The formyl peptide receptors (FPR) belong to a class of G protein-coupled receptors involved in chemotaxis. In humans, there are three formyl peptide receptor isoforms, each encoded by a separate gene that are named FPR1, FPR2, and FPR3.
|CSN25759||WRW4||878557-55-2||WRW4 is a selective antagonist of formyl peptide receptor 2 (FPR2) signaling. It can inhibit WKYMVm binding to FPR2 with IC50 of 0.23 μM.|
|CSN26347||WKYMVM||187986-17-0||WKYMVM is a very potent agonist of formyl peptide receptor members FPR1/FPR2 (EC50 1 nM) and FPRL1/FPRL2 (75 pM and 3 nM, respectively).|
|CSN25764||WKYMVM||187986-11-4||WKYMVM is a selective agonist for the formyl peptide receptors FPR2 and FPR3.|
|CSN25761||TC-FPR 43||903895-98-7||TC-FPR 43 is a potent formyl peptide receptor 2 (FPR2) agonist with EC50 of 44 nM.|
|CSN25760||PBP 10||794466-43-6||PBP 10 is a selective antagonist of formyl peptide receptor 2 (FPR2). It can selectively inhibit FPR2-mediated NADPH oxidase activity but has no effect on FPR1 signaling in neutrophils.|
|CSN22896||Cyclosporin H||83602-39-5||Cyclosporin H is a potent and effective inhibitor of formyl peptide receptor (FPR) with Ki of 0.1 uM.|
|CSN25758||Boc-MLF||67247-12-5||Boc-MLF is an antagonist of formyl peptide receptor 1 (FPR1).|