GR 113808
98%
货号：A109758
产品仅供科研
GR 113808 is a potent, selective 5-HT4 receptor antagonist with Kd of 0.15 nM for binding to cloned human 5-HT4 receptors.
GR 113808 化学结构
CAS号：144625-51-4
GR 113808 3D分子结构
CAS号：144625-51-4
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咨询
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+
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| Desvenlafaxine |
++
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98% |
| Lamotrigine |
+
5-HT (human platelets), IC50: 240 μM
5-HT (rat brain synaptosomes), IC50: 474 μM
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98% |
| Venlafaxine |
✔
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98% |
| Fluvoxamine maleate |
✔
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99% |
| Iloperidone |
✔
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98% |
| Ziprasidone HCl |
✔
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98+% |
| Atomoxetine HCI |
+
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98% |
| Dapoxetine HCl |
✔
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97% |
| Trazodone |
✔
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98+% |
| Clomipramine HCl |
✔
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98% |
| Mirtazapine |
✔
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99+% |
| Escitalopram oxalate |
+++
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97% |
| Duloxetine |
✔
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98+% |
| Sertraline HCl |
++
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98% |
| Citalopram HBr |
+++
serotonin reuptake, IC50: 1.8 nM
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98% |
| WAY-100635 maleate |
+++
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99% |
| Latrepirdine 2HCl |
✔
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GluR
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98+% |
| Fluoxetine hydrochloride |
✔
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98% |
| Paroxetine hydrochloride |
✔
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AChR
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97% |
| BMY 7378 |
|
++
5-HT1D, pIC50: 5.9
5-HT1A, pIC50: 6.4
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+
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97% |
| Flibanserin |
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+++
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+
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98% |
| LY310762 |
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+
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99%+ |
| Cyclobenzaprine HCI |
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✔
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99% |
| Blonanserin |
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+++
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98% HPLC |
| Cyproheptadine HCl |
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++++
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99+% |
| Olanzapine |
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✔
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99+% |
| Pimavanserin hemitartrate |
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+++
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99% |
| Ketanserin |
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+++
5-HT2C (Human), Ki: 2.5 nM
5-HT2C (Rat), Ki: 50 nM
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99%+ |
| Loxapine succinate |
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++
5-HT2 (human), Ki: 6.8 nM
5-HT2 (bovine), Ki: 6.6 nM
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99% |
| Agomelatine |
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✔
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98% |
| Clozapine |
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✔
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98% |
| Amitriptyline |
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+
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SERT
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98% |
| PRX-08066 maleate |
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+++
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98+% |
| RS-127445 |
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++++
5-HT2B, pKi: 9.5
5-HT2B, pIC50: 10.4
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98%+ |
| Sarpogrelate HCl |
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++++
5-HT2C, Kd: 1.1 nM
5-HT2A, Kd: 2.1 nM
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98% |
| Tropisetron |
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✔
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99% |
| Palonosetron |
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✔
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98+% |
| Ramosetron HCl |
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++++
5-HT3 receptor, Ki: 0.091 nM
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98% |
| Ondansetron |
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✔
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99% |
| Granisetron |
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✔
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98% |
| Alosetron HCl |
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✔
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98% |
| Ondansetron hydrochloride dihydrate |
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✔
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98% |
| VUF10166 |
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++++
5-HT3AB, Ki: 22 nM
5-HT3A, Ki: 0.04 nM
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99%+ |
| Azasetron hydrochloride |
|
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++++
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98% |
| Asenapine maleate |
|
+++
5-HT1B, pKi: 8.4
5-HT1A, pKi: 8.6
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++++
5-HT2C, pKi: 10.46
5-HT2A, pKi: 9.75
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+++
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++++
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++++
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97% |
| Risperidone |
|
++
5-HT1B, Ki: 14.9 nM
5-HT1D, Ki: 84.6 nM
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++++
5-HT2A, Ki: 61.9 nM
5-HT2C, Ki: 12 nM
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+
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++
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98% |
| SB 271046 HCl |
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+++
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99%+ |
| Intepirdine |
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++++
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99%+ |
| SB-269970 HCl |
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++
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98+% |
| BRL 15572 |
|
++
5-HT1D, pKi: 6
5-HT1B, pKi: 6.1
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++
5-HT2B, pKi: 6.2
5-HT2A, pKi: 6.6
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+
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+
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98% |
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1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
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GR 113808 实验方案
| 计算器 |
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| 存储液制备 |
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1mg |
5mg |
10mg |
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1 mM
5 mM
10 mM
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2.54mL
0.51mL
0.25mL
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12.71mL
2.54mL
1.27mL
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25.41mL
5.08mL
2.54mL
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GR 113808 技术信息
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