400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / MAPK/ERK Pathway / ERK / SCH772984
CAS No.: 942183-80-4
Synonyms: SCH772984
SCH772984 is a specific inhibitor of ERK1/2 with IC50 of 4 nM and 1 nM, respectively.
生物活性
实验方案
技术信息
CAS号 | 942183-80-4 | 储存条件 |
|
|||||||||||||
分子式 | C33H33N9O2 | 运输 | 蓝冰 | |||||||||||||
分子量 | 587.67 | 别名 | SCH772984 | |||||||||||||
溶解度 |
|
动物实验配方 |
|
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
---|
2P-ERK2 | - | Growth Inhibition Assay | - | IC50=0.24 nM | 25350931 |
5637 | - | Growth Inhibition Assay | - | IC50=610 nM | 23614898 |
769P | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
786-O | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
8505C | - | Growth Inhibition Assay | - | IC50=50 nM | 23614898 |
A172 | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
A204 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
A2058 | - | Growth Inhibition Assay | - | IC50=360 nM | 23614898 |
A2780 | - | Growth Inhibition Assay | - | IC50=143 nM | 23614898 |
A375-SM | - | Growth Inhibition Assay | - | IC50=75 nM | 23614898 |
A427 | - | Growth Inhibition Assay | - | IC50=1433 nM | 23614898 |
A498 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
A549 | - | Growth Inhibition Assay | - | IC50=326 nM | 23614898 |
A673 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
ACHN | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
AsPc-1 | - | Growth Inhibition Assay | - | IC50=270 nM | 23614898 |
BHT-101 | - | Growth Inhibition Assay | - | IC50=300 nM | 23614898 |
BT-474 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
Caki-1 | - | Growth Inhibition Assay | - | IC50=450 nM | 23614898 |
CAPAN-1 | - | Growth Inhibition Assay | - | IC50=104 nM | 23614898 |
CFPAC-1 | - | Growth Inhibition Assay | - | IC50=1001 nM | 23614898 |
CHL-1 | - | Growth Inhibition Assay | - | IC50=1460 nM | 23614898 |
Colo-205 | - | Growth Inhibition Assay | - | IC50=36 nM | 23614898 |
DAOY | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
Daudi | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
DBTRG-05MG | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
DLD-1 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
DU145 | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
EKVX | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
ES-2 | - | Growth Inhibition Assay | - | IC50=2659 nM | 23614898 |
FTC-133 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
H226 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
H23 | - | Growth Inhibition Assay | - | IC50=1000 nM | 23614898 |
H322 | - | Growth Inhibition Assay | - | IC50=325 nM | 23614898 |
H522 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
H716 | - | Growth Inhibition Assay | - | IC50=334 nM | 23614898 |
HCT-116 | - | Growth Inhibition Assay | - | IC50=128 nM | 23614898 |
HCT-15 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
HCT-8 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
HeLa | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
HL-60 | - | Growth Inhibition Assay | - | IC50=30 nM | 23614898 |
HOP62 | - | Growth Inhibition Assay | - | IC50=676 nM | 23614898 |
HOP92 | - | Growth Inhibition Assay | - | IC50=820 nM | 23614898 |
HPAC | - | Growth Inhibition Assay | - | IC50=170 nM | 23614898 |
Hs-294T | - | Growth Inhibition Assay | - | IC50=945 nM | 23614898 |
Hs-695T | - | Growth Inhibition Assay | - | IC50=165 nM | 23614898 |
HS746T | - | Growth Inhibition Assay | - | IC50=1000 nM | 23614898 |
HT-1197 | - | Growth Inhibition Assay | - | IC50=316 nM | 23614898 |
HT-1376 | - | Growth Inhibition Assay | - | IC50=2800 nM | 23614898 |
HT-144 | - | Growth Inhibition Assay | - | IC50=60 nM | 23614898 |
HT-29 | - | Growth Inhibition Assay | - | IC50=50 nM | 23614898 |
HTB-177 | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
IGROV-1 | - | Growth Inhibition Assay | - | IC50=146 nM | 23614898 |
J-82 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
Jijoye | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
Jurkat | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
K1 | - | Growth Inhibition Assay | - | IC50=130 nM | 23614898 |
K562 | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
KG-1 | - | Growth Inhibition Assay | - | IC50=900 nM | 23614898 |
Ln Cap | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
LoVo | - | Growth Inhibition Assay | - | IC50=47 nM | 23614898 |
LOX | - | Growth Inhibition Assay | - | IC50=100 nM | 23614898 |
M14 | - | Growth Inhibition Assay | - | IC50=47 nM | 23614898 |
MB-231 | - | Growth Inhibition Assay | - | IC50=1000 nM | 23614898 |
MB-453 | - | Growth Inhibition Assay | - | IC50=672 nM | 23614898 |
MB-468 | - | Growth Inhibition Assay | - | IC50=1000 nM | 23614898 |
MCF-7 | - | Growth Inhibition Assay | - | IC50=1001 nM | 23614898 |
MDAH-2774 | - | Growth Inhibition Assay | - | IC50=2657 nM | 23614898 |
MiaPaCa | - | Growth Inhibition Assay | - | IC50=53 nM | 23614898 |
Molt-3 | - | Growth Inhibition Assay | - | IC50=600 nM | 23614898 |
Molt-4 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
N-87 | - | Growth Inhibition Assay | - | IC50=307 nM | 23614898 |
NCI-H157 | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
NCI-H292 | - | Growth Inhibition Assay | - | IC50=90 nM | 23614898 |
NCI-H520 | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
OVCAR-5 | - | Growth Inhibition Assay | - | IC50=208 nM | 23614898 |
PA-1 | - | Growth Inhibition Assay | - | IC50=1001 nM | 23614898 |
Panc-1 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
PC3 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
RD | - | Growth Inhibition Assay | - | IC50=123 nM | 23614898 |
Ro82-W-1 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
RPMI-7951 | - | Growth Inhibition Assay | - | IC50=344 nM | 23614898 |
RT-4 | - | Growth Inhibition Assay | - | IC50=810 nM | 23614898 |
SCABER | - | Growth Inhibition Assay | - | IC50=1000 nM | 23614898 |
SF-268 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
SF-295 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
SF-539 | - | Growth Inhibition Assay | - | IC50=1000 nM | 23614898 |
SJCRH30 | - | Growth Inhibition Assay | - | IC50=2002 nM | 23614898 |
SK-Hep-1 | - | Growth Inhibition Assay | - | IC50=1422 nM | 23614898 |
SK-Mel-1 | - | Growth Inhibition Assay | - | IC50=37 nM | 23614898 |
SK-Mel-2 | - | Growth Inhibition Assay | - | IC50=34 nM | 23614898 |
SK-Mel-28 | - | Growth Inhibition Assay | - | IC50=85 nM | 23614898 |
SK-Mel-3 | - | Growth Inhibition Assay | - | IC50=118 nM | 23614898 |
SK-Mel-5 | - | Growth Inhibition Assay | - | IC50=66 nM | 23614898 |
SK-N-SH | - | Growth Inhibition Assay | - | IC50=150 nM | 23614898 |
SK-OV-3 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
SNB-19 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
SNB-75 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
SNU-1 | - | Growth Inhibition Assay | - | IC50=354 nM | 23614898 |
SNU-16 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
SU.86.86 | - | Growth Inhibition Assay | - | IC50=1001 nM | 23614898 |
SW-480 | - | Growth Inhibition Assay | - | IC50=165 nM | 23614898 |
SW-527 | - | Growth Inhibition Assay | - | IC50=121 nM | 23614898 |
SW-620 | - | Growth Inhibition Assay | - | IC50=104 nM | 23614898 |
SW-626 | - | Growth Inhibition Assay | - | IC50=33 nM | 23614898 |
TCC-SUP | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
TT | - | Growth Inhibition Assay | - | IC50=406 nM | 23614898 |
U-251 | - | Growth Inhibition Assay | - | IC50=1000 nM | 23614898 |
U373-MG | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
U87MG | - | Growth Inhibition Assay | - | IC50=2000 nM | 23614898 |
U-937 | - | Growth Inhibition Assay | - | IC50=3000 nM | 23614898 |
UACC-62 | - | Growth Inhibition Assay | - | IC50=30 nM | 23614898 |
UM-UC-3 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
WiDr | - | Growth Inhibition Assay | - | IC50=39 nM | 23614898 |
WM-266-4 | - | Growth Inhibition Assay | - | IC50=20 nM | 23614898 |
ZR-75-1 | - | Growth Inhibition Assay | - | IC50=3001 nM | 23614898 |
靶点 | Description | IC50 |
---|---|---|
ERK1 | IC50:4nM | |
ERK2 | IC50:1nM |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网