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CAS No.: 439087-18-0
Synonyms: A 3309;AZD 7806;AJG-533
Elobixibat is a potent ileal bile acid transporter (IBAT) inhibitor with IC50 values of 0.53 ± 0.17 nM, 0.13 ± 0.03 nM, and 5.8 ± 1.6 nM for human IBAT, mouse IBAT, and canine IBAT.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01069783 | Dyslipidemia | Phase 2 | Completed | - | Sweden ... more >> BCRC Linköping, Sweden Collapse << |
NCT01895543 | - | - | Completed | - | - |
NCT01038687 | Functional Constipation | Phase 2 | Completed | - | United States, Minnesota ... more >> Mayo Clinic in Rochester Rochester, Minnesota, United States, 55905 Collapse << |
实验方案
技术信息
CAS号 | 439087-18-0 | 储存条件 |
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分子式 | C36H45N3O7S2 | 运输 | 蓝冰 | |
分子量 | 695.89 | 别名 | A 3309;AZD 7806;AJG-533 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01069783 | Dyslipidemia | Phase 2 | Completed | - | Sweden ... more >> BCRC Linköping, Sweden Collapse << |
NCT01895543 | - | - | Completed | - | - |
NCT01038687 | Functional Constipation | Phase 2 | Completed | - | United States, Minnesota ... more >> Mayo Clinic in Rochester Rochester, Minnesota, United States, 55905 Collapse << |
NCT01895543 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Completed | - | - |
NCT01833065 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Terminated(Terminated due to a... more >> distribution issue with the trial medication) Collapse << | - | - |
NCT01827592 | - | - | Terminated(Terminated due to a... more >> distribution issue with the trial medication) Collapse << | - | - |
NCT01007123 | Constipation ... more >>Chronic Constipation Collapse << | Phase 2 | Completed | - | - |
NCT01833065 | - | - | Terminated(Terminated due to a... more >> distribution issue with the trial medication) Collapse << | - | - |
NCT01007123 | - | - | Completed | - | - |
NCT02392546 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 2 | Withdrawn(Business reasons) | April 2016 | United States, Minnesota ... more >> Mayo Clinic Rochester, Minnesota, United States Collapse << |
NCT01827592 | Chronic Idiopathic Constipatio... more >>n Collapse << | Phase 3 | Terminated(Terminated due to a... more >> distribution issue with the trial medication) Collapse << | - | - |
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