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CAS No.: 1158838-45-9
Synonyms: Aurora A Inhibitor I
Aurora an inhibitor I is a potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM in a cell-free assay. It is 1000-fold selective for Aurora A than Aurora B.
生物活性
实验方案
技术信息
CAS号 | 1158838-45-9 | 储存条件 |
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分子式 | C31H31ClFN7O2 | 运输 | 蓝冰 | |
分子量 | 588.08 | 别名 | Aurora A Inhibitor I |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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HCT116 cells | - | Proliferation assay | 4 days | Antiproliferative activity against human HCT116 cells after 4 days by celltiter assay, IC50=0.19 μM | 19402633 |
HT-29 cells | - | Proliferation assay | 4 days | Antiproliferative activity against human HT-29 cells after 4 days by celltiter assay, IC50=2.9 μM | 19402633 |
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