Thioperamide
98%
货号：A966063
同义名：
MR-12842
产品仅供科研
Thioperamide is a potent HRH4 antagonist and selective HRH3 antagonist capable of crossing the blood–brain barrier.
Thioperamide 化学结构
CAS号：106243-16-7
Thioperamide 3D分子结构
CAS号：106243-16-7
| 规格 |
价格 |
会员价
|
库存 |
数量 |
| {[ item.pr_size ]} |
{[ getRatePrice(item.pr_rmb, 1,1) ]}
{[ getRatePrice(item.pr_rmb_sale, 1,1) ]}
|
{[ getRatePrice(item.pr_rmb, 1,1) ]}
{[ getRatePrice(item.pr_rmb,item.pr_rate,1) ]}
|
{[ getRatePrice(item.pr_rmb, 1,1) ]} |
{[ getRatePrice(item.pr_rmb_sale, 1,1) ]}
{[ getRatePrice(item.pr_rmb,item.pr_rate,item.mem_rate) ]}
{[ getRatePrice(item.pr_rmb,1,item.mem_rate) ]}
|
现货 |
咨询
|
-
+
|
| Hydroxyzine 2HCl |
|
|
|
|
|
|
99+% |
| Cyclizine |
✔
|
|
|
|
|
|
97% |
| Loratadine |
+
|
|
|
|
|
|
98% |
| Desloratadine |
++
Histamine H1 receptor, IC50: 51 nM
|
|
|
|
|
|
98% |
| Doxylamine succinate |
✔
|
|
|
|
|
|
99% |
| Ebastine |
✔
|
|
|
|
|
|
98% |
| Tripelennamine HCl |
+
|
|
|
|
|
|
98% |
| Meclizine dihydrochloride |
✔
|
|
|
|
|
|
98% |
| Diphenhydramine HCl |
✔
|
|
|
|
|
|
99% |
| Alcaftadine |
++++
|
++
|
|
|
|
|
98%+ |
| Fexofenadine HCl |
++
Histamine H1 receptor, IC50: 246 nM
|
|
|
|
|
|
99%+ |
| Bilastine |
+++
H1 receptor, Ki: 44.15 nM
|
|
|
|
|
|
98% |
| Pemirolast potassium |
✔
|
|
|
|
|
|
98% |
| Bepotastine besilate |
+
Histamine H1 receptor, pIC50: 5.7
|
|
|
|
|
|
98% |
| Mizolastine |
+++
Histamine H1 receptor, IC50: 47 nM
|
|
|
|
|
|
98% |
| Brompheniramine maleate |
✔
|
|
|
|
|
|
98% |
| Carbinoxamine maleate salt |
✔
|
|
|
|
|
|
99+% |
| Clemastine fumarate |
++++
Histamine H1 receptor, IC50: 3 nM
|
|
|
|
|
|
98% |
| Ketotifen fumarate salt |
✔
|
|
|
|
|
|
95% |
| Rupatadine Fumarate |
++
Histamine H1 receptor, Ki: 102 nM
|
|
|
|
|
PAFR
|
98% |
| Famotidine |
|
✔
|
|
|
|
|
97% |
| Roxatidine Acetate HCl |
|
+
Histamine H2 receptor, IC50: 3.2 μM
|
|
|
|
|
98% |
| Lafutidine |
|
✔
|
|
|
|
|
99% |
| Cimetidine |
|
✔
|
|
|
|
|
98% |
| Nizatidine |
|
++++
Histamine H2 receptor, IC50: 0.9 nM
|
|
|
|
AChE
|
98% |
| Ranitidine |
|
✔
|
|
|
|
|
99% |
| Betahistine |
|
|
+
Histamine H3 receptor, IC50: 1.9 μM
|
|
|
|
98% |
| Ciproxifan maleate |
|
|
+++
Histamine H3 receptor, IC50: 9.2 nM
|
|
|
|
99%+ |
| S 38093 |
|
|
++
human H3 receptor, Ki: 1.2 μM
rat H3 receptor, Ki: 1.44 μM
|
|
|
|
99%+ |
| JNJ-7777120 |
|
|
|
++++
Histamine H4 receptor, Ki: 4.5 nM
|
|
|
98% |
| Azelastine HCl |
|
|
|
|
✔
|
|
98% |
| Epinastine HCl |
|
|
|
|
✔
|
|
98% |
| Levodropropizine |
|
|
|
|
✔
|
|
97% |
| Cyproheptadine hydrochloride |
|
|
|
|
✔
|
|
98% |
| Hesperetin |
|
|
|
|
✔
|
|
97% |
| Olopatadine HCl |
|
|
|
|
✔
|
|
98% |
| Mianserin hydrochloride |
|
|
|
|
✔
|
|
99+% |
| Buclizine 2HCl |
|
|
|
|
✔
|
|
97% |
| Latrepirdine 2HCl |
|
|
|
|
✔
|
GluR
|
98+% |
| Cetirizine 2HCl |
|
|
|
|
✔
|
|
98% |
|
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。
|
Thioperamide 生物活性
| 描述 |
Thioperamide is a potent HRH4 antagonist and selective HRH3 antagonist capable of crossing the blood–brain barrier. |
Thioperamide 参考文献
Thioperamide 实验方案
| 计算器 |
|
| 存储液制备 |
 |
1mg |
5mg |
10mg |
|
1 mM
5 mM
10 mM
|
3.42mL
0.68mL
0.34mL
|
17.10mL
3.42mL
1.71mL
|
34.19mL
6.84mL
3.42mL
|
Thioperamide 技术信息
搜索
