Dienogest is an agonist of progesterone receptor with endometrial activity that is used to treat endometriosis.

α-Estradiol is an endogenous estrogen receptor ligand (Ki values are 0.2 and 1.2 nM for ERα and ERβ receptors respectively).

Levonorgestrel is a synthetic progestogen and can used as an active ingredient in some hormonal contraceptives.

Mestranol is an agonist of estrogen receptor. It is used as contraceptives.

Estradiol is an estrogenic hormone that is produced in the ovaries, placenta, testis.

Mifepristone is an antagonist of progesterone receptor (IC50 = 0.2 nM) and glucocorticoid receptor (IC50 = 2.6 nM).

Estrone is an estrogenic hormone secreted by the ovary as well as adipose tissue.

Norethindrone acetate is a female progestin approved by FDA for the treatment of endometriosis, uterine bleeding caused by abnormal hormone levels, and secondary amenorrhea.

Estradiol Valeate is a synthetic estrogen. Formulations containing estradiol valerate with other steroid hormones have been used to treat endometriosis.

Altrenogest is a progestogen used as veterinary medicine and structurally related to steroid trenbolone.

Ethynyl Estradiol is an estrogen used in formulations of combined contraceptive pills.

Ulipristal acetate is a selective modulator of progesterone receptor and can be used to treat uterine myoma.

Ethynodiol diacetate is a hormonal contraceptive with significant estrogenic effects.

Norethindrone is a synthetic progestin which can mimic the effects of endogenous ovarian hormones.

2-methoxyestradiol is a natural metabolite of estrogen that is known to inhibit HIF-1 alpha with an IC50 of 0.71 ± 0.11 μM for the inhibition of BPAEC migration.

Estriol is G-protein coupled estrogen receptor antagonist in estrogen receptor-negative breast cancer cells. It is a major urinary estrogen which is largely produced by the placenta during pregnancy.

Quinestrol is a synthetic estrogen which is used in hormone replacement therapy.

Allylestrenol is a synthetic steroidal progestin that is used to prevent recurrent pregnancy loss, threatened miscarriage, and premature labor.