欢迎来到CSNpharm!产品仅用于科研!

400-920-2911 sales@csnpharm.cn

0

VEGFR

VEGFR

货号 产品名 CAS号 信息
CSN18068 ZM323881 HCl 193000-39-4 ZZZM 323881 HCl is a potent and selective VEGFR2 inhibitor with IC50 of < 2 nM, almost no activity on VEGFR1, PDGFRβ, FGFR1, EGFR and ErbB2.
CSN25326 Tyrphostin AG1433 168835-90-3 Tyrphostin AG1433 is a tyrosine kinases inhibitor and also a selective PDGFRβ and VEGFR-2 (Flk-1/KDR) inhibitor with IC50s of 5.0 μM and 9.3 μM, respectively.
CSN20516 SU5408 15966-93-5 SU5408 is a VEGFR2 kinase inhibitor with IC50 of 70 nM in murine.
CSN21274 SU5208 62540-08-3 SU5208 is an analogue of SU5025.
CSN20604 Su5205 3476-86-6 Su5205 is an inhibitor of VEGFR2.
CSN20550 SU 4312 5812-07-7 SU 4312 is a potent and selective inhibitor of VEGFR and PDGFR tyrosine kinases (IC50 values are 0.8 and 19.4 μM respectively), which is selective over EGFR and c-Src tyrosine kinases.
CSN17169 SKLB1002 1225451-84-2 SKLB1002 is a selective inhibitor of VEGFR2 with IC50 of 32 nM.
CSN17854 SAR131675 1433953-83-3 SAR131675 is selective inhibitor of VEGFR3 with IC50 and Ki of 23 nM, 12 nM, respectively.
CSN17331 Regorafenib Monohydrate 1019206-88-2 Regorafenib is a multi-target inhibitor. It can inhibit the activities of VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 and their IC50 values ​​range from 1.5 nM to 46 nM.
CSN18523 R1530 882531-87-5 R1530 is the multikinase inhibitor with potential antiangiogenesis and antineoplastic activities.
CSN23179 Vatalanib Succinate 212142-18-2 Potent VEGFR inhibitor; also aromatase inhibitor
CSN17192 Motesanib Diphosphate 857876-30-3 Motesanib diphosphate is ATP-competitive inhibitor of VEGFR1, VEGFR2 and VEGFR3 with IC50 of 2 nM, 3 nM and 6 nM, respectively. It also shows better inhibitory activity against c-Kit, PDGFR, and RET.
CSN27743 GW806742X   579515-63-2 GW806742X is an ATP mimetic MLKL inhibitor with Kd value of 9.3μM, and a VEGFR2 inhibitor with IC50 value of 2nM.
CSN27589 Donafenib 1130115-44-4 Donafenib, also known as CM-4307, is a multikinase inhibitor of Raf kinase and receptor tyrosine kinases with IC50 of 6 nM, 20 nM and 22 nM for Raf-1, B-Raf and VEGFR-3, respectively.
CSN26133 Decursin 5928-25-6 Decursin is a cumarin isolated from Radix peucedani that exhibits a number of physiological actions including anticancer, antibacterial, antinematodal and antioxidant. It inhibited proliferation and angiogenesis of endothelial cells to suppress diabetic retinopathy via VEGFR2.
CSN21898 Cediranib 288383-20-0 Cediranib is a multiple RTKs inhibitor with IC50 values of <0.001μM, 0.005μM, ≤0.003μM, 0.002μM and 0.005μM for VEGFR-2, VEGFR-1, VEGFR-3, c-Kit and PDGFR-β(measured kinase activity), respectively.
CSN21290 SU5204 186611-11-0 Analogue of SU5025
CSN23266 4,4-Bis(4-aminophenoxy)biphenyl 13080-85-8 4,4'-Bis(4-aminophenoxy)biphenyl is a potent Flk-1 (VEGFR2) inhibitor.
<< PREV 1 2 3 NEXT >>
联系
我们