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Androgen Receptor

Androgen Receptor

货号 产品名 CAS号 信息
CSN12743 RU 58841 154992-24-2 RU 58841 is a nonsteroidal antiandrogen for potential use as a topical treatment for androgen-dependent conditions including acne, pattern hair loss, and excessive hair growth.
CSN27360 Prochloraz 67747-09-5 Prochloraz is an imidazole antifungal that inhibits ergosterol biosynthesis via inhibition of the cytochrome P450-dependent 14α-demethylation of lanosterol, which results in disruption of the fungal cell membrane and cell death. Prochloraz inhibits human placenta microsomal aromatase in vitro (IC50 = 40 nM). Prochloraz also acts as an antagonist of the estrogen receptor (ER) and androgen receptor (AR) (IC50s = 25 μM and 4 μM, respectively) as well as activates the aryl hydrocarbon receptor (AhR; EC50 = 1 μM).
CSN17663 ORM-15341 1297537-33-7 ORM-15341 is a potent and full antagonist for human AR (hAR) with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells stably expressing full-length hAR and an androgen-responsive luciferase reporter gene construct.
CSN13442 Nomegestrol 58691-88-6 Nomegestrol is a steroidal progestin.
CSN16774 Nilutamide 63612-50-0 Nilutamide is a non-steroidal androgen receptor antagonist and also inhibits androgen biosynthesis in vitro.
CSN11374 Megestryl Acetate 595-33-5 Megestryl Acetate is a synthetic progesterone analog.
CSN10977 Hydroxyflutamide 52806-53-8 Hydroxyflutamide is a derivative of the synthetic steroid ethisterone, that suppresses the production of gonadotrophins, and has some weak androgenic effects.
CSN11169 Hydromadinone 16469-74-2 Hydromadinone, is a steroidal progestin of the 17α-hydroxyprogesterone group.
CSN16707 Flutamide 13311-84-7 Flutamide is a competitive non-steroidal antagonist of androgen receptor.
CSN10728 Cyproterone Acetate 427-51-0 Cyproterone Acetate is an antagonist and partial agonist of androgen receptor with IC50 value of 7.1 nM and EC50 value of 4μM.
CSN18075 Cortexolone 17 alpha-Propionate 19608-29-8 Cortexolone 17 alpha-propionate is a topical and peripherally selective androgen antagonist, which is used in treatment of acne and androgenic alopecia.
CSN16582 BMS-564929 627530-84-1 BMS-564929 is an androgen receptor (AR) agonist, binds to androgen receptor (AR) with a Ki of 2.11±0.16 nM.
CSN12437 Bicalutamide 90357-06-5 Bicalutamide is non-steroidal androgen receptor antagonist with IC50 value of 190 nM.
CSN17338 Dimethylcurcumin 52328-98-0 ASC-J9, an antitumor agent, suppresses castration-resistant prostate cancer growth via degradation of full-length and splice variant androgen receptors.
CSN13830 Apalutamide 956104-40-8 ARN-509 can compeitively and selectively inhibit androgen receptor with IC50 value of 16 nM.
CSN19392 3,3'-Diindolylmethane 1968-05-4 3,3'-Diindolylmethane is an AR structurally similar androgen receptor antagonist.
CSN23255 1-Phenylpentan-1-ol 583-03-9 1-Phenylpentan-1-ol is an intermediate for synthesis of β-amino-carbonyl-based androgen receptor antagonist.
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