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P2Y Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN27554 | Uridine 5′-diphosphoglucose disodium salt | 28053-08-9 | Uridine 5′-diphosphoglucose disodium salt (UDP-D-Glucose disodium salt) is the precursor of glucose-containing oligosaccharides, polysaccharides, glycoproteins, and glycolipids in animal tissues and in some microorganisms. Uridine-5′-diphosphoglucose is an agonist of the P2Y14 receptor, a neuroimmune system GPCR. |
| CSN23371 | UDP disodium salt | 27821-45-0 | UDP disodium salt is an endogenous agonist of P2Y receptor which preferentially activates P2Y6. It exhibis antagonistic effect on the P2Y14 receptor. |
| CSN12090 | Ticlopidine | 55142-85-3 | Ticlopidine is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor. |
| CSN13719 | Ticlopidine HCl | 53885-35-1 | Ticlopidine HCl is an adenosine diphosphate (ADP) receptor inhibitor that against platelet aggregation with IC50 of ~2 μM. |
| CSN12826 | Ticagrelor | 274693-27-5 | Ticagrelor is a reversibly and oral active P2Y12 receptor antagonist with Ki of 2 nM, also inhibits CYP2C9 and midazolam 4-hydroxylation with IC50 of 10.5 μM and 8.2 μM respectively. |
| CSN12020 | Suramin Sodium | 129-46-4 | Suramin sodium salt is a polysulfonated naphthylurea that inhibits the binding of calmodulin to recognition sites on the ryanodine receptor-1 (IC50 = 4.9 μM), blocks G protein coupling to GPCRs, and non-selectively antagonizes P2 purinergic receptors(10-100 μM). |
| CSN17880 | Suramin | 145-63-1 | Suramin is a polysulfonated naphthylurea that inhibits the binding of calmodulin to recognition sites on the ryanodine receptor-1 (IC50 = 4.9 μM), blocks G protein coupling to GPCRs, and non-selectively antagonizes P2 purinergic receptors(10-100 μM). |
| CSN16171 | Prasugrel | 150322-43-3 | Prasugrel is a platelet inhibitor with IC50 value of 1.8 μM. |
| CSN12325 | Prasugren HCl | 389574-19-0 | Prasugrel HCl is a platelet inhibitor with IC50 value of 1.8 μM. |
| CSN13178 | N6-(4-Hydroxybenzyl)-adenosine | 110505-75-4 | N6-(4-Hydroxybenzyl)adenosine is an inhibitor of platelet aggregation induced in vitro by collagen and their activity range was demonstrated (IC50: 6.77-141 μM). |
| CSN11479 | MRS 2578 | 711019-86-2 | MRS2578 is a potent and selective P2Y6 nucleotide receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors. |
| CSN15727 | Clopidogrel | 113665-84-2 | Clopidogrel is a P2Y12 receptor blocker (IC50 = 100 nM). |
| CSN15854 | Clopidogrel Hydrogen Sulfate | 120202-66-6 | Clopidogrel Hydrogen Sulfate is the functional enantiomer of clopidogrel and a potent P2Y12 receptor antagonist. |