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CAS No.: 943540-74-7
JNJ-38877618 is a potent, highly selective, orally bioavailable Met kinase inhibitor with IC50s of 2 and 3 nM for wild type and mutant Met, respectively.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01964872 | Healthy Volunteers | Phase 1 | Completed | - | United Kingdom ... more >> Nottingham, United Kingdom Collapse << |
NCT03138083 | Neoplasms | Phase 1 Phase 2 | Recruiting | December 2020 | France ... more >> lNSTITUT GUSTAVE ROUSSY Recruiting Villejuif, France, 94805 Contact: Eric Angevin, MD Netherlands Erasmus Mc Recruiting Rotterdam, Netherlands, 3000 CA Contact: Martijn Lolkema, MD/PhD Universitair Medisch Centrum Utrecht Recruiting Utrecht, Netherlands, 3584 CX Contact: Filip De Vos, MD United Kingdom University College London Hospitals Nhs Foundation Trust Recruiting London, United Kingdom, NW1 2BU Contact: Martin Forster, MD The Christie Nhs Foundation Trust Recruiting Manchester, United Kingdom, M20 4BX Contact: Matthew G Krebs, MD PhD MRCP Matthew.Krebs@christie.nhs.uk The Newcastle Upon Tyne Hospitals Nhs Foundation Trust Recruiting Newcastle upon Tyne, United Kingdom, NE7 7DN Contact: Ruth Plummer, MD Ruth.Plummer@newcastle.ac.uk University of Oxford, Department of Oncology Recruiting Oxford, United Kingdom, OX3 7LE Contact: Sarah P Blagden, MD +441865227212 sarah.blagden@oncology.ox.ac.uk Collapse << |
实验方案
技术信息
CAS号 | 943540-74-7 | 储存条件 |
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分子式 | C20H12F2N6 | 运输 | 蓝冰 | |
分子量 | 374.35 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01964872 | Healthy Volunteers | Phase 1 | Completed | - | United Kingdom ... more >> Nottingham, United Kingdom Collapse << |
NCT03138083 | Neoplasms | Phase 1 Phase 2 | Recruiting | December 2020 | France ... more >> lNSTITUT GUSTAVE ROUSSY Recruiting Villejuif, France, 94805 Contact: Eric Angevin, MD Netherlands Erasmus Mc Recruiting Rotterdam, Netherlands, 3000 CA Contact: Martijn Lolkema, MD/PhD Universitair Medisch Centrum Utrecht Recruiting Utrecht, Netherlands, 3584 CX Contact: Filip De Vos, MD United Kingdom University College London Hospitals Nhs Foundation Trust Recruiting London, United Kingdom, NW1 2BU Contact: Martin Forster, MD The Christie Nhs Foundation Trust Recruiting Manchester, United Kingdom, M20 4BX Contact: Matthew G Krebs, MD PhD MRCP Matthew.Krebs@christie.nhs.uk The Newcastle Upon Tyne Hospitals Nhs Foundation Trust Recruiting Newcastle upon Tyne, United Kingdom, NE7 7DN Contact: Ruth Plummer, MD Ruth.Plummer@newcastle.ac.uk University of Oxford, Department of Oncology Recruiting Oxford, United Kingdom, OX3 7LE Contact: Sarah P Blagden, MD +441865227212 sarah.blagden@oncology.ox.ac.uk Collapse << |
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