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VEGFR
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN18068 | ZM323881 HCl | 193000-39-4 | ZZZM 323881 HCl is a potent and selective VEGFR2 inhibitor with IC50 of < 2 nM, almost no activity on VEGFR1, PDGFRβ, FGFR1, EGFR and ErbB2. |
| CSN25326 | Tyrphostin AG1433 | 168835-90-3 | Tyrphostin AG1433 is a tyrosine kinases inhibitor and also a selective PDGFRβ and VEGFR-2 (Flk-1/KDR) inhibitor with IC50s of 5.0 μM and 9.3 μM, respectively. |
| CSN20516 | SU5408 | 15966-93-5 | SU5408 is a VEGFR2 kinase inhibitor with IC50 of 70 nM in murine. |
| CSN21274 | SU5208 | 62540-08-3 | SU5208 is an analogue of SU5025. |
| CSN20604 | Su5205 | 3476-86-6 | Su5205 is an inhibitor of VEGFR2. |
| CSN20550 | SU 4312 | 5812-07-7 | SU 4312 is a potent and selective inhibitor of VEGFR and PDGFR tyrosine kinases (IC50 values are 0.8 and 19.4 μM respectively), which is selective over EGFR and c-Src tyrosine kinases. |
| CSN17169 | SKLB1002 | 1225451-84-2 | SKLB1002 is a selective inhibitor of VEGFR2 with IC50 of 32 nM. |
| CSN17854 | SAR131675 | 1433953-83-3 | SAR131675 is selective inhibitor of VEGFR3 with IC50 and Ki of 23 nM, 12 nM, respectively. |
| CSN17331 | Regorafenib Monohydrate | 1019206-88-2 | Regorafenib is a multi-target inhibitor. It can inhibit the activities of VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 and their IC50 values range from 1.5 nM to 46 nM. |
| CSN18523 | R1530 | 882531-87-5 | R1530 is the multikinase inhibitor with potential antiangiogenesis and antineoplastic activities. |
| CSN23179 | Vatalanib Succinate | 212142-18-2 | Potent VEGFR inhibitor; also aromatase inhibitor |
| CSN17192 | Motesanib Diphosphate | 857876-30-3 | Motesanib diphosphate is ATP-competitive inhibitor of VEGFR1, VEGFR2 and VEGFR3 with IC50 of 2 nM, 3 nM and 6 nM, respectively. It also shows better inhibitory activity against c-Kit, PDGFR, and RET. |
| CSN27743 | GW806742X | 579515-63-2 | GW806742X is an ATP mimetic MLKL inhibitor with Kd value of 9.3μM, and a VEGFR2 inhibitor with IC50 value of 2nM. |
| CSN27589 | Donafenib | 1130115-44-4 | Donafenib, also known as CM-4307, is a multikinase inhibitor of Raf kinase and receptor tyrosine kinases with IC50 of 6 nM, 20 nM and 22 nM for Raf-1, B-Raf and VEGFR-3, respectively. |
| CSN26133 | Decursin | 5928-25-6 | Decursin is a cumarin isolated from Radix peucedani that exhibits a number of physiological actions including anticancer, antibacterial, antinematodal and antioxidant. It inhibited proliferation and angiogenesis of endothelial cells to suppress diabetic retinopathy via VEGFR2. |
| CSN21898 | Cediranib | 288383-20-0 | Cediranib is a multiple RTKs inhibitor with IC50 values of <0.001μM, 0.005μM, ≤0.003μM, 0.002μM and 0.005μM for VEGFR-2, VEGFR-1, VEGFR-3, c-Kit and PDGFR-β(measured kinase activity), respectively. |
| CSN21290 | SU5204 | 186611-11-0 | Analogue of SU5025 |
| CSN23266 | 4,4-Bis(4-aminophenoxy)biphenyl | 13080-85-8 | 4,4'-Bis(4-aminophenoxy)biphenyl is a potent Flk-1 (VEGFR2) inhibitor. |
