Salt-inducible Kinases | Immunology/Inflammation| CSNpharm

SIK

SIK
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货号	产品名	CAS号	信息
CSN28431	YKL-05-099	1936529-65-5	YKL-05-099 is a selective SIK inhibitor with IC50 values of 10 nM, 40 nM and 30 nM for SIK1, SIK2 and SIK3, respectively.
CSN24297	YKL-06-061	2172617-15-9	YKL 06-061 is a pan-SIK inhibitor with IC50 values of 6.56nM, 1.77nM and 20.5nM for SIK1, SIK2 and SIK3, respectively.
CSN33249	WH-4-025	1876463-35-2	WH-4-025 is a SIK inhibitor extracted from WO2016023014 A2.
CSN14948	Pterosin B	34175-96-7	Pterosin B is a natural product isolated and purified from the aerial parts of Pteris semipinnata, is a salt-inducible kinase 3 (Sik3) pathway inhibitor, preventing chondrocyte hypertrophy and osteoarthritis in mice by inhibiting Sik3.
CSN25230	ODM-203	1430723-35-5	ODM-203 is a selective inhibitor of FGFR and VEGFR with IC50 values of 11, 16, 6, 35nM for recombinant FGFR1-4 and 26, 9, 5nM for VEGFR1-3, respectively.
CSN17882	HG-9-91-01	1456858-58-4	HG-9-91-01 is a potent and highly selective salt-inducible kinase (SIKs) inhibitor with IC50s of 0.92 nM, 6.6 nM and 9.6 nM for SIK1, SIK2 and SIK3 respectively.
CSN24497	ARN-3236	1613710-01-2	ARN-3236 is a selective SIK2 inhibitor with IC50 values of <1 nM, 21.63 nM and 6.63 nM for SIK2, SIK1 and SIK3, respectively.