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Sigma Receptor

Sigma Receptor

货号 产品名 CAS号 信息
CSN21074 Blarcamesine hydrochloride 195615-84-0 σ1 agonist (IC50 = 860 nM); also displays affinity for muscarinic M1-M4 receptors (Ki values < 500 nM), but not for σ2 receptors. Exhibits neuroprotective effects, prevents tau hyperphosphorylation, and attenuates scopolamine- and (+)-MK 801-induced learning deficits in a mouse model of amyloid toxicity.
CSN16114 Siramesine 147817-50-3 Siramesine is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potent anticancer activity in vivo.
CSN16281 Siramesine hydrochloride 224177-60-0 Siramesine HCl is an agonist of sigma-2 receptor which can trigger cell death and exhibit anticancer activity.
CSN17988 Cutamesine 165377-43-5 SA4503 is an agonist of opioid sigma1 receptor (σ1R) with IC50 of 17.4 nM.
CSN11878 Cutamesine dihydrochloride 165377-44-6 SA4503 2HCl is the 2HCl form of SA4503 which is an agonist of opioid sigma1 receptor (σ1R) with IC50 of 17.4 nM.
CSN16936 S1RA 878141-96-9 S1RA is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM) antagonist, showed good selectivity against σ2R (Ki > 1000 nM).
CSN17645 S1RA hydrochloride 1265917-14-3 S1RA HCl is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM) antagonist, showed good selectivity against σ2R (Ki > 1000 nM).
CSN33114 Roluperidone 359625-79-9 Roluperidone is a 5-HT2A and sigma 2 receptor antagonist.
CSN21927 Pridopidine 346688-38-8 Pridopidine exhibits high affinity towards sigma 1 receptor (S1R) (Ki = 70-80 nM) which can counteract the effects of excessive or insufficient dopaminergic transmission and it can used as a dopamine (DA) stabilizer.
CSN18418 PRE-084 hydrochloride 75136-54-8 PRE-084 HCl is a high affinity, selective σ1 agonist, has an IC50 of 44 nM in the sigma receptor assay.
CSN26761 PD 144418 oxalate 1794760-28-3 PD-144418 Oxalate is a novel selective sigma ligand.
CSN26378 Ditolylguanidine 97-39-2 Ditolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor)[1].
CSN33115 CYR-101 HCl 2H2O 1937215-88-7 CYR-101 hydrochloride dihydrate is a 5-HT2A and sigma 2 receptor antagonist.
CSN26439 BD1063 150208-28-9 BD1063 is a selective sigma receptor antagonist, with a Ki of 9 ± 1 nM for the sigma-1 receptor.
CSN24789 BD1063 dhydrochloride 206996-13-6 BD1063 dhydrochloride is a potent and selective sigma 1 receptor antagonist.
CSN16267 BD-1047 dihydrobromide 138356-21-5 BD-1047 dihydrobromide is a selective functional antagonist of sigma receptors, shows antipsychotic activity in animal models predictive of efficacy in schizophrenia.
CSN17929 4-IBP 155798-08-6 4-IBP is selective σ1 agonist with Ki of 1.7 nM and 25.2 nM for σ2 receptor.
CSN38573 DuP 734 135135-87-4
CSN40713 OPC-14523 free base 145969-30-8
CSN34043 OPC-14523 hydrochloride 145969-31-9
CSN36657 L-745870 hydrochloride 1173023-36-3
CSN37126 L-745870 trihydrochloride 866021-03-6
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