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CAS No.: 1951408-58-4

MAK683 Catalog No. CSN21253

Synonyms: EED inhibitor-1

An inhibitor of embryonic ectoderm development protein (EED) and allosteric inhibitor of polycomb repressive complex 2 (PRC2), with potential antineoplastic activity.

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靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02900651Diffuse Large B-cell LymphomaPhase 1 Phase 2RecruitingAugust 5, 2019United States, California ... more >> Novartis Investigative Site Recruiting San Francisco, California, United States, 94115 Novartis Investigative Site Recruiting Santa Monica, California, United States, 90404 Contact: Ruth M. Gonzalez       Rngonzalez@mednet.ucla.edu    Principal Investigator: Zev A. Wainberg          United States, Texas Novartis Investigative Site Recruiting Houston, Texas, United States, 77030 Contact: Anna Lui    713-563-4667    alui@mdanderson.org    Principal Investigator: Vivek Subbiah          Canada, Ontario Novartis Investigative Site Recruiting Toronto, Ontario, Canada, M5G 2M9 France Novartis Investigative Site Recruiting Villejuif Cedex, France, 94805 Germany Novartis Investigative Site Recruiting Koeln, Germany, 50937 Hong Kong Novartis Investigative Site Recruiting Hong Kong, Hong Kong Italy Novartis Investigative Site Recruiting Milano, MI, Italy, 20133 Japan Novartis Investigative Site Recruiting Sunto-gun, Shizuoka, Japan, 411-8777 Singapore Novartis Investigative Site Recruiting Singapore, Singapore, 169610 Spain Novartis Investigative Site Recruiting Madrid, Spain, 28041 Collapse <<
  • 参考文献

实验方案

技术信息

CAS号 1951408-58-4 储存条件
分子式 C20H17FN6O 运输 蓝冰
分子量 376.39 别名 EED inhibitor-1

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