Human Epidermal Growth Factor Receptor 2 | Protein Tyrosine Kinase/RTK| CSNpharm

HER2

HER2
第页，共 1 页

货号	产品名	CAS号	信息
CSN12170	Tyrphostin AG 879	148741-30-4	Tyrphostin AG 879 potently inhibits HER2/ErbB2 with IC50 of 1 μM, 100- and 500-fold higher selective to ErbB2 than PDGFR and EGFR.
CSN12702	CP-724714 (Random Configuration)	537705-08-1	CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, > 640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc in cell-free assays.
CSN10535	Canertinib 2HCl	289499-45-2	Canertinib 2HCl, an irreversible quinazoline-based HER family tyrosine kinase inhibitor, inhibits EGFR and ErbB2 with IC50 of 1.5 nM and 9.0 nM respectively. Phase II.