seeds of Ginkgo biloba L. Amentoflavone inhibited SARS-CoV 3CL(pro) with IC50 value of 8.3μM.
CSN23722 MAT2A Inhibitor 1 13299-99-5 AG-270 is a potent and orally active methionine adenosyltransferase 2A (MAT2A) inhibitor with potential antineoplastic activity.
CSN12803 (R)-(+)-Etomoxir Sodium 828934-41-4 (R)-(+)-etomoxir sodium salt is inhibitor of carnitine palmitoyltransferase I (CPT1) and can reduce β-oxidation in mitochondria. It shows inhibition of cardiolipin biosynthesis.
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