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Sigma Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN21074 | Blarcamesine hydrochloride | 195615-84-0 | σ1 agonist (IC50 = 860 nM); also displays affinity for muscarinic M1-M4 receptors (Ki values < 500 nM), but not for σ2 receptors. Exhibits neuroprotective effects, prevents tau hyperphosphorylation, and attenuates scopolamine- and (+)-MK 801-induced learning deficits in a mouse model of amyloid toxicity. |
| CSN16114 | Siramesine | 147817-50-3 | Siramesine is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potent anticancer activity in vivo. |
| CSN16281 | Siramesine hydrochloride | 224177-60-0 | Siramesine HCl is an agonist of sigma-2 receptor which can trigger cell death and exhibit anticancer activity. |
| CSN17988 | Cutamesine | 165377-43-5 | SA4503 is an agonist of opioid sigma1 receptor (σ1R) with IC50 of 17.4 nM. |
| CSN11878 | Cutamesine dihydrochloride | 165377-44-6 | SA4503 2HCl is the 2HCl form of SA4503 which is an agonist of opioid sigma1 receptor (σ1R) with IC50 of 17.4 nM. |
| CSN16936 | S1RA | 878141-96-9 | S1RA is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM) antagonist, showed good selectivity against σ2R (Ki > 1000 nM). |
| CSN17645 | S1RA hydrochloride | 1265917-14-3 | S1RA HCl is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM) antagonist, showed good selectivity against σ2R (Ki > 1000 nM). |
| CSN33114 | Roluperidone | 359625-79-9 | Roluperidone is a 5-HT2A and sigma 2 receptor antagonist. |
| CSN21927 | Pridopidine | 346688-38-8 | Pridopidine exhibits high affinity towards sigma 1 receptor (S1R) (Ki = 70-80 nM) which can counteract the effects of excessive or insufficient dopaminergic transmission and it can used as a dopamine (DA) stabilizer. |
| CSN18418 | PRE-084 hydrochloride | 75136-54-8 | PRE-084 HCl is a high affinity, selective σ1 agonist, has an IC50 of 44 nM in the sigma receptor assay. |
| CSN26761 | PD 144418 oxalate | 1794760-28-3 | PD-144418 Oxalate is a novel selective sigma ligand. |
| CSN26378 | Ditolylguanidine | 97-39-2 | Ditolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor)[1]. |
| CSN33115 | CYR-101 HCl 2H2O | 1937215-88-7 | CYR-101 hydrochloride dihydrate is a 5-HT2A and sigma 2 receptor antagonist. |
| CSN26439 | BD1063 | 150208-28-9 | BD1063 is a selective sigma receptor antagonist, with a Ki of 9 ± 1 nM for the sigma-1 receptor. |
| CSN24789 | BD1063 dhydrochloride | 206996-13-6 | BD1063 dhydrochloride is a potent and selective sigma 1 receptor antagonist. |
| CSN16267 | BD-1047 dihydrobromide | 138356-21-5 | BD-1047 dihydrobromide is a selective functional antagonist of sigma receptors, shows antipsychotic activity in animal models predictive of efficacy in schizophrenia. |
| CSN17929 | 4-IBP | 155798-08-6 | 4-IBP is selective σ1 agonist with Ki of 1.7 nM and 25.2 nM for σ2 receptor. |
| CSN38573 | DuP 734 | 135135-87-4 | |
| CSN40713 | OPC-14523 free base | 145969-30-8 | |
| CSN34043 | OPC-14523 hydrochloride | 145969-31-9 | |
| CSN36657 | L-745870 hydrochloride | 1173023-36-3 | |
| CSN37126 | L-745870 trihydrochloride | 866021-03-6 |
