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CAS No.: 1643913-93-2
Synonyms: PAK4-IN-1
PAK4-IN-1 is an inhibitor of p21-activated kinases (PAKs), with IC50 of ≤100 nM in MTT assay.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02702492 | NHL Solid Tum... more >>ors Collapse << | Phase 1 | Recruiting | November 2019 | United States, Colorado ... more >> University of Colorado Cancer Center Recruiting Aurora, Colorado, United States, 80045 Contact: Stephen Leong, MD Stephen.Leong@ucdenver.edu Principal Investigator: Stephen Leong, MD United States, District of Columbia Georgetown University, Lombardi Comprehensive Cancer Center Recruiting Washington, District of Columbia, United States, 20007 Contact: Michael Pishvaian, MD, PhD pishvaim@georgetown.edu Principal Investigator: Michael Pishvaian, MD, PhD United States, Minnesota Mayo Clinic Rochester Recruiting Rochester, Minnesota, United States, 55905 Contact: Amit Mahipal, MBBS, MPH 507-293-0462 mahipal.amit@mayo.edu Principal Investigator: Amit Mahipal, MBBS, MPH United States, New York NYU-Laura & Isaac Perlmutter Cancer Center Recruiting New York, New York, United States, 100016 Contact: Daniel Cho 212-731-5871 daniel.cho@nyumc.org Principal Investigator: Daniel Cho, MD United States, Tennessee Vanderbilt-Ingram Cancer Center Recruiting Nashville, Tennessee, United States, 37232 Contact: Jordan Berlin, MD Contact Jordan.Berlin@vanderbilt.edu Principal Investigator: Jordan Berlin, MD United States, Texas MD Anderson Cancer Center Recruiting Houston, Texas, United States, 77030 Contact: Aung Naing 713-563-0803 anaing@mdanderson.org Principal Investigator: Aung Naing, MD Canada, Ontario Princess Margaret Hospital Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Albiruni Razak, MB, BCh 416-586-4800 ext 3883 Principal Investigator: Albiruni Razak, MB, Bch Collapse << |
实验方案
技术信息
CAS号 | 1643913-93-2 | 储存条件 |
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分子式 | C35H29F3N4O3 | 运输 | 蓝冰 | |
分子量 | 610.63 | 别名 | PAK4-IN-1 |