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CAS No.: 717907-75-0
Synonyms: VS-6062
PF-562271 is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, ~10-fold less potent for Pyk2 than FAK and > 100-fold selectivity against other protein kinases, except for some CDKs.
生物活性
靶点 | FAK IC50:1.5nM | Pyk2 IC50:13nM |
实验方案
技术信息
CAS号 | 717907-75-0 | 储存条件 |
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分子式 | C21H20F3N7O3S | 运输 | 蓝冰 | |||||||||||||
分子量 | 507.49 | 别名 | VS-6062 | |||||||||||||
溶解度 |
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动物实验配方 |
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Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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KG-1 | - | Growth Inhibition Assay | - | IC50=5.74005 μM | SANGER |
KINGS-1 | - | Growth Inhibition Assay | - | IC50=12.3421 μM | SANGER |
KLE | - | Growth Inhibition Assay | - | IC50=28.9906 μM | SANGER |
KM12 | - | Growth Inhibition Assay | - | IC50=0.38557 μM | SANGER |
KM-H2 | - | Growth Inhibition Assay | - | IC50=31.7306 μM | SANGER |
KMOE-2 | - | Growth Inhibition Assay | - | IC50=21.3288 μM | SANGER |
KNS-42 | - | Growth Inhibition Assay | - | IC50=9.43407 μM | SANGER |
KNS-81-FD | - | Growth Inhibition Assay | - | IC50=21.8631 μM | SANGER |
KOSC-2 | - | Growth Inhibition Assay | - | IC50=2.63879 μM | SANGER |
KP-4 | - | Growth Inhibition Assay | - | IC50=8.41853 μM | SANGER |
KP-N-YS | - | Growth Inhibition Assay | - | IC50=8.29308 μM | SANGER |
KS-1 | - | Growth Inhibition Assay | - | IC50=4.42459 μM | SANGER |
KU-19-19 | - | Growth Inhibition Assay | - | IC50=39.6282 μM | SANGER |
KU812 | - | Growth Inhibition Assay | - | IC50=19.5944 μM | SANGER |
KURAMOCHI | - | Growth Inhibition Assay | - | IC50=5.02834 μM | SANGER |
KY821 | - | Growth Inhibition Assay | - | IC50=47.6434 μM | SANGER |
KYSE-140 | - | Growth Inhibition Assay | - | IC50=36.7298 μM | SANGER |
KYSE-150 | - | Growth Inhibition Assay | - | IC50=1.35236 μM | SANGER |
KYSE-180 | - | Growth Inhibition Assay | - | IC50=2.28874 μM | SANGER |
KYSE-270 | - | Growth Inhibition Assay | - | IC50=1.04714 μM | SANGER |
KYSE-410 | - | Growth Inhibition Assay | - | IC50=2.56517 μM | SANGER |
KYSE-510 | - | Growth Inhibition Assay | - | IC50=5.79581 μM | SANGER |
KYSE-520 | - | Growth Inhibition Assay | - | IC50=26.5553 μM | SANGER |
KYSE-70 | - | Growth Inhibition Assay | - | IC50=31.3008 μM | SANGER |
L-363 | - | Growth Inhibition Assay | - | IC50=4.55996 μM | SANGER |
L-540 | - | Growth Inhibition Assay | - | IC50=11.899 μM | SANGER |
LAN-6 | - | Growth Inhibition Assay | - | IC50=31.4992 μM | SANGER |
LB1047-RCC | - | Growth Inhibition Assay | - | IC50=5.90148 μM | SANGER |
LB2241-RCC | - | Growth Inhibition Assay | - | IC50=13.1469 μM | SANGER |
LB2518-MEL | - | Growth Inhibition Assay | - | IC50=20.3953 μM | SANGER |
LB373-MEL-D | - | Growth Inhibition Assay | - | IC50=16.6138 μM | SANGER |
LB771-HNC | - | Growth Inhibition Assay | - | IC50=7.18038 μM | SANGER |
LB831-BLC | - | Growth Inhibition Assay | - | IC50=2.00988 μM | SANGER |
LB996-RCC | - | Growth Inhibition Assay | - | IC50=42.8008 μM | SANGER |
LC-1F | - | Growth Inhibition Assay | - | IC50=47.6105 μM | SANGER |
LC-2-ad | - | Growth Inhibition Assay | - | IC50=2.26966 μM | SANGER |
LC4-1 | - | Growth Inhibition Assay | - | IC50=5.39303 μM | SANGER |
LCLC-103H | - | Growth Inhibition Assay | - | IC50=1.55818 μM | SANGER |
LCLC-97TM1 | - | Growth Inhibition Assay | - | IC50=7.21273 μM | SANGER |
LK-2 | - | Growth Inhibition Assay | - | IC50=15.0862 μM | SANGER |
LNCaP-Clone-FGC | - | Growth Inhibition Assay | - | IC50=37.1903 μM | SANGER |
LOUCY | - | Growth Inhibition Assay | - | IC50=2.26128 μM | SANGER |
LoVo | - | Growth Inhibition Assay | - | IC50=8.95566 μM | SANGER |
LOXIMVI | - | Growth Inhibition Assay | - | IC50=33.3679 μM | SANGER |
LS-1034 | - | Growth Inhibition Assay | - | IC50=48.8954 μM | SANGER |
LS-123 | - | Growth Inhibition Assay | - | IC50=15.0165 μM | SANGER |
LS-411N | - | Growth Inhibition Assay | - | IC50=30.1475 μM | SANGER |
LS-513 | - | Growth Inhibition Assay | - | IC50=22.0367 μM | SANGER |
LU-134-A | - | Growth Inhibition Assay | - | IC50=12.93 μM | SANGER |
LU-165 | - | Growth Inhibition Assay | - | IC50=33.008 μM | SANGER |
LU-65 | - | Growth Inhibition Assay | - | IC50=10.2943 μM | SANGER |
LU-99A | - | Growth Inhibition Assay | - | IC50=27.1754 μM | SANGER |
LXF-289 | - | Growth Inhibition Assay | - | IC50=2.58273 μM | SANGER |
M059J | - | Growth Inhibition Assay | - | IC50=6.55625 μM | SANGER |
MC-CAR | - | Growth Inhibition Assay | - | IC50=23.5183 μM | SANGER |
MC-IXC | - | Growth Inhibition Assay | - | IC50=33.5655 μM | SANGER |
MDA-MB-175-VII | - | Growth Inhibition Assay | - | IC50=27.6975 μM | SANGER |
MDA-MB-231 | - | Growth Inhibition Assay | - | IC50=2.49572 μM | SANGER |
MDA-MB-453 | - | Growth Inhibition Assay | - | IC50=39.0218 μM | SANGER |
MDA-MB-468 | - | Growth Inhibition Assay | - | IC50=1.91272 μM | SANGER |
MEG-01 | - | Growth Inhibition Assay | - | IC50=6.93546 μM | SANGER |
MEL-HO | - | Growth Inhibition Assay | - | IC50=1.97993 μM | SANGER |
MEL-JUSO | - | Growth Inhibition Assay | - | IC50=1.72891 μM | SANGER |
MES-SA | - | Growth Inhibition Assay | - | IC50=1.30682 μM | SANGER |
MFE-280 | - | Growth Inhibition Assay | - | IC50=21.3188 μM | SANGER |
MFE-296 | - | Growth Inhibition Assay | - | IC50=2.47792 μM | SANGER |
MFH-ino | - | Growth Inhibition Assay | - | IC50=9.29007 μM | SANGER |
MG-63 | - | Growth Inhibition Assay | - | IC50=0.80637 μM | SANGER |
MHH-ES-1 | - | Growth Inhibition Assay | - | IC50=1.79568 μM | SANGER |
MHH-NB-11 | - | Growth Inhibition Assay | - | IC50=2.12818 μM | SANGER |
MHH-PREB-1 | - | Growth Inhibition Assay | - | IC50=8.73107 μM | SANGER |
MIA-PaCa-2 | - | Growth Inhibition Assay | - | IC50=15.4163 μM | SANGER |
MKN1 | - | Growth Inhibition Assay | - | IC50=4.70665 μM | SANGER |
MKN28 | - | Growth Inhibition Assay | - | IC50=8.24598 μM | SANGER |
MKN45 | - | Growth Inhibition Assay | - | IC50=8.96063 μM | SANGER |
ML-2 | - | Growth Inhibition Assay | - | IC50=1.66802 μM | SANGER |
MLMA | - | Growth Inhibition Assay | - | IC50=7.54689 μM | SANGER |
MN-60 | - | Growth Inhibition Assay | - | IC50=17.7936 μM | SANGER |
MOLT-16 | - | Growth Inhibition Assay | - | IC50=4.31016 μM | SANGER |
MOLT-4 | - | Growth Inhibition Assay | - | IC50=2.60712 μM | SANGER |
MONO-MAC-6 | - | Growth Inhibition Assay | - | IC50=2.41248 μM | SANGER |
MRK-nu-1 | - | Growth Inhibition Assay | - | IC50=44.7414 μM | SANGER |
MS-1 | - | Growth Inhibition Assay | - | IC50=6.95192 μM | SANGER |
MV-4-11 | - | Growth Inhibition Assay | - | IC50=0.2766 μM | SANGER |
MZ1-PC | - | Growth Inhibition Assay | - | IC50=1.62312 μM | SANGER |
MZ2-MEL | - | Growth Inhibition Assay | - | IC50=20.5814 μM | SANGER |
MZ7-mel | - | Growth Inhibition Assay | - | IC50=27.5548 μM | SANGER |
NB1 | - | Growth Inhibition Assay | - | IC50=4.06644 μM | SANGER |
NB10 | - | Growth Inhibition Assay | - | IC50=19.6268 μM | SANGER |
NB5 | - | Growth Inhibition Assay | - | IC50=13.5503 μM | SANGER |
NCCIT | - | Growth Inhibition Assay | - | IC50=2.5724 μM | SANGER |
NCI-H1299 | - | Growth Inhibition Assay | - | IC50=18.8918 μM | SANGER |
NCI-H1304 | - | Growth Inhibition Assay | - | IC50=6.12497 μM | SANGER |
NCI-H1355 | - | Growth Inhibition Assay | - | IC50=35.7718 μM | SANGER |
NCI-H1395 | - | Growth Inhibition Assay | - | IC50=49.0492 μM | SANGER |
NCI-H1417 | - | Growth Inhibition Assay | - | IC50=33.9585 μM | SANGER |
NCI-H1437 | - | Growth Inhibition Assay | - | IC50=12.1447 μM | SANGER |
NCI-H1648 | - | Growth Inhibition Assay | - | IC50=6.1516 μM | SANGER |
NCI-H1650 | - | Growth Inhibition Assay | - | IC50=8.29185 μM | SANGER |
NCI-H1651 | - | Growth Inhibition Assay | - | IC50=28.2592 μM | SANGER |
NCI-H1694 | - | Growth Inhibition Assay | - | IC50=21.9863 μM | SANGER |
NCI-H1703 | - | Growth Inhibition Assay | - | IC50=46.0592 μM | SANGER |
NCI-H1734 | - | Growth Inhibition Assay | - | IC50=4.26695 μM | SANGER |
NCI-H1770 | - | Growth Inhibition Assay | - | IC50=15.2868 μM | SANGER |
NCI-H1792 | - | Growth Inhibition Assay | - | IC50=12.3851 μM | SANGER |
NCI-H1793 | - | Growth Inhibition Assay | - | IC50=32.6163 μM | SANGER |
NCI-H187 | - | Growth Inhibition Assay | - | IC50=46.1869 μM | SANGER |
NCI-H1882 | - | Growth Inhibition Assay | - | IC50=21.8596 μM | SANGER |
NCI-H1963 | - | Growth Inhibition Assay | - | IC50=3.08825 μM | SANGER |
NCI-H2009 | - | Growth Inhibition Assay | - | IC50=5.30538 μM | SANGER |
NCI-H2030 | - | Growth Inhibition Assay | - | IC50=2.98029 μM | SANGER |
NCI-H2052 | - | Growth Inhibition Assay | - | IC50=10.5105 μM | SANGER |
NCI-H2081 | - | Growth Inhibition Assay | - | IC50=3.65288 μM | SANGER |
NCI-H2087 | - | Growth Inhibition Assay | - | IC50=2.71646 μM | SANGER |
NCI-H2122 | - | Growth Inhibition Assay | - | IC50=22.1677 μM | SANGER |
NCI-H2126 | - | Growth Inhibition Assay | - | IC50=7.09791 μM | SANGER |
NCI-H2141 | - | Growth Inhibition Assay | - | IC50=12.658 μM | SANGER |
NCI-H2170 | - | Growth Inhibition Assay | - | IC50=39.9977 μM | SANGER |
NCI-H2228 | - | Growth Inhibition Assay | - | IC50=31.5625 μM | SANGER |
NCI-H226 | - | Growth Inhibition Assay | - | IC50=18.8299 μM | SANGER |
NCI-H2342 | - | Growth Inhibition Assay | - | IC50=45.1117 μM | SANGER |
NCI-H2347 | - | Growth Inhibition Assay | - | IC50=6.94715 μM | SANGER |
NCI-H2405 | - | Growth Inhibition Assay | - | IC50=16.2218 μM | SANGER |
NCI-H2452 | - | Growth Inhibition Assay | - | IC50=10.6181 μM | SANGER |
NCI-H28 | - | Growth Inhibition Assay | - | IC50=29.012 μM | SANGER |
NCI-H292 | - | Growth Inhibition Assay | - | IC50=4.09429 μM | SANGER |
NCI-H358 | - | Growth Inhibition Assay | - | IC50=4.48532 μM | SANGER |
NCI-H441 | - | Growth Inhibition Assay | - | IC50=33.2235 μM | SANGER |
NCI-H446 | - | Growth Inhibition Assay | - | IC50=23.6093 μM | SANGER |
NCI-H460 | - | Growth Inhibition Assay | - | IC50=2.04839 μM | SANGER |
NCI-H522 | - | Growth Inhibition Assay | - | IC50=33.654 μM | SANGER |
NCI-H524 | - | Growth Inhibition Assay | - | IC50=19.5725 μM | SANGER |
NCI-H526 | - | Growth Inhibition Assay | - | IC50=3.13961 μM | SANGER |
NCI-H596 | - | Growth Inhibition Assay | - | IC50=31.0621 μM | SANGER |
NCI-H630 | - | Growth Inhibition Assay | - | IC50=30.8953 μM | SANGER |
NCI-H64 | - | Growth Inhibition Assay | - | IC50=21.4756 μM | SANGER |
NCI-H650 | - | Growth Inhibition Assay | - | IC50=0.83154 μM | SANGER |
NCI-H661 | - | Growth Inhibition Assay | - | IC50=24.5217 μM | SANGER |
NCI-H69 | - | Growth Inhibition Assay | - | IC50=12.0139 μM | SANGER |
NCI-H716 | - | Growth Inhibition Assay | - | IC50=9.93322 μM | SANGER |
NCI-H719 | - | Growth Inhibition Assay | - | IC50=9.18391 μM | SANGER |
NCI-H727 | - | Growth Inhibition Assay | - | IC50=22.8836 μM | SANGER |
NCI-H747 | - | Growth Inhibition Assay | - | IC50=4.08674 μM | SANGER |
NCI-H748 | - | Growth Inhibition Assay | - | IC50=18.8585 μM | SANGER |
NCI-H810 | - | Growth Inhibition Assay | - | IC50=1.10776 μM | SANGER |
NCI-H838 | - | Growth Inhibition Assay | - | IC50=6.51703 μM | SANGER |
NCI-SNU-1 | - | Growth Inhibition Assay | - | IC50=4.49701 μM | SANGER |
NEC8 | - | Growth Inhibition Assay | - | IC50=36.4924 μM | SANGER |
NH-12 | - | Growth Inhibition Assay | - | IC50=9.02542 μM | SANGER |
NKM-1 | - | Growth Inhibition Assay | - | IC50=1.27506 μM | SANGER |
NMC-G1 | - | Growth Inhibition Assay | - | IC50=5.09139 μM | SANGER |
no-10 | - | Growth Inhibition Assay | - | IC50=6.4784 μM | SANGER |
no-11 | - | Growth Inhibition Assay | - | IC50=36.8536 μM | SANGER |
NOMO-1 | - | Growth Inhibition Assay | - | IC50=3.49204 μM | SANGER |
NOS-1 | - | Growth Inhibition Assay | - | IC50=20.1577 μM | SANGER |
NTERA-S-cl-D1 | - | Growth Inhibition Assay | - | IC50=5.29218 μM | SANGER |
NUGC-3 | - | Growth Inhibition Assay | - | IC50=13.7453 μM | SANGER |
NY | - | Growth Inhibition Assay | - | IC50=28.6579 μM | SANGER |
OAW-42 | - | Growth Inhibition Assay | - | IC50=42.2942 μM | SANGER |
OCUB-M | - | Growth Inhibition Assay | - | IC50=21.9688 μM | SANGER |
OE19 | - | Growth Inhibition Assay | - | IC50=4.63145 μM | SANGER |
OE33 | - | Growth Inhibition Assay | - | IC50=12.9456 μM | SANGER |
ONS-76 | - | Growth Inhibition Assay | - | IC50=7.69416 μM | SANGER |
OPM-2 | - | Growth Inhibition Assay | - | IC50=2.89978 μM | SANGER |
OS-RC-2 | - | Growth Inhibition Assay | - | IC50=10.3227 μM | SANGER |
OVCAR-3 | - | Growth Inhibition Assay | - | IC50=5.88206 μM | SANGER |
OVCAR-4 | - | Growth Inhibition Assay | - | IC50=9.84828 μM | SANGER |
OVCAR-5 | - | Growth Inhibition Assay | - | IC50=3.36352 μM | SANGER |
OVCAR-8 | - | Growth Inhibition Assay | - | IC50=30.6794 μM | SANGER |
PA-1 | - | Growth Inhibition Assay | - | IC50=8.66694 μM | SANGER |
PANC-03-27 | - | Growth Inhibition Assay | - | IC50=8.3692 μM | SANGER |
PANC-08-13 | - | Growth Inhibition Assay | - | IC50=4.0773 μM | SANGER |
PANC-10-05 | - | Growth Inhibition Assay | - | IC50=20.4613 μM | SANGER |
PC-14 | - | Growth Inhibition Assay | - | IC50=23.6623 μM | SANGER |
PC-3 | - | Growth Inhibition Assay | - | IC50=6.13072 μM | SANGER |
PF-382 | - | Growth Inhibition Assay | - | IC50=40.7487 μM | SANGER |
PFSK-1 | - | Growth Inhibition Assay | - | IC50=21.6837 μM | SANGER |
PSN1 | - | Growth Inhibition Assay | - | IC50=48.1401 μM | SANGER |
Raji | - | Growth Inhibition Assay | - | IC50=20.2568 μM | SANGER |
RCC10RGB | - | Growth Inhibition Assay | - | IC50=2.32507 μM | SANGER |
RCM-1 | - | Growth Inhibition Assay | - | IC50=37.5358 μM | SANGER |
RD | - | Growth Inhibition Assay | - | IC50=5.29771 μM | SANGER |
REH | - | Growth Inhibition Assay | - | IC50=12.1573 μM | SANGER |
RERF-LC-MS | - | Growth Inhibition Assay | - | IC50=8.48595 μM | SANGER |
RKO | - | Growth Inhibition Assay | - | IC50=21.3202 μM | SANGER |
RL95-2 | - | Growth Inhibition Assay | - | IC50=3.71864 μM | SANGER |
RO82-W-1 | - | Growth Inhibition Assay | - | IC50=23.2511 μM | SANGER |
RPMI-2650 | - | Growth Inhibition Assay | - | IC50=4.12975 μM | SANGER |
RPMI-7951 | - | Growth Inhibition Assay | - | IC50=3.20137 μM | SANGER |
RPMI-8402 | - | Growth Inhibition Assay | - | IC50=13.5031 μM | SANGER |
RS4-11 | - | Growth Inhibition Assay | - | IC50=3.48715 μM | SANGER |
RT-112 | - | Growth Inhibition Assay | - | IC50=0.9846 μM | SANGER |
RT4 | - | Growth Inhibition Assay | - | IC50=48.8377 μM | SANGER |
RVH-421 | - | Growth Inhibition Assay | - | IC50=3.60311 μM | SANGER |
RXF393 | - | Growth Inhibition Assay | - | IC50=10.1392 μM | SANGER |
Saos-2 | - | Growth Inhibition Assay | - | IC50=47.3123 μM | SANGER |
SAS | - | Growth Inhibition Assay | - | IC50=43.4288 μM | SANGER |
SBC-5 | - | Growth Inhibition Assay | - | IC50=3.67882 μM | SANGER |
SCC-15 | - | Growth Inhibition Assay | - | IC50=2.75252 μM | SANGER |
SCC-25 | - | Growth Inhibition Assay | - | IC50=6.42493 μM | SANGER |
SCC-4 | - | Growth Inhibition Assay | - | IC50=3.95782 μM | SANGER |
SCC-9 | - | Growth Inhibition Assay | - | IC50=4.44299 μM | SANGER |
SF126 | - | Growth Inhibition Assay | - | IC50=5.41465 μM | SANGER |
SF268 | - | Growth Inhibition Assay | - | IC50=7.8356 μM | SANGER |
SF295 | - | Growth Inhibition Assay | - | IC50=6.4498 μM | SANGER |
SF539 | - | Growth Inhibition Assay | - | IC50=9.21098 μM | SANGER |
SH-4 | - | Growth Inhibition Assay | - | IC50=4.72633 μM | SANGER |
SIG-M5 | - | Growth Inhibition Assay | - | IC50=1.48387 μM | SANGER |
SIMA | - | Growth Inhibition Assay | - | IC50=4.144 μM | SANGER |
SJRH30 | - | Growth Inhibition Assay | - | IC50=10.1844 μM | SANGER |
SJSA-1 | - | Growth Inhibition Assay | - | IC50=16.9219 μM | SANGER |
SK-CO-1 | - | Growth Inhibition Assay | - | IC50=9.76235 μM | SANGER |
SKG-IIIa | - | Growth Inhibition Assay | - | IC50=23.3546 μM | SANGER |
SK-HEP-1 | - | Growth Inhibition Assay | - | IC50=8.35723 μM | SANGER |
SK-LMS-1 | - | Growth Inhibition Assay | - | IC50=9.75535 μM | SANGER |
SK-LU-1 | - | Growth Inhibition Assay | - | IC50=2.98334 μM | SANGER |
SK-MEL-2 | - | Growth Inhibition Assay | - | IC50=19.2155 μM | SANGER |
SK-MEL-24 | - | Growth Inhibition Assay | - | IC50=29.5466 μM | SANGER |
SK-MEL-30 | - | Growth Inhibition Assay | - | IC50=6.96315 μM | SANGER |
SK-MES-1 | - | Growth Inhibition Assay | - | IC50=5.85891 μM | SANGER |
SK-MM-2 | - | Growth Inhibition Assay | - | IC50=12.4087 μM | SANGER |
SK-N-AS | - | Growth Inhibition Assay | - | IC50=28.3171 μM | SANGER |
SK-N-DZ | - | Growth Inhibition Assay | - | IC50=24.4977 μM | SANGER |
SK-NEP-1 | - | Growth Inhibition Assay | - | IC50=6.4036 μM | SANGER |
SK-OV-3 | - | Growth Inhibition Assay | - | IC50=8.79772 μM | SANGER |
SK-PN-DW | - | Growth Inhibition Assay | - | IC50=2.86204 μM | SANGER |
SK-UT-1 | - | Growth Inhibition Assay | - | IC50=1.44647 μM | SANGER |
SN12C | - | Growth Inhibition Assay | - | IC50=9.76806 μM | SANGER |
SNB75 | - | Growth Inhibition Assay | - | IC50=4.7466 μM | SANGER |
SNU-387 | - | Growth Inhibition Assay | - | IC50=2.5282 μM | SANGER |
SNU-423 | - | Growth Inhibition Assay | - | IC50=4.42685 μM | SANGER |
SNU-449 | - | Growth Inhibition Assay | - | IC50=11.6072 μM | SANGER |
SNU-C1 | - | Growth Inhibition Assay | - | IC50=27.6491 μM | SANGER |
SNU-C2B | - | Growth Inhibition Assay | - | IC50=22.6746 μM | SANGER |
SR | - | Growth Inhibition Assay | - | IC50=5.53645 μM | SANGER |
ST486 | - | Growth Inhibition Assay | - | IC50=1.53278 μM | SANGER |
SUP-T1 | - | Growth Inhibition Assay | - | IC50=3.7832 μM | SANGER |
SW13 | - | Growth Inhibition Assay | - | IC50=10.6374 μM | SANGER |
SW1463 | - | Growth Inhibition Assay | - | IC50=36.6566 μM | SANGER |
SW1573 | - | Growth Inhibition Assay | - | IC50=23.0646 μM | SANGER |
SW1710 | - | Growth Inhibition Assay | - | IC50=1.62628 μM | SANGER |
SW1990 | - | Growth Inhibition Assay | - | IC50=24.5883 μM | SANGER |
SW48 | - | Growth Inhibition Assay | - | IC50=32.3825 μM | SANGER |
SW620 | - | Growth Inhibition Assay | - | IC50=31.6283 μM | SANGER |
SW626 | - | Growth Inhibition Assay | - | IC50=11.2889 μM | SANGER |
SW684 | - | Growth Inhibition Assay | - | IC50=24.7624 μM | SANGER |
SW756 | - | Growth Inhibition Assay | - | IC50=39.5091 μM | SANGER |
SW780 | - | Growth Inhibition Assay | - | IC50=4.76849 μM | SANGER |
SW872 | - | Growth Inhibition Assay | - | IC50=3.76958 μM | SANGER |
SW948 | - | Growth Inhibition Assay | - | IC50=13.013 μM | SANGER |
SW954 | - | Growth Inhibition Assay | - | IC50=2.00151 μM | SANGER |
SW962 | - | Growth Inhibition Assay | - | IC50=30.2477 μM | SANGER |
SW982 | - | Growth Inhibition Assay | - | IC50=0.3282 μM | SANGER |
T-24 | - | Growth Inhibition Assay | - | IC50=28.1925 μM | SANGER |
T98G | - | Growth Inhibition Assay | - | IC50=27.1973 μM | SANGER |
TE-1 | - | Growth Inhibition Assay | - | IC50=29.2167 μM | SANGER |
TE-10 | - | Growth Inhibition Assay | - | IC50=4.22887 μM | SANGER |
TE-11 | - | Growth Inhibition Assay | - | IC50=1.63522 μM | SANGER |
TE-12 | - | Growth Inhibition Assay | - | IC50=6.72377 μM | SANGER |
TE-15 | - | Growth Inhibition Assay | - | IC50=5.57779 μM | SANGER |
TE-441-T | - | Growth Inhibition Assay | - | IC50=3.8293 μM | SANGER |
TE-5 | - | Growth Inhibition Assay | - | IC50=8.70296 μM | SANGER |
TE-6 | - | Growth Inhibition Assay | - | IC50=5.44569 μM | SANGER |
TE-8 | - | Growth Inhibition Assay | - | IC50=18.0669 μM | SANGER |
TE-9 | - | Growth Inhibition Assay | - | IC50=5.61788 μM | SANGER |
TGBC1TKB | - | Growth Inhibition Assay | - | IC50=23.7461 μM | SANGER |
TGBC24TKB | - | Growth Inhibition Assay | - | IC50=38.0239 μM | SANGER |
TGW | - | Growth Inhibition Assay | - | IC50=25.2337 μM | SANGER |
THP-1 | - | Growth Inhibition Assay | - | IC50=16.4665 μM | SANGER |
TK10 | - | Growth Inhibition Assay | - | IC50=16.3742 μM | SANGER |
TUR | - | Growth Inhibition Assay | - | IC50=2.65369 μM | SANGER |
U031 | - | Growth Inhibition Assay | - | IC50=19.2219 μM | SANGER |
U251 | - | Growth Inhibition Assay | - | IC50=1.74031 μM | SANGER |
U-266 | - | Growth Inhibition Assay | - | IC50=4.94919 μM | SANGER |
U-2-OS | - | Growth Inhibition Assay | - | IC50=27.0271 μM | SANGER |
U-698-M | - | Growth Inhibition Assay | - | IC50=9.997 μM | SANGER |
U-87-MG | - | Growth Inhibition Assay | - | IC50=26.5305 μM | SANGER |
UACC-257 | - | Growth Inhibition Assay | - | IC50=18.2062 μM | SANGER |
UACC-62 | - | Growth Inhibition Assay | - | IC50=9.37297 μM | SANGER |
UMC-11 | - | Growth Inhibition Assay | - | IC50=10.9373 μM | SANGER |
VA-ES-BJ | - | Growth Inhibition Assay | - | IC50=1.90315 μM | SANGER |
VM-CUB-1 | - | Growth Inhibition Assay | - | IC50=3.7751 μM | SANGER |
VMRC-RCZ | - | Growth Inhibition Assay | - | IC50=14.236 μM | SANGER |
YAPC | - | Growth Inhibition Assay | - | IC50=14.2407 μM | SANGER |
YKG-1 | - | Growth Inhibition Assay | - | IC50=7.02678 μM | SANGER |
YT | - | Growth Inhibition Assay | - | IC50=10.4001 μM | SANGER |
22RV1 | - | Growth Inhibition Assay | - | IC50=7.67975 μM | SANGER |
23132-87 | - | Growth Inhibition Assay | - | IC50=6.90901 μM | SANGER |
5637 | - | Growth Inhibition Assay | - | IC50=2.92439 μM | SANGER |
639-V | - | Growth Inhibition Assay | - | IC50=6.75127 μM | SANGER |
647-V | - | Growth Inhibition Assay | - | IC50=5.62042 μM | SANGER |
697 | - | Growth Inhibition Assay | - | IC50=3.81657 μM | SANGER |
769-P | - | Growth Inhibition Assay | - | IC50=12.019 μM | SANGER |
786-0 | - | Growth Inhibition Assay | - | IC50=3.05784 μM | SANGER |
8305C | - | Growth Inhibition Assay | - | IC50=1.09904 μM | SANGER |
8505C | - | Growth Inhibition Assay | - | IC50=12.612 μM | SANGER |
8-MG-BA | - | Growth Inhibition Assay | - | IC50=5.37077 μM | SANGER |
A101D | - | Growth Inhibition Assay | - | IC50=5.39689 μM | SANGER |
A172 | - | Growth Inhibition Assay | - | IC50=12.1207 μM | SANGER |
A204 | - | Growth Inhibition Assay | - | IC50=3.90956 μM | SANGER |
A2058 | - | Growth Inhibition Assay | - | IC50=5.30438 μM | SANGER |
A253 | - | Growth Inhibition Assay | - | IC50=17.825 μM | SANGER |
A2780 | - | Growth Inhibition Assay | - | IC50=3.10341 μM | SANGER |
A375 | - | Growth Inhibition Assay | - | IC50=37.7647 μM | SANGER |
A3-KAW | - | Growth Inhibition Assay | - | IC50=4.35552 μM | SANGER |
A431 | - | Growth Inhibition Assay | - | IC50=4.68228 μM | SANGER |
A498 | - | Growth Inhibition Assay | - | IC50=22.8177 μM | SANGER |
A4-Fuk | - | Growth Inhibition Assay | - | IC50=4.07861 μM | SANGER |
A673 | - | Growth Inhibition Assay | - | IC50=29.732 μM | SANGER |
ABC-1 | - | Growth Inhibition Assay | - | IC50=2.25196 μM | SANGER |
ACHN | - | Growth Inhibition Assay | - | IC50=4.0237 μM | SANGER |
ACN | - | Growth Inhibition Assay | - | IC50=2.34745 μM | SANGER |
AGS | - | Growth Inhibition Assay | - | IC50=1.52124 μM | SANGER |
ALL-PO | - | Growth Inhibition Assay | - | IC50=1.01584 μM | SANGER |
AM-38 | - | Growth Inhibition Assay | - | IC50=8.80439 μM | SANGER |
AN3-CA | - | Growth Inhibition Assay | - | IC50=1.21867 μM | SANGER |
ATN-1 | - | Growth Inhibition Assay | - | IC50=4.10777 μM | SANGER |
BB30-HNC | - | Growth Inhibition Assay | - | IC50=7.94553 μM | SANGER |
BB49-HNC | - | Growth Inhibition Assay | - | IC50=31.112 μM | SANGER |
BC-1 | - | Growth Inhibition Assay | - | IC50=1.61664 μM | SANGER |
BC-3 | - | Growth Inhibition Assay | - | IC50=4.43477 μM | SANGER |
BCPAP | - | Growth Inhibition Assay | - | IC50=1.01288 μM | SANGER |
Becker | - | Growth Inhibition Assay | - | IC50=15.8926 μM | SANGER |
BFTC-905 | - | Growth Inhibition Assay | - | IC50=5.60421 μM | SANGER |
BHT-101 | - | Growth Inhibition Assay | - | IC50=3.15798 μM | SANGER |
BHY | - | Growth Inhibition Assay | - | IC50=1.65663 μM | SANGER |
BL-41 | - | Growth Inhibition Assay | - | IC50=11.7173 μM | SANGER |
BL-70 | - | Growth Inhibition Assay | - | IC50=46.7737 μM | SANGER |
BPH-1 | - | Growth Inhibition Assay | - | IC50=1.28766 μM | SANGER |
BT-20 | - | Growth Inhibition Assay | - | IC50=14.9384 μM | SANGER |
BV-173 | - | Growth Inhibition Assay | - | IC50=35.8264 μM | SANGER |
BxPC-3 | - | Growth Inhibition Assay | - | IC50=2.35436 μM | SANGER |
C2BBe1 | - | Growth Inhibition Assay | - | IC50=9.39652 μM | SANGER |
C-33-A | - | Growth Inhibition Assay | - | IC50=8.61529 μM | SANGER |
C3A | - | Growth Inhibition Assay | - | IC50=8.76561 μM | SANGER |
C-4-II | - | Growth Inhibition Assay | - | IC50=6.83117 μM | SANGER |
C8166 | - | Growth Inhibition Assay | - | IC50=4.47753 μM | SANGER |
CA46 | - | Growth Inhibition Assay | - | IC50=4.16104 μM | SANGER |
Ca9-22 | - | Growth Inhibition Assay | - | IC50=4.55516 μM | SANGER |
CAKI-1 | - | Growth Inhibition Assay | - | IC50=8.06521 μM | SANGER |
CAL-120 | - | Growth Inhibition Assay | - | IC50=3.5735 μM | SANGER |
CAL-12T | - | Growth Inhibition Assay | - | IC50=14.4336 μM | SANGER |
CAL-27 | - | Growth Inhibition Assay | - | IC50=12.1369 μM | SANGER |
CAL-33 | - | Growth Inhibition Assay | - | IC50=1.12938 μM | SANGER |
CAL-39 | - | Growth Inhibition Assay | - | IC50=2.41628 μM | SANGER |
CAL-51 | - | Growth Inhibition Assay | - | IC50=3.57612 μM | SANGER |
CAL-54 | - | Growth Inhibition Assay | - | IC50=29.6046 μM | SANGER |
CAL-62 | - | Growth Inhibition Assay | - | IC50=1.31909 μM | SANGER |
CAL-72 | - | Growth Inhibition Assay | - | IC50=14.1906 μM | SANGER |
CAL-85-1 | - | Growth Inhibition Assay | - | IC50=1.8049 μM | SANGER |
Calu-1 | - | Growth Inhibition Assay | - | IC50=4.58707 μM | SANGER |
Calu-3 | - | Growth Inhibition Assay | - | IC50=6.14689 μM | SANGER |
Calu-6 | - | Growth Inhibition Assay | - | IC50=6.65435 μM | SANGER |
CAMA-1 | - | Growth Inhibition Assay | - | IC50=9.06012 μM | SANGER |
CAPAN-1 | - | Growth Inhibition Assay | - | IC50=25.7501 μM | SANGER |
Capan-2 | - | Growth Inhibition Assay | - | IC50=39.0509 μM | SANGER |
CaR-1 | - | Growth Inhibition Assay | - | IC50=25.357 μM | SANGER |
CAS-1 | - | Growth Inhibition Assay | - | IC50=10.4608 μM | SANGER |
Ca-Ski | - | Growth Inhibition Assay | - | IC50=24.9237 μM | SANGER |
CCF-STTG1 | - | Growth Inhibition Assay | - | IC50=13.4039 μM | SANGER |
CCRF-CEM | - | Growth Inhibition Assay | - | IC50=25.7459 μM | SANGER |
CESS | - | Growth Inhibition Assay | - | IC50=17.9326 μM | SANGER |
CGTH-W-1 | - | Growth Inhibition Assay | - | IC50=1.61679 μM | SANGER |
ChaGo-K-1 | - | Growth Inhibition Assay | - | IC50=10.1776 μM | SANGER |
CHL-1 | - | Growth Inhibition Assay | - | IC50=4.18961 μM | SANGER |
CHP-126 | - | Growth Inhibition Assay | - | IC50=9.9329 μM | SANGER |
CHP-212 | - | Growth Inhibition Assay | - | IC50=2.09539 μM | SANGER |
CMK | - | Growth Inhibition Assay | - | IC50=2.41795 μM | SANGER |
COLO-205 | - | Growth Inhibition Assay | - | IC50=0.48658 μM | SANGER |
COLO-320-HSR | - | Growth Inhibition Assay | - | IC50=11.8519 μM | SANGER |
COLO-678 | - | Growth Inhibition Assay | - | IC50=40.595 μM | SANGER |
COLO-679 | - | Growth Inhibition Assay | - | IC50=10.4285 μM | SANGER |
COLO-680N | - | Growth Inhibition Assay | - | IC50=6.37638 μM | SANGER |
COLO-684 | - | Growth Inhibition Assay | - | IC50=5.25371 μM | SANGER |
COLO-792 | - | Growth Inhibition Assay | - | IC50=21.5827 μM | SANGER |
COLO-800 | - | Growth Inhibition Assay | - | IC50=7.90685 μM | SANGER |
COLO-824 | - | Growth Inhibition Assay | - | IC50=6.27868 μM | SANGER |
COLO-829 | - | Growth Inhibition Assay | - | IC50=0.75176 μM | SANGER |
COR-L105 | - | Growth Inhibition Assay | - | IC50=11.3237 μM | SANGER |
COR-L23 | - | Growth Inhibition Assay | - | IC50=4.6728 μM | SANGER |
CP50-MEL-B | - | Growth Inhibition Assay | - | IC50=25.9901 μM | SANGER |
CP66-MEL | - | Growth Inhibition Assay | - | IC50=46.2789 μM | SANGER |
CTV-1 | - | Growth Inhibition Assay | - | IC50=3.25377 μM | SANGER |
D-247MG | - | Growth Inhibition Assay | - | IC50=25.4743 μM | SANGER |
D-263MG | - | Growth Inhibition Assay | - | IC50=31.0424 μM | SANGER |
D-283MED | - | Growth Inhibition Assay | - | IC50=28.8708 μM | SANGER |
D-336MG | - | Growth Inhibition Assay | - | IC50=1.85614 μM | SANGER |
Daoy | - | Growth Inhibition Assay | - | IC50=9.24143 μM | SANGER |
Daudi | - | Growth Inhibition Assay | - | IC50=26.5158 μM | SANGER |
DB | - | Growth Inhibition Assay | - | IC50=15.6941 μM | SANGER |
DBTRG-05MG | - | Growth Inhibition Assay | - | IC50=3.81676 μM | SANGER |
DEL | - | Growth Inhibition Assay | - | IC50=13.5503 μM | SANGER |
Detroit562 | - | Growth Inhibition Assay | - | IC50=1.35222 μM | SANGER |
DJM-1 | - | Growth Inhibition Assay | - | IC50=32.1386 μM | SANGER |
DMS-273 | - | Growth Inhibition Assay | - | IC50=9.125 μM | SANGER |
DOK | - | Growth Inhibition Assay | - | IC50=21.7687 μM | SANGER |
DoTc2-4510 | - | Growth Inhibition Assay | - | IC50=11.1389 μM | SANGER |
DSH1 | - | Growth Inhibition Assay | - | IC50=26.5406 μM | SANGER |
DU-145 | - | Growth Inhibition Assay | - | IC50=2.49118 μM | SANGER |
DU-4475 | - | Growth Inhibition Assay | - | IC50=2.14759 μM | SANGER |
DV-90 | - | Growth Inhibition Assay | - | IC50=4.29397 μM | SANGER |
EB2 | - | Growth Inhibition Assay | - | IC50=17.7426 μM | SANGER |
ECC12 | - | Growth Inhibition Assay | - | IC50=7.72901 μM | SANGER |
EFE-184 | - | Growth Inhibition Assay | - | IC50=35.6829 μM | SANGER |
EFM-19 | - | Growth Inhibition Assay | - | IC50=24.1844 μM | SANGER |
EFO-21 | - | Growth Inhibition Assay | - | IC50=10.0093 μM | SANGER |
EFO-27 | - | Growth Inhibition Assay | - | IC50=2.51888 μM | SANGER |
EGI-1 | - | Growth Inhibition Assay | - | IC50=10.9455 μM | SANGER |
EHEB | - | Growth Inhibition Assay | - | IC50=33.0494 μM | SANGER |
EKVX | - | Growth Inhibition Assay | - | IC50=49.6731 μM | SANGER |
EM-2 | - | Growth Inhibition Assay | - | IC50=3.48674 μM | SANGER |
EoL-1-cell | - | Growth Inhibition Assay | - | IC50=44.9136 μM | SANGER |
ES4 | - | Growth Inhibition Assay | - | IC50=12.9487 μM | SANGER |
ES5 | - | Growth Inhibition Assay | - | IC50=14.2599 μM | SANGER |
ES6 | - | Growth Inhibition Assay | - | IC50=11.576 μM | SANGER |
ES8 | - | Growth Inhibition Assay | - | IC50=5.41409 μM | SANGER |
ESS-1 | - | Growth Inhibition Assay | - | IC50=6.76072 μM | SANGER |
ETK-1 | - | Growth Inhibition Assay | - | IC50=2.2846 μM | SANGER |
EW-1 | - | Growth Inhibition Assay | - | IC50=3.40544 μM | SANGER |
EW-11 | - | Growth Inhibition Assay | - | IC50=17.9958 μM | SANGER |
EW-13 | - | Growth Inhibition Assay | - | IC50=1.63466 μM | SANGER |
EW-16 | - | Growth Inhibition Assay | - | IC50=2.03983 μM | SANGER |
EW-18 | - | Growth Inhibition Assay | - | IC50=3.0532 μM | SANGER |
EW-7 | - | Growth Inhibition Assay | - | IC50=20.1628 μM | SANGER |
FADU | - | Growth Inhibition Assay | - | IC50=26.5152 μM | SANGER |
G-361 | - | Growth Inhibition Assay | - | IC50=4.0906 μM | SANGER |
G-401 | - | Growth Inhibition Assay | - | IC50=3.29808 μM | SANGER |
G-402 | - | Growth Inhibition Assay | - | IC50=2.81447 μM | SANGER |
GAMG | - | Growth Inhibition Assay | - | IC50=14.5577 μM | SANGER |
GB-1 | - | Growth Inhibition Assay | - | IC50=11.7619 μM | SANGER |
GCIY | - | Growth Inhibition Assay | - | IC50=8.23713 μM | SANGER |
GDM-1 | - | Growth Inhibition Assay | - | IC50=5.41781 μM | SANGER |
GI-1 | - | Growth Inhibition Assay | - | IC50=6.94348 μM | SANGER |
GI-ME-N | - | Growth Inhibition Assay | - | IC50=7.16906 μM | SANGER |
GOTO | - | Growth Inhibition Assay | - | IC50=4.79293 μM | SANGER |
GP5d | - | Growth Inhibition Assay | - | IC50=2.83827 μM | SANGER |
GR-ST | - | Growth Inhibition Assay | - | IC50=11.6181 μM | SANGER |
GT3TKB | - | Growth Inhibition Assay | - | IC50=4.48822 μM | SANGER |
H4 | - | Growth Inhibition Assay | - | IC50=3.47569 μM | SANGER |
HAL-01 | - | Growth Inhibition Assay | - | IC50=12.6174 μM | SANGER |
HC-1 | - | Growth Inhibition Assay | - | IC50=35.4024 μM | SANGER |
HCC1143 | - | Growth Inhibition Assay | - | IC50=7.37898 μM | SANGER |
HCC1187 | - | Growth Inhibition Assay | - | IC50=19.1796 μM | SANGER |
HCC1569 | - | Growth Inhibition Assay | - | IC50=46.5917 μM | SANGER |
HCC1806 | - | Growth Inhibition Assay | - | IC50=12.6952 μM | SANGER |
HCC1937 | - | Growth Inhibition Assay | - | IC50=37.0154 μM | SANGER |
HCC2157 | - | Growth Inhibition Assay | - | IC50=5.56896 μM | SANGER |
HCC2218 | - | Growth Inhibition Assay | - | IC50=35.2185 μM | SANGER |
HCC2998 | - | Growth Inhibition Assay | - | IC50=3.94843 μM | SANGER |
HCC70 | - | Growth Inhibition Assay | - | IC50=9.27309 μM | SANGER |
HCE-T | - | Growth Inhibition Assay | - | IC50=21.5094 μM | SANGER |
HCT-116 | - | Growth Inhibition Assay | - | IC50=3.50711 μM | SANGER |
HDLM-2 | - | Growth Inhibition Assay | - | IC50=28.2459 μM | SANGER |
HEC-1 | - | Growth Inhibition Assay | - | IC50=30.0053 μM | SANGER |
HEL | - | Growth Inhibition Assay | - | IC50=6.02188 μM | SANGER |
HGC-27 | - | Growth Inhibition Assay | - | IC50=4.09549 μM | SANGER |
HH | - | Growth Inhibition Assay | - | IC50=35.4141 μM | SANGER |
HL-60 | - | Growth Inhibition Assay | - | IC50=3.2114 μM | SANGER |
HLE | - | Growth Inhibition Assay | - | IC50=11.2119 μM | SANGER |
HMV-II | - | Growth Inhibition Assay | - | IC50=2.58997 μM | SANGER |
HO-1-N-1 | - | Growth Inhibition Assay | - | IC50=7.24024 μM | SANGER |
HOP-62 | - | Growth Inhibition Assay | - | IC50=5.56887 μM | SANGER |
HOP-92 | - | Growth Inhibition Assay | - | IC50=2.30673 μM | SANGER |
HOS | - | Growth Inhibition Assay | - | IC50=4.38567 μM | SANGER |
HSC-2 | - | Growth Inhibition Assay | - | IC50=1.5395 μM | SANGER |
HSC-3 | - | Growth Inhibition Assay | - | IC50=6.17396 μM | SANGER |
HSC-4 | - | Growth Inhibition Assay | - | IC50=2.78389 μM | SANGER |
HT | - | Growth Inhibition Assay | - | IC50=12.9437 μM | SANGER |
HT-1080 | - | Growth Inhibition Assay | - | IC50=7.78555 μM | SANGER |
HT-1376 | - | Growth Inhibition Assay | - | IC50=19.2029 μM | SANGER |
HT-144 | - | Growth Inhibition Assay | - | IC50=15.9497 μM | SANGER |
HT-29 | - | Growth Inhibition Assay | - | IC50=9.12373 μM | SANGER |
HT-3 | - | Growth Inhibition Assay | - | IC50=7.0349 μM | SANGER |
HTC-C3 | - | Growth Inhibition Assay | - | IC50=9.77984 μM | SANGER |
HuCCT1 | - | Growth Inhibition Assay | - | IC50=4.33723 μM | SANGER |
HuH-7 | - | Growth Inhibition Assay | - | IC50=26.9086 μM | SANGER |
HuO9 | - | Growth Inhibition Assay | - | IC50=7.48794 μM | SANGER |
HuP-T3 | - | Growth Inhibition Assay | - | IC50=28.0495 μM | SANGER |
HuP-T4 | - | Growth Inhibition Assay | - | IC50=10.7068 μM | SANGER |
HUTU-80 | - | Growth Inhibition Assay | - | IC50=1.44886 μM | SANGER |
IA-LM | - | Growth Inhibition Assay | - | IC50=33.6746 μM | SANGER |
IGR-1 | - | Growth Inhibition Assay | - | IC50=2.83987 μM | SANGER |
IGROV-1 | - | Growth Inhibition Assay | - | IC50=0.81038 μM | SANGER |
IMR-5 | - | Growth Inhibition Assay | - | IC50=22.287 μM | SANGER |
IPC-298 | - | Growth Inhibition Assay | - | IC50=8.27709 μM | SANGER |
IST-MEL1 | - | Growth Inhibition Assay | - | IC50=19.1754 μM | SANGER |
IST-MES1 | - | Growth Inhibition Assay | - | IC50=49.8944 μM | SANGER |
IST-SL1 | - | Growth Inhibition Assay | - | IC50=3.29465 μM | SANGER |
IST-SL2 | - | Growth Inhibition Assay | - | IC50=7.52272 μM | SANGER |
J82 | - | Growth Inhibition Assay | - | IC50=8.34124 μM | SANGER |
JiyoyeP-2003 | - | Growth Inhibition Assay | - | IC50=11.0892 μM | SANGER |
J-RT3-T3-5 | - | Growth Inhibition Assay | - | IC50=11.1209 μM | SANGER |
K5 | - | Growth Inhibition Assay | - | IC50=21.3893 μM | SANGER |
K-562 | - | Growth Inhibition Assay | - | IC50=21.4971 μM | SANGER |
KALS-1 | - | Growth Inhibition Assay | - | IC50=15.0158 μM | SANGER |
KARPAS-422 | - | Growth Inhibition Assay | - | IC50=37.4431 μM | SANGER |
KARPAS-45 | - | Growth Inhibition Assay | - | IC50=6.03787 μM | SANGER |
KASUMI-1 | - | Growth Inhibition Assay | - | IC50=2.3288 μM | SANGER |
靶点 | Description | IC50 |
---|---|---|
FAK | IC50:1.5nM | |
Pyk2 | IC50:13nM |
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