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GNRH Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN22066 | Sufugolix | 308831-61-0 | Sufugolix is a highly potent and orally available luteinizing hormone-releasing hormone (LHRH) receptor antagonist with IC50 of 0.1 nM |
| CSN17262 | Relugolix | 737789-87-6 | Relugolix is a non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum. It possesses higher affinity and potent antagonistic activity compared with TAK-013. |
| CSN11279 | Lecirelin | 61012-19-9 | Lecirelin is a synthetic GnRH analogue which showed a great efficacy in the treatment of bovine ovarian follicular cysts. |
| CSN11007 | Fertirelin | 38234-21-8 | Fertirelin is an analog of gonadotropin-releasing hormone agonist . |
| CSN22393 | Elagolix sodium | 832720-36-2 | Elagolix sodium is an antagonist of human GnRH receptor (GnRHR) with IC50 and Ki of 0.25 nM and 3.7 nM, respectively. |
| CSN18452 | (R)-Elagolix | 834153-87-6 | Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). |
| CSN18109 | Degarelix | 214766-78-6 | Degarelix is a gonadotrophin-releasing hormone (GnRH) antagonist for the first-line treatment of androgen-dependent advanced prostate cancer. |
| CSN22891 | Cetrorelix diacetate | 130143-01-0 | Cetrorelix acetate(1:2) is the acetate form of cetrorelix which is an antagonist of gonadotropin-releasing hormone (GnRH) used in inhibiting premature luteinizing hormone surges. |
| CSN18990 | Cetrorelix Acetate | 145672-81-7 | Cetrorelix acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with IC50 of 1.21 nM. |
| CSN11805 | Alarelin Acetate | 79561-22-1 | Alarelin acetate is a synthetic agonist of GnRH. |
| CSN25815 | 5-((3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl)methyl)-N-(2,4,6-trimethoxyphenyl)furan-2-carboxamide | 263847-55-8 | AG 045572 is a selective antagonist of gonadotropin-releasing hormone (GnRH) receptor with Ki value of 6.0 nM. |
| CSN20400 | Zoptarelin doxorubicin | 139570-93-7 | AEZS-108 is a peptide agonist of the gonadotropin releasing hormone-1 receptor (GnRH-1R). |
| CSN10194 | Abarelix | 183552-38-7 | Abarelix is a potent gonadotrophin-releasing hormone (GnRH) antagonist, used for prostate cancer treatment. |
