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Dopamine Receptor

Dopamine Receptor

货号 产品名 CAS号 信息
CSN23250 Trimethobenzamide HCl 554-92-7 Trimethobenzamide HCl is a dopamine D2 receptor antagonist and antiemetic drug.
CSN12086 Tiamenidine 31428-61-2 Thioridazine is an antipsychotic drug, used in the treatment of schizophrenia and psychosis, shows D4 selectivity or serotonin antagonism.
CSN21847 Sultopride 53583-79-2 Sultopride is a selective antagonist of dopamine D2 receptor.
CSN22118 Sultopride HCl 23694-17-9 Sultopride HCl is a selective antagonist of dopamine D2 receptor
CSN11918 Sertindole 106516-24-9 Sertindole, a neuroleptic, is one of the antipsychotic medications available, with a high affinity for dopamine D2, serotonin 5-HT2A, 5-HT2C, and α1-adrenergic receptors.
CSN23655 Ro 10-5824 2HCl 189744-94-3 Ro 10-5824 2HCl is an agonist of dopamine D4 receptor with Ki of 5.2 nM.
CSN23271 PD 168077 Maleate 630117-19-0 PD 168077 maleate is an agonist of D4 dopamine receptor with Ki of 8.7 nM. It can induce synaptic translocation of CaMK II to postsynaptic sites in cultured prefrontal cortical neurons.
CSN18173 Pardoprunox HCl 269718-83-4 Pardoprunox HCl is a partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist.
CSN25427 Melanocyte-stimulating hormone release inhibiting factor 2002-44-0 Oxytocin C-terminal tripeptide is shown to be effective in treating human depression with greater efficacy and faster onset of action than traditional anti-depressants. Also, it is used in the synthesis of novel analogs to be tested for their ability to enhance the binding of -N-propylnorapomorphine to short isoform of human dopamine D2 receptors.
CSN11617 Oroxylin A 480-11-5 Oroxylin A shows inhibition of the dopamine reuptake and allosteric modulation of GABAA receptor. It is a natural active flavonoid isolated from scutellaria baicalensis and oroxylum indicum.
CSN11590 Nuciferine 475-83-2 Nuciferine is naturally occuring alkaloid found in the plants Nymphaea caerulea and Nelumbo nucifera as a potent inverse agonist at human 5-HT7 receptor.
CSN19863 NGB 2904 HCl 189061-11-8 NGB 2904 is a potent and selective dopamine D3 receptor antagonist (Ki values are 1.4, 217, 223, 642, > 5000, > 10000 and > 10000 nM for D3, D2, 5-HT2, α1, D4, D1 and D5 receptors respectively).
CSN41416 MPP+ iodide 36913-39-0 MPP+ iodide is a metabolite of dopaminergic neurotoxin MPTP.
CSN23832 Mesoridazine Besylate 32672-69-8 Mesoridazine besylate is a phenothiazine dopamine receptor anatagonist. Mesoridazine besylate is described to demonstrate inhibition for D2DR and D4DR. It has a high affinity for dopamine D4 receptor. Mesoridazine besylate is an antipsychotic agent.
CSN25316 L-745870 158985-00-3 L-745870 is a high-affinity, selective and orally active human dopamine D4 receptor antagonist with a Ki of 0.43 nM and excellent brain penetration.
CSN27239 Fluphenazine 69-23-8 Fluphenazine is a typical antipsychotic used for symptomatic management of psychosis in patients with schizophrenia.
CSN22033 Dixyrazine 2470-73-7 Dixyrazine, a phenothiazine derivative, can prevent brain oedema induced by intracarotid injection of protamine sulphate.
CSN19084 CGP-25454A 104391-26-6 CGP 25454A is a selective presynaptic dopamine autoreceptor antagonist.
CSN20529 BP897 314776-92-6 BP897 is a partially selective dopamine D3 receptor agonist (Ki = 0.92 nM) that developed for the study of cocaine addiction.
CSN21450 Abaperidone 183849-43-6 Abaperidone is an antagonist of 5-HT2A receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM respectively.
CSN24069 A-381393 726174-00-1 A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM)[1].
CSN22323 (+)-Dihydrexidine HCl 158704-02-0 (+)-Dihydrexidine HCl is a dopamine D1 receptor agonist with an EC50 of 72± 21 nM.
CSN25685 (+)-AJ 76 HCl 85378-82-1 (+)-AJ 76 hydrochloride is an antagonist of dopamine receptor with preferential action at presynaptic receptors (pKi values are 6.95, 6.67, 6.37, 6.21 and 6.07 at hD3, D4, hD2S, hD2L and rD2 receptors respectively).
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