GPR88

GPR88
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货号	产品名	CAS号	信息
CSN24070	RTI-13951-33	2244884-08-8	RTI-13951-33 is a potent, selective, and brain-penetrant GPR88 agonist, with an EC50 of 25 nM in GPR88 cAMP functional assay. RTI-13951-33 reduces alcohol reinforcement and intake behaviors in rats[1].
CSN21168	AR-13324 M1 metabolite	2309668-15-1	AR-13324 M1 metabolite is a hydrolysis metabolite of AR-13324 mesylate.
CSN21170	2-Pcca	1984859-71-3	2-PCCA is a racemic form of the GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells.
CSN21171	2-PCCA HCl	N/A	2-PCCA HCl is a GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells.
CSN21175	(1S,2S)-2-pcca	1609624-97-6	(1S,2S)-2-PCCA is a less active diastereomer of 2-PCCA. 2-PCCA is a GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells.
CSN21173	2-PCCA hydrochloride	1609563-70-3	(1S,2S)-2-PCCA HCl is a less active diastereomer of 2-PCCA. 2-PCCA is a GPR88 agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells.
CSN21172	(1R,2R)-2-PCCA	1287205-42-8	(1R,2R)-2-PCCA is a diastereomer of 2-PCCA, and acts as a potent GPR88 agonist, with an EC50 of 3 nM.
CSN21174	(1R,2R)-2-PCCA hydrochloride	1609563-71-4	(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 agonist, with an EC50 of 3 nM.