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Prostaglandin Receptor

Prostaglandin Receptor

货号 产品名 CAS号 信息
CSN23731 U-46619 56985-40-1 U 46619, PGH2 (TXA2) analog that is a potent and stable thromboxane A2 (TP) receptor agonist with EC50 of 0.035 μM.
CSN17319 Treprostinil Sodium 289480-64-4 Treprostinil sodium is a potent DP1 and EP2 agonist with EC50 values of 0.6±0.1 and 6.2±1.2 nM, respectively.
CSN21858 Tiaprost 71116-82-0 Tiaprost is a prostaglandin F2 alpha analogue as an estrus-synchronizing agent.
CSN17989 Terutroban 165538-40-9 Terutroban is a thromboxane/prostaglandin endoperoxide receptor antagonist.
CSN21854 Terbogrel 149979-74-8 Terbogrel is an orally available thromboxane A2 receptor antagonist and a thromboxane A2 synthase inhibitor with both IC50s of about 10 nM.
CSN18419 Taprenepag 752187-80-7 Taprenepag is an agonist of prostaglandin E2 receptor with EC50 of 2.8 nM with hypotensive activity.
CSN12962 Tafluprost 209860-87-7 Tafluprost is an anti-glaucoma prostaglandin (PG) analog.
CSN25726 SC 51089 146033-02-5 SC-51089, also known as CID132748, is an antagonist of PGE2 and selective for the EP1 receptor subtype with antinociceptive activity.
CSN25725 SC 51322 146032-79-3 SC 51322 is an antagonist of EP1 prostanoid receptor with Ki of 13.8 nM.
CSN23716 Treprostinil 81846-19-7 Rumodolinl, a analog of prostacyclin, is an agonist of IP receptor that used clinically to treat pulmonary arterial hypertension. It is a vasodilator with antithrombotic and anti-inflammatory properties.
CSN21394 RO1138452 221529-58-4 RO1138452 is a selective antagonist of prostacyclin (IP) receptor with pKi of 9.3 ± 0.1 in human platelets.
CSN20322 Prostaglandin D2 41598-07-6 Prostaglandin D2 is the major eicosanoid product of mast cells and is released in large quantities during allergic and asthmatic anaphylaxis.
CSN23451 p-Hydroxy-Cinnamic Acid 7400-08-0 p-Hydroxy-cinnamic acid is the isomer of cinnamic acid with anti-mutagenic and anti-tumor activities.
CSN18259 ONO-AE3-208 402473-54-5 ONO-AE3-208 is an antagonist of EP4 with Ki of 1.3 nM and exhibits suppression the invasion and metastasis of prostate cancer cells.
CSN25724 ONO 8130 459841-96-4 ONO 8130 is an antagonist of EP1 receptor.
CSN11531 Nedocromil 69049-73-6 Nedocromil is an inhaled anti-inflammatory agent for the preventive management of asthma.
CSN18339 Laropiprant 571170-77-9 Laropiprant is a potent, selective DP1 receptor antagonist with Ki value of 0.57 nM and exhibits > 1,000 fold selectivity over DP2 receptor (Ki=0.75 μM).
CSN20466 L-798,106 244101-02-8 L-798106 is a potent and highly selective prostanoid EP3 receptor antagonist (Ki values are 0.3, 916, > 5000 and > 5000 nM at EP3, EP4, EP1 and EP2, respectively), and it can attenuate sulprostone-induced inhibition of EFS-evoked twitch and contractile responses in vivo.
CSN25731 L-161,982 147776-06-5 L-161,982 is a potent EP4 receptor antagonist with Ki value of 0.024 μM.
CSN22113 Ifetroban 143443-90-7 Ifetroban is a long-acting thromboxane A2 receptor antagonist, with antiplatelet activity.
CSN18130 Evatanepag 223488-57-1 Evatanepag is an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation with EC50 of 0.3 nM.
CSN20029 Esuberaprost Sodium 88475-69-8 Esuberaprost is a potential substance for treating pulmonary arterial hypertension (PAH).
CSN20026 Esuberaprost 94132-88-4 Esuberaprost is a potential substance for treating pulmonary arterial hypertension (PAH).
CSN26370 Epoprostenol sodium 61849-14-7 Epoprostenol sodium, a potent agonist at IP prostanoid receptors, the synthetic form of the natural prostaglandin derivative prostacyclin (prostaglandin I2), is registered worldwide for the treatment of Pulmonary arterial hypertension (PAH)[1]. Epoprostenol sodium is used in pulmonary hypertension and transplantation as a potent inhibitor of platelet aggregation[2].
CSN25728 DG 041 861238-35-9 DG-041 is a potent and selective antagonist of prostanoid EP3 receptor with IC50 of 4.6 nM.
CSN21985 Decursinol angelate 130848-06-5 Decursinol angelate (DA) blocks PGE2-induced activation of the EP2 receptor signaling pathway, including the activation of PKA and the phosphorylation of CREB.
CSN25453 Cloprostenol Sodium Salt 55028-72-3 Cloprostenol sodium salt (ICI 80996 sodium salt) is a potent synthetic prostaglandin analogue, acts as a luteolytic agent, and is a PGF2α receptor agonist.
CSN26158 (+)-Cloprostenol (sodium salt) 62561-03-9 Cloprostenol is a PGF2 α analogue, working as an FP receptor agonist.
CSN22111 Carbacyclin 69552-46-1 Carbacyclin is a PGI2 analogue, acts as a prostacyclin (PGI2) receptor agonist and vasodilator, and potently inhibits platelet aggregation.
CSN21535 BW245C 72814-32-5 BW 245C is a selective agonist for the DP1 receptor.
CSN17217 Bimatoprost 155206-00-1 Bimatoprost, a analog of prostaglandin, can control the progression of glaucoma and ocular hypertension.
CSN19378 Alprostadil 745-65-3 Alprostadil is an analog of prostaglandin which is prostaglandin E1 agonist with vasodilatory properties and can be used to treat erectile dysfunction.
CSN21466 Aligeron 70713-45-0 Aligeron is a non-selective antagonist of prostaglandin (PG) with vasodilatory properties.  
CSN25755 (+)-Fluprostenol 54276-17-4 (+)-Fluprostenol is an agonist of prostaglandin F2α (FP) receptor with Ki of 49.9 nM and EC50 of 2.4 nM.
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