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CAS No.: 1191252-49-9
Synonyms: IOWH-032
IOWH-032 is a potent CFTR inhibitor (IC50=1.01 μM) in T84 and CHO-CFTR cell based assays.
生物活性
靶点 | CFTR IC50:1.01μM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01823939 | Diarrhea Chol... more >>era Collapse << | Phase 1 | Completed | - | Bangladesh ... more >> Dhaka Hospital - icddr,b (International Centre for Diarrhoeal Disease Research, Bangladesh) Mohakhali, Dhaka, Bangladesh, 1212 Collapse << |
NCT02111304 | Secretory Diarrhea | Phase 2 | Withdrawn(Trial was never init... more >>iated due to PATH executive decision.) Collapse << | May 2016 | Bangladesh ... more >> International Centre for Diarrhoeal Disease Research, Bangladesh Dhaka, Bangladesh, 1212 Collapse << |
实验方案
技术信息
CAS号 | 1191252-49-9 | 储存条件 |
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分子式 | C22H15Br2N3O4 | 运输 | 蓝冰 | |||||||
分子量 | 545.18 | 别名 | IOWH-032 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01823939 | Diarrhea Chol... more >>era Collapse << | Phase 1 | Completed | - | Bangladesh ... more >> Dhaka Hospital - icddr,b (International Centre for Diarrhoeal Disease Research, Bangladesh) Mohakhali, Dhaka, Bangladesh, 1212 Collapse << |
NCT02111304 | Secretory Diarrhea | Phase 2 | Withdrawn(Trial was never init... more >>iated due to PATH executive decision.) Collapse << | May 2016 | Bangladesh ... more >> International Centre for Diarrhoeal Disease Research, Bangladesh Dhaka, Bangladesh, 1212 Collapse << |
靶点 | Description | IC50 |
---|---|---|
CFTR | IC50:1.01μM |
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