SBI-553 is a potent, brain-penetrant and allosteric modulator of NTR1 with EC50 of 0.34 μM.

Neurotensin Fragment 8-13 is the smallest active fragment of neurotensin which is a potent cellular mitogen for various colorectal and pancreatic cancers which possess high-affinity neurotensin receptors (NTR).

PD 90780 is a non-peptide inhibitor of nerve growth factor (NGF) binding to p75NTR receptor. It inhibits NGF-p75 NTR interaction with IC50s values of 23.1 µM and 1.8 µM in PC12 cells and PC12 nnr5 cells, respectively.

Neurotensin, a potent hypothalamic peptide neurotransmitter, is an endogenous anti-psychotic compound which has a high affinity for neurotensin receptors.

JMV 449 is a potent, metabolically stable neurotensin receptor agonist peptide.

Kinetensin is endogenous neurotensin-like peptide originally isolated from pepsin-treated human plasma. It can induce histamine release from rat peritoneal mast cells in vitro.

ML314 is a potent molecule agonist of NTR1 (EC50 = 1.9 μM) and shows good selectivity against NTR2 and GPR35, but did not stimulate Ca2+ mobilization.

Xenopsin is the neurotensin-like octapeptide from Xenopus skin at the carboxyl terminus of its precursor.