400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Protein Tyrosine Kinase/RTK / c-Met/HGFR / BMS-794833
CAS No.: 1174046-72-0
Synonyms: BMS-794833
BMS-794833 is a potent ATP competitive inhibitor of Met and VEGFR2 with IC50 of 1.7 and 15 nM.
生物活性
靶点 | c-Met IC50:1.7nM | VEGFR2 IC50:15nM | Axl IC50:3nM | FLT3 IC50:3nM | Ron IC50:3nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00792558 | Advanced Solid Tumors | Phase 1 | Withdrawn | November 2010 | Australia, South Australia ... more >> Local Institution Adelaide, South Australia, Australia, 5000 Australia, Western Australia Local Institution Nedlands, Western Australia, Australia, 6009 Singapore Local Institution Singapore, Singapore, 169610 Collapse << |
实验方案
技术信息
CAS号 | 1174046-72-0 | 储存条件 |
|
|||||||
分子式 | C23H15ClF2N4O3 | 运输 | 蓝冰 | |||||||
分子量 | 468.84 | 别名 | BMS-794833 | |||||||
溶解度 |
|
动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00792558 | Advanced Solid Tumors | Phase 1 | Withdrawn | November 2010 | Australia, South Australia ... more >> Local Institution Adelaide, South Australia, Australia, 5000 Australia, Western Australia Local Institution Nedlands, Western Australia, Australia, 6009 Singapore Local Institution Singapore, Singapore, 169610 Collapse << |
靶点 | Description | IC50 |
---|---|---|
c-Met | IC50:1.7nM | |
VEGFR2 | IC50:15nM | |
Axl | IC50:3nM | |
FLT3 | IC50:3nM | |
Ron | IC50:3nM |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网