Insulin Receptor | Protein Tyrosine Kinase/RTK| CSNpharm

Insulin Receptor

Insulin Receptor
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货号	产品名	CAS号	信息
CSN12103	Tolazamide	1156-19-0	Tolazamide is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.
CSN12572	Rhoifolin	17306-46-6	Rhoifolin, a natural product isolated and purified from the leaves of Turpinia arguya Seem, hows monolithic proliferation inhibitory activities against Hela, A549 and MCF-7 cell lines, and may be beneficial for diabetic complications through their enhanced adiponectin secretion, tyrosine phosphorylation of insulin receptor-β and GLUT4. It was found to efficiently block the enzymatic activity of SARS-CoV 3CLpro.
CSN26520	Mps1-IN-1 dihydrochloride	1883548-93-3	Mps1-IN-1 dihydrochloride is a potent, selective and ATP-competitive Mps1 kinase inhibitor, with an IC50 and a Kd of 367 nM and 27 nM[1].
CSN18062	KU14R	189224-48-4	KU14R is an I(3)-R antagonist, which selectively blocks the insulin secretory response to imidazolines.
CSN23448	Cinnamic acid	621-82-9	Cinnamic acid can stimulate insulin secretion and improve glucose tolerance.
CSN15865	BMS-754807	1001350-96-4	BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.8 nM/1.7 nM, less potent to Met, Aurora A/B, TrkA/B and Ron, and shows little activity to Flt3, Lck, MK2, PKA, PKC etc.
CSN16463	BMS-536924	468740-43-4	BMS-536924 is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM.